Synthesis and biological evaluation of some thiazolidinones as antimicrobial agents

European Journal of Medicinal Chemistry

Volumn 48, Issue , 2012, Pages 354-362

  Patel, Divyesh ^a   Kumari, Premlata ^a   Patel, Navin ^b  

^a SARDAR VALLABHBHAI NATIONAL INSTITUTE OF TECHNOLOGY   (India)

^b VEER NARMAD SOUTH GUJARAT UNIVERSITY   (India)

Author keywords

Antibacterial activity; Antifungal activity; Structure activity relationship; Thiazolidinones

Indexed keywords

2 [3 [4 [4 DIMETHYLAMINO 6 (1 METHYL 2 OXO 1,2 DIHYDRO QUINOLIN 4 YLOXY)[1,3,5]TRIAZIN 2B YLAMINO]PHENYL] 5 (4 ETHYLPIPERAZIN 1 YLMETHYL) 4 OXOTHIAZOLIDIN 2 YL]BENZOIC ACID; 4 [3 [4 [4 DIMETHYLAMINO 6 (1 METHYL 2 OXO 1,2 DIHYDRO QUINOLIN 4 YLOXY)[1,3,5]TRIAZIN 2B YLAMINO]PHENYL] 5 (4 ETHYLPIPERAZIN 1 YLMETHYL) 4 OXOTHIAZOLIDIN 2 YL]BENZOIC ACID; 4 [4 [4 [2 (2 BROMOPHENYL) 5 (4 ETHYLPIPERAZIN 1 YLMETHYL) 4 OXOTHIAZOLIDIN 3 YL]PHENYLAMIO] 6 DIMETHYLAMINO[1,3,5]TRIAZIN 2 YLOXY] 1 METHYL 1H QUINOLIN 2 ONE; 4 [4 [4 [2 (2,3 DIHYDROXYPHENYL) 5 (4 ETHYLPIPERAZIN 1 YLMETHYL) 4 OXOTHIAZOLIDIN 3 YL]PHENYLAMIO] 6 DIMETHYLAMINO[1,3,5]TRIAZIN 2 YLOXY] 1 METHYL 1H QUINOLIN 2 ONE; 4 [4 [4 [2 (2,4 DICHLOROPHENYL) 5 (4 ETHYLPIPERAZIN 1 YLMETHYL) 4 OXOTHIAZOLIDIN 3 YL]PHENYLAMIO] 6 DIMETHYLAMINO[1,3,5]TRIAZIN 2 YLOXY] 1 METHYL 1H QUINOLIN 2 ONE; 4 [4 [4 [2 (2,4 DIHYDROXYPHENYL) 5 (4 ETHYLPIPERAZIN 1 YLMETHYL) 4 OXOTHIAZOLIDIN 3 YL]PHENYLAMIO] 6 DIMETHYLAMINO[1,3,5]TRIAZIN 2 YLOXY] 1 METHYL 1H QUINOLIN 2 ONE; 4 [4 [4 [2 (3,4 DICHLOROPHENYL) 5 (4 ETHYLPIPERAZIN 1 YLMETHYL) 4 OXOTHIAZOLIDIN 3 YL]PHENYLAMIO] 6 DIMETHYLAMINO[1,3,5]TRIAZIN 2 YLOXY] 1 METHYL 1H QUINOLIN 2 ONE; 4 [4 [4 [2 (3,4 DIMETHOXYPHENYL) 5 (4 ETHYLPIPERAZIN 1 YLMETHYL) 4 OXOTHIAZOLIDIN 3 YL]PHENYLAMIO] 6 DIMETHYLAMINO[1,3,5]TRIAZIN 2 YLOXY] 1 METHYL 1H QUINOLIN 2 ONE; 4 [4 [4 [2 (4 BROMOPHENYL) 5 (4 ETHYLPIPERAZIN 1 YLMETHYL) 4 OXOTHIAZOLIDIN 3 YL]PHENYLAMIO] 6 DIMETHYLAMINO[1,3,5]TRIAZIN 2 YLOXY] 1 METHYL 1H QUINOLIN 2 ONE; 4 [4 [4 [2 (4 CHLOROPHENYL) 5 (4 ETHYLPIPERAZIN 1 YLMETHYL) 4 OXOTHIAZOLIDIN 3 YL]PHENYLAMIO] 6 DIMETHYLAMINO[1,3,5]TRIAZIN 2 YLOXY] 1 METHYL 1H QUINOLIN 2 ONE; 4 [4 DIMETHYLAMINO 6 [4 [5 (4 ETHYLPIPERAZIN 1 YLMETHYL) 2 (2 NITROPHENYL) 4 OXOTHIAZOLIDIN 3 YL]PHENYLAMINO][1,3,5]TRIAZIN 2 YLOXY] 1 METHYL 1H QUINOLIN 2 ONE; 4 [4 DIMETHYLAMINO 6 [4 [5 (4 ETHYLPIPERAZIN 1 YLMETHYL) 2 (3 FLUOROPHENYL) 4 OXOTHIAZOLIDIN 3 YL]PHENYLAMINO][1,3,5]TRIAZIN 2 YLOXY] 1 METHYL 1H QUINOLIN 2 ONE; 4 [4 DIMETHYLAMINO 6 [4 [5 (4 ETHYLPIPERAZIN 1 YLMETHYL) 2 (4 FLUOROPHENYL) 4 OXOTHIAZOLIDIN 3 YL]PHENYLAMINO][1,3,5]TRIAZIN 2 YLOXY] 1 METHYL 1H QUINOLIN 2 ONE; 4 [4 DIMETHYLAMINO 6 [4 [5 (4 ETHYLPIPERAZIN 1 YLMETHYL) 2 (4 HYDROXYPHENYL) 4 OXOTHIAZOLIDIN 3 YL]PHENYLAMINO][1,3,5]TRIAZIN 2 YLOXY] 1 METHYL 1H QUINOLIN 2 ONE; 4 [4 DIMETHYLAMINO 6 [4 [5 (4 ETHYLPIPERAZIN 1 YLMETHYL) 2 (4 METHOXYPHENYL) 4 OXOTHIAZOLIDIN 3 YL]PHENYLAMINO][1,3,5]TRIAZIN 2 YLOXY] 1 METHYL 1H QUINOLIN 2 ONE; 4 [4 DIMETHYLAMINO 6 [4 [5 (4 ETHYLPIPERAZIN 1 YLMETHYL) 2 (4 NITROPHENYL) 4 OXOTHIAZOLIDIN 3 YL]PHENYLAMINO][1,3,5]TRIAZIN 2 YLOXY] 1 METHYL 1H QUINOLIN 2 ONE; 4 [4 DIMETHYLAMINO 6 [4 [5 (4 ETHYLPIPERAZIN 1 YLMETHYL) 4 OXO 2 4 TOLYLTHIAZOLIDIN 3 YL]PHENYLAMINO][1,3,5]TRIAZIN 2 YLOXY] 1 METHYL 1H QUINOLIN 2 ONE; 4 [4 DIMETHYLAMINO 6 [4 [5 (4 ETHYLPIPERAZIN 1 YLMETHYL) 4 OXO 2 PHENYLTHIAZOLIDIN 3 YL]PHENYLAMINO][1,3,5]TRIAZIN 2 YLOXY] 1 METHYL 1H QUINOLIN 2 ONE; ALDEHYDE DERIVATIVE; ANTIBIOTIC AGENT; ANTIFUNGAL AGENT; CIPROFLOXACIN; KETOCONAZOLE; SCHIFF BASE; THIAZOLIDINONE DERIVATIVE; UNCLASSIFIED DRUG;

