SCOPUS 정보 검색 플랫폼

ChemMedChem

Volumn 6, Issue 11, 2011, Pages 1967-1970

Revisiting the rule of five on the basis of pharmacokinetic data from rat

(4) Ridder, Lars a Wang, Hongwu a de Vlieg, Jacob a,b,c Wagener, Markus a,d

a MERCK RESEARCH LABORATORIES (United States)

b RADBOUD UNIVERSITY MEDICAL CENTER (Netherlands)

c NETHERLANDS ESCIENCE CENTER (Netherlands)

d Particle Instruments (Germany)

Author keywords

LMW gonadotropins; Oral absorption; Physicochemical properties; Rat pharmacokinetics; Rule of five

Indexed keywords

DRUG;

ARTICLE; DRUG ABSORPTION; DRUG BIOAVAILABILITY; DRUG METABOLISM; HUMAN; NONHUMAN; PRIORITY JOURNAL; RAT;

ADMINISTRATION, ORAL; ANIMALS; BIOLOGICAL AVAILABILITY; GONADOTROPINS; MODELS, BIOLOGICAL; PHARMACEUTICAL PREPARATIONS; PHARMACOKINETICS; PHYSICOCHEMICAL PHENOMENA; RATS; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 80054989260 PISSN: 18607179 EISSN: 18607187 Source Type: Journal
DOI: 10.1002/cmdc.201100306 Document Type: Article

Times cited : (12)

References (29)

1
- 39749120717
- A. Ruiz-Garcia, M. Bermejo, A. Moss, V. G. Casabo, J. Pharm. Sci. 2008, 97, 654-690.
- (2008) J. Pharm. Sci. , vol.97 , pp. 654-690
- Ruiz-Garcia, A.¹ Bermejo, M.² Moss, A.³ Casabo, V.G.⁴

2
- 4344645978
- I. Kola, J. Landis, Nat. Rev. Drug Discovery 2004, 3, 711-715.
- (2004) Nat. Rev. Drug Discovery , vol.3 , pp. 711-715
- Kola, I.¹ Landis, J.²

3
- 15244348590
- H. Van De Waterbeemd, Basic Clin. Pharmacol. Toxicol. 2005, 96, 162-166.
- (2005) Basic Clin. Pharmacol. Toxicol. , vol.96 , pp. 162-166
- Waterbeemd, H.V.D.¹

4
- 3543026365
- K. Ito, J. B. Houston, Pharm. Res. 2004, 21, 785-792.
- (2004) Pharm. Res. , vol.21 , pp. 785-792
- Ito, K.¹ Houston, J.B.²

5
- 35348895572
- J. Yang, M. Jamei, K. R. Yeo, G. T. Tucker, A. Rostami-Hodjegan, Curr. Drug Metab. 2007, 8, 676-684.
- (2007) Curr. Drug Metab. , vol.8 , pp. 676-684
- Yang, J.¹ Jamei, M.² Yeo, K.R.³ Tucker, G.T.⁴ Rostami-Hodjegan, A.⁵

6
- 34247245174
- T. Hou, J. Wang, W. Zhang, X. Xu, J. Chem. Inf. Model. 2007, 47, 460-463.
- (2007) J. Chem. Inf. Model. , vol.47 , pp. 460-463
- Hou, T.¹ Wang, J.² Zhang, W.³ Xu, X.⁴

7
- 0031024171
- C. A. Lipinski, F. Lombardo, B. W. Dominy, P. J. Feeney, Adv. Drug Delivery Rev. 1997, 23, 3-25.
- (1997) Adv. Drug Delivery Rev. , vol.23 , pp. 3-25
- Lipinski, C.A.¹ Lombardo, F.² Dominy, B.W.³ Feeney, P.J.⁴

8
- 18244370266
- Y. C. Martin, J. Med. Chem. 2005, 48, 3164-3170.
- (2005) J. Med. Chem. , vol.48 , pp. 3164-3170
- Martin, Y.C.¹

9
- 0032714220
- J. Kelder, P. D. Grootenhuis, D. M. Bayada, L. P. Delbressine, J. P. Ploemen, Pharm. Res. 1999, 16, 1514-1519.
- (1999) Pharm. Res. , vol.16 , pp. 1514-1519
- Kelder, J.¹ Grootenhuis, P.D.² Bayada, D.M.³ Delbressine, L.P.⁴ Ploemen, J.P.⁵

