Structures of peptide agonists for human protease activated receptor 2

Bioorganic and Medicinal Chemistry Letters

Volumn 22, Issue 2, 2012, Pages 916-919

  Stoermer, Martin J ^a   Flanagan, Bernadine ^a   Beyer, Renée L ^a   Madala, Praveen K ^a   Fairlie, David P ^a  

^a UNIVERSITY OF QUEENSLAND   (Australia)

Author keywords

Agonist; Circular dichroism; Molecular modeling; Protease activated receptor 2; Structure

Indexed keywords

2 FUROYL LEUCYLISOLEUCYLGLYCYLARGINYLLEUCYLORNITHYLAMIDE; AGENTS INTERACTING WITH TRANSMITTER, HORMONE OR DRUG RECEPTORS; DIMETHYL SULFOXIDE; PEPTIDOMIMETIC AGENT; PROTEINASE ACTIVATED RECEPTOR 2; SERYLLEUCYLISOLEUCYLGLYCYLARGINYLLEUCYLAMIDE; SERYLLEUCYLISOLEUCYLGLYCYLLYSYLVALYLAMIDE; UNCLASSIFIED DRUG;

AMINO TERMINAL SEQUENCE; ARTICLE; CIRCULAR DICHROISM; DRUG RECEPTOR BINDING; DRUG STRUCTURE; HUMAN; NONHUMAN; PROTEIN CONFORMATION; PROTEIN MOTIF; PROTON NUCLEAR MAGNETIC RESONANCE; RAT;

HUMANS; MODELS, MOLECULAR; MOLECULAR CONFORMATION; OLIGOPEPTIDES; RECEPTOR, PAR-2; STRUCTURE-ACTIVITY RELATIONSHIP;

RATTUS;

EID: 84855655342     PISSN: 0960894X     EISSN: 14643405     Source Type: Journal    
DOI: 10.1016/j.bmcl.2011.12.029     Document Type: Article

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