18F-Fluoroglucosylation of peptides, exemplified on cyclo(RGDfK)

European Journal of Nuclear Medicine and Molecular Imaging

Volumn 36, Issue 9, 2009, Pages 1469-1474

  Hultsch, Christina ^a   Schottelius, Margret ^a   Auernheimer, Jörg ^a   Alke, Andrea ^a   Wester, Hans Jürgen ^a  

^a TECHNICAL UNIVERSITY OF MUNICH   (Germany)

Author keywords

18F; Aminooxy; FDG; Fluoroglucosylation; Oxime; Peptide; PET

Indexed keywords

FLUORINE 18; FLUORODEOXYGLUCOSE F 18; PEPTIDE;

ARTICLE; CONTROLLED STUDY; DRUG DISTRIBUTION; GLYCOSYLATION; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; IN VIVO STUDY; ISOTOPE LABELING; MELANOMA; MOUSE; NONHUMAN;

ANIMALS; FLUORODEOXYGLUCOSE F18; GLYCOSYLATION; MELANOMA, EXPERIMENTAL; MICE; MICE, NUDE; NEOPLASM TRANSPLANTATION; PEPTIDES, CYCLIC; POSITRON-EMISSION TOMOGRAPHY; RADIOPHARMACEUTICALS; TISSUE DISTRIBUTION;

EID: 68949220252     PISSN: 16197070     EISSN: None     Source Type: Journal    
DOI: 10.1007/s00259-009-1122-0     Document Type: Article

References (9)

1. AJ Beer M Schwaiger 2008 Imaging of integrin alphavbeta3 expression Cancer Metastasis Rev 27 4 631 644 10.1007/s10555-008-9158-3
2. R Haubner B Kuhnast C Mang WA Weber H Kessler HJ Wester, et al 2004 [18F]Galacto-RGD: synthesis, radiolabeling, metabolic stability, and radiation dose estimates Bioconjug Chem 15 61 69 10.1021/bc034170n
3. T Poethko M Schottelius G Thumshirn U Hersel M Herz G Henriksen, et al 2004 Two-step methodology for high-yield routine radiohalogenation of peptides: (18)F-labeled RGD and octreotide analogs J Nucl Med 45 892 902
4. O Prante J Einsiedel R Haubner P Gmeiner HJ Wester T Kuwert, et al 2007 3,4,6-Tri-O-acetyl-2-deoxy-2-[18F]fluoroglucopyranosyl phenylthiosulfonate: a thiol-reactive agent for the chemoselective 18F-glycosylation of peptides Bioconjug Chem 18 254 262 10.1021/bc060340v
5. F Wuest M Berndt R Bergmann J van den Hoff J Pietzsch 2008 Synthesis and application of [18F]FDG-maleimidehexyloxime ([18F]FDG-MHO): a [18F]FDG-based prosthetic group for the chemoselective 18F-labeling of peptides and proteins. Bioconjug Chem 19 1202 1210 10.1021/bc8000112
6. HH Wasserman GD Berger KR Cho 1982 Transamidation reactions using β-lactams. The synthesis of homaline Tetrahedron Lett 23 465 468 10.1016/S0040-4039(00) 86862-8
7. HJ Wester BW Schoultz C Hultsch G Henriksen 2009 Fast and repetitive in-capillary production of [18F]FDG Eur J Nucl Med Mol Imaging 36 653 658
8. R Tomatis M Marastoni G Balboni R Guerrini A Capasso L Sorrentino, et al 1997 Synthesis and pharmacological activity of deltorphin and demorphin-related glycopeptides J Med Chem 40 2948 2952 10.1021/jm970119r
9. T Mizuma N Sakai S Awazu 1994 Na+-dependent transport of aminopeptidase-resistant sugar-coupled tripeptides in rat intestine Biochem Biophys Res Commun 203 1412 1416 10.1006/bbrc.1994.2342