ANTIBACTERIAL ACTIVITY; ANTIFUNGAL ACTIVITY; ARTICLE; ASPERGILLUS; ASPERGILLUS CLAVATUS; ASPERGILLUS FUMIGATUS; ASPERGILLUS NIDULANS; BACILLUS CEREUS; CANDIDA ALBICANS; CARBON NUCLEAR MAGNETIC RESONANCE; CYCLIZATION; DRUG STRUCTURE; DRUG SYNTHESIS; ESCHERICHIA COLI; KLEBSIELLA PNEUMONIAE; MINIMUM INHIBITORY CONCENTRATION; NONHUMAN; POLYMERIZATION; PROTEUS VULGARIS; PROTON NUCLEAR MAGNETIC RESONANCE; PSEUDOMONAS AERUGINOSA; SALMONELLA TYPHI; SHIGELLA FLEXNERI; STAPHYLOCOCCUS AUREUS; STRUCTURE ACTIVITY RELATION;

ANTI-INFECTIVE AGENTS; BACTERIA; MAGNETIC RESONANCE SPECTROSCOPY; MICROBIAL SENSITIVITY TESTS; SPECTROSCOPY, FOURIER TRANSFORM INFRARED; STRUCTURE-ACTIVITY RELATIONSHIP; THIAZOLIDINES;

EID: 84856011929     PISSN: 02235234     EISSN: 17683254     Source Type: Journal    
DOI: 10.1016/j.ejmech.2011.11.041     Document Type: Article

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