Optimized labeling of NOTA-conjugated octreotide with F-18

Tumor Biology

Volumn 33, Issue 2, 2012, Pages 427-434

  Laverman, Peter ^a   D'Souza, Christopher A ^b   Eek, Annemarie ^a   McBride, William J ^b   Sharkey, Robert M ^c   Oyen, Wim J G ^a   Goldenberg, David M ^c   Boerman, Otto C ^a  

^a RADBOUD UNIVERSITY MEDICAL CENTER   (Netherlands)

^b IMMUNOMEDICS INC   (United States)

^c CENTER FOR MOLECULAR MEDICINE AND IMMUNOLOGY   (United States)

Author keywords

Aluminum fluoride; NOTA; Octreotide; Peptide; PET; Radiofluorination

Indexed keywords

1,4,7 TRIAZACYCLONONANE 1,4,7 TRIACETIC ACID CONJUGATED OCTREOTIDE F 18; ACETONITRILE; ALCOHOL; ALUMINUM FLUORIDE; BUFFER; IMP 466; PENTETREOTIDE; PEPTIDE; RADIOISOTOPE; UNCLASSIFIED DRUG; 1,4,7 TRIAZACYCLONONANE 1,4,7 TRIACETIC ACID; 1,4,7-TRIAZACYCLONONANE-N,N',N''-TRIACETIC ACID; ALUMINUM DERIVATIVE; ANTINEOPLASTIC HORMONE AGONISTS AND ANTAGONISTS; CHELATING AGENT; FLUORIDE; FLUORINE; HETEROCYCLIC COMPOUND; ION; OCTREOTIDE; SOLVENT;

ANIMAL CELL; ANIMAL EXPERIMENT; ANIMAL MODEL; ANIMAL TISSUE; ARTICLE; COMPUTER ASSISTED EMISSION TOMOGRAPHY; CONTROLLED STUDY; DRUG BLOOD LEVEL; DRUG BONE LEVEL; DRUG DISTRIBUTION; DRUG PURIFICATION; DRUG STABILITY; DRUG TUMOR LEVEL; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; IC 50; IN VITRO STUDY; IN VIVO STUDY; IONIC STRENGTH; ISOTOPE LABELING; MALE; MICRO-COMPUTED TOMOGRAPHY; MOUSE; NONHUMAN; PANCREAS TUMOR; PRIORITY JOURNAL; QUANTITATIVE ANALYSIS; RADIOCHEMISTRY; RAT; RECEPTOR AFFINITY; TEMPERATURE; ANIMAL; BAGG ALBINO MOUSE; CHEMISTRY; COMPUTER ASSISTED TOMOGRAPHY; HUMAN; METHODOLOGY; NUDE MOUSE; POSITRON EMISSION TOMOGRAPHY; TUMOR CELL LINE;

ALUMINUM COMPOUNDS; ANIMALS; ANTINEOPLASTIC AGENTS, HORMONAL; CELL LINE, TUMOR; CHELATING AGENTS; CHROMATOGRAPHY, HIGH PRESSURE LIQUID; FLUORIDES; FLUORINE RADIOISOTOPES; HETEROCYCLIC COMPOUNDS; HUMANS; INHIBITORY CONCENTRATION 50; IONS; MALE; MICE; MICE, INBRED BALB C; MICE, NUDE; OCTREOTIDE; POSITRON-EMISSION TOMOGRAPHY; RATS; SOLVENTS; TEMPERATURE; TOMOGRAPHY, X-RAY COMPUTED;

EID: 84860271819     PISSN: 10104283     EISSN: 14230380     Source Type: Journal    
DOI: 10.1007/s13277-011-0250-x     Document Type: Article

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