10
- 0037030653
- D. F. Veber, S. R. Johnson, H. Y. Cheng, B. R. Smith, K. W. Ward, K. D. Kopple, J. Med. Chem. 2002, 45, 2615-2623.
- (2002) J. Med. Chem. , vol.45 , pp. 2615-2623
- Veber, D.F.¹ Johnson, S.R.² Cheng, H.Y.³ Smith, B.R.⁴ Ward, K.W.⁵ Kopple, K.D.⁶

11
- 71049126548
- F. Lovering, J. Bikker, C. Humblet, J. Med. Chem. 2009, 52, 6752-6756.
- (2009) J. Med. Chem. , vol.52 , pp. 6752-6756
- Lovering, F.¹ Bikker, J.² Humblet, C.³

12
- 70350409235
- T. J. Ritchie, S. J. Macdonald, Drug Discovery Today 2009, 14, 1011-1020.
- (2009) Drug Discovery Today , vol.14 , pp. 1011-1020
- Ritchie, T.J.¹ Macdonald, S.J.²

13
- 65449179589
- M. J. Waring, Bioorg. Med. Chem. Lett. 2009, 19, 2844-2851.
- (2009) Bioorg. Med. Chem. Lett. , vol.19 , pp. 2844-2851
- Waring, M.J.¹

14
- 39749181550
- M. P. Gleeson, J. Med. Chem. 2008, 51, 817-834.
- (2008) J. Med. Chem. , vol.51 , pp. 817-834
- Gleeson, M.P.¹

15
- 78651490914
- A. Böcker, P. R. Bonneau, O. Hucke, A. Jakalian, P. J. Edwards, ChemMedChem 2010, 5, 2102-2113.
- (2010) ChemMedChem , vol.5 , pp. 2102-2113
- Böcker, A.¹ Bonneau, P.R.² Hucke, O.³ Jakalian, A.⁴ Edwards, P.J.⁵

16
- 8644219619
- J. J. Lu, K. Crimin, J. T. Goodwin, P. Crivori, C. Orrenius, L. Xing, P. J. Tandler, T. J. Vidmar, B. M. Amore, A. G. Wilson, P. F. Stouten, P. S. Burton, J. Med. Chem. 2004, 47, 6104-6107.
- (2004) J. Med. Chem. , vol.47 , pp. 6104-6107
- Lu, J.J.¹ Crimin, K.² Goodwin, J.T.³ Crivori, P.⁴ Orrenius, C.⁵ Xing, L.⁶ Tandler, P.J.⁷ Vidmar, T.J.⁸ Amore, B.M.⁹ Wilson, A.G.¹⁰ Stouten, P.F.¹¹ Burton, P.S.¹²

17
- 33646715920
- R. Morphy, J. Med. Chem. 2006, 49, 2969-2978.
- (2006) J. Med. Chem. , vol.49 , pp. 2969-2978
- Morphy, R.¹

18
- 0031786518
- W. L. Chiou, A. Barve, Pharm. Res. 1998, 15, 1792-1795.
- (1998) Pharm. Res. , vol.15 , pp. 1792-1795
- Chiou, W.L.¹ Barve, A.²

19
- 0029894013
- G. W. Bemis, M. A. Murcko, J. Med. Chem. 1996, 39, 2887-2893.
- (1996) J. Med. Chem. , vol.39 , pp. 2887-2893
- Bemis, G.W.¹ Murcko, M.A.²

20
- 0036783410
- R. J. Riley, I. J. Martin, A. E. Cooper, Curr. Drug Metab. 2002, 3, 527-550.
- (2002) Curr. Drug Metab. , vol.3 , pp. 527-550
- Riley, R.J.¹ Martin, I.J.² Cooper, A.E.³

21
- 77955159974
- K. Sugano, M. Kansy, P. Artursson, A. Avdeef, S. Bendels, L. Di, G. F. Ecker, B. Faller, H. Fischer, G. Gerebtzoff, H. Lennernaes, F. Senner, Nat. Rev. Drug Discov. 2010, 9, 597-614.
- (2010) Nat. Rev. Drug Discov. , vol.9 , pp. 597-614
- Sugano, K.¹ Kansy, M.² Artursson, P.³ Avdeef, A.⁴ Bendels, S.⁵ Di, L.⁶ Ecker, G.F.⁷ Faller, B.⁸ Fischer, H.⁹ Gerebtzoff, G.¹⁰ Lennernaes, H.¹¹ Senner, F.¹²

22
- 16244418685
- N. Salamat-Miller, T. P. Johnston, Int. J. Pharm. 2005, 294, 201-206.
- (2005) Int. J. Pharm. , vol.294 , pp. 201-206
- Salamat-Miller, N.¹ Johnston, T.P.²

23
- 0035940057
- C. J. H. Porter, W. N. Charman, Adv. