A combinatorial approach to 2,4,6-trisubstituted triazines with potent antimalarial activity: Combining conventional synthesis and microwave-assistance

ChemMedChem

Volumn 3, Issue 6, 2008, Pages 873-876

  Melato, Sergio ^a   Prosperi, Davide ^a   Coghi, Paolo ^a   Basilico, Nicoletta ^b   Monti, Diego ^a  

^a CNR   (Italy)

^b UNIVERSITY OF MILAN   (Italy)

Author keywords

Aminoquinolines; Antimalarial agents; Combinatorial chemistry; Microwave assistance; Triazines

Indexed keywords

ANTIMALARIAL AGENT; TRIAZINE DERIVATIVE;

ANIMAL; ARTICLE; CELL LINE; CHEMICAL STRUCTURE; COMBINATORIAL CHEMISTRY; DRUG EFFECT; DRUG SENSITIVITY; ENDOTHELIUM CELL; FIBROBLAST; HUMAN; MICROWAVE RADIATION; PLASMODIUM FALCIPARUM; RADIATION EXPOSURE; STEREOISOMERISM; STRUCTURE ACTIVITY RELATION; SYNTHESIS;

ANIMALS; ANTIMALARIALS; CELL LINE; COMBINATORIAL CHEMISTRY TECHNIQUES; ENDOTHELIAL CELLS; FIBROBLASTS; HUMANS; MICROWAVES; MOLECULAR STRUCTURE; PARASITIC SENSITIVITY TESTS; PLASMODIUM FALCIPARUM; STEREOISOMERISM; STRUCTURE-ACTIVITY RELATIONSHIP; TRIAZINES;

EID: 48149090074     PISSN: 18607179     EISSN: 18607187     Source Type: Journal    
DOI: 10.1002/cmdc.200700344     Document Type: Article

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