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Volumn 2, Issue 12, 2011, Pages 1201-1207

Design, synthesis and biological evaluation of novel benzothiazole and triazole analogs as falcipain inhibitors

(7) Shah, Falgun a Wu, Yunshan a Gut, Jiri b Pedduri, Yakambram a Legac, Jennifer b Rosenthal, Philip J b Avery, Mitchell A a

a UNIVERSITY OF MISSISSIPPI (United States)

b UNIVERSITY OF CALIFORNIA (United States)

Author keywords

[No Author keywords available]

Indexed keywords

BENZOTHIAZOLE DERIVATIVE; CHLOROQUINE; CYSTEINE PROTEINASE; FALCIPAIN 2; FALCIPAIN 3; TRIAZOLE DERIVATIVE; UNCLASSIFIED DRUG;

AMINO ACID SEQUENCE; ANTIMALARIAL ACTIVITY; ANTIMALARIAL DRUG RESISTANCE; ARTICLE; BINDING SITE; CONCENTRATION RESPONSE; DRUG PROTEIN BINDING; DRUG STRUCTURE; DRUG SYNTHESIS; ENZYME INHIBITION; MOLECULAR DOCKING; NONHUMAN; PLASMODIUM FALCIPARUM; PRIORITY JOURNAL;

EID: 82455186225 PISSN: 20402503 EISSN: 20402511 Source Type: Journal
DOI: 10.1039/c1md00129a Document Type: Article

Times cited : (36)

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