Positive and negative allosteric modulators promote biased signaling at the calcium-sensing receptor

Endocrinology

Volumn 153, Issue 3, 2012, Pages 1232-1241

  Davey, Anna E ^a   Leach, Katie ^a   Valant, Celine ^a   Conigrave, Arthur D ^b   Sexton, Patrick M ^a   Christopoulos, Arthur ^a  

^a MONASH UNIVERSITY   (Australia)

^b UNIVERSITY OF SYDNEY   (Australia)

Author keywords

[No Author keywords available]

Indexed keywords

2 CHLORO 6 [3 [1,1 DIMETHYL 2 (2 NAPHTHYL)ETHYLAMINO] 2 HYDROXYPROPOXY]BENZONITRILE; CALCILYTIC; CALCIMIMETIC AGENT; CALCIUM ION; CALCIUM SENSING RECEPTOR; CINACALCET; MITOGEN ACTIVATED PROTEIN KINASE 1; MITOGEN ACTIVATED PROTEIN KINASE 3; TECALCET; UNCLASSIFIED DRUG;

ALLOSTERISM; ARTICLE; CELL LINE; CELL MEMBRANE; DRUG EFFECT; ENZYME PHOSPHORYLATION; HUMAN; HUMAN CELL; KIDNEY CELL; PRIORITY JOURNAL;

ALLOSTERIC SITE; ANILINE COMPOUNDS; CALCIMIMETIC AGENTS; CALCIUM; CELL MEMBRANE; HEK293 CELLS; HUMANS; HYPERPARATHYROIDISM; KIDNEY DISEASES; KIDNEY FAILURE, CHRONIC; LIGANDS; NAPHTHALENES; PHOSPHORYLATION; RECEPTORS, CALCIUM-SENSING; SIGNAL TRANSDUCTION; TREATMENT OUTCOME;

EID: 84857386424     PISSN: 00137227     EISSN: 19457170     Source Type: Journal    
DOI: 10.1210/en.2011-1426     Document Type: Article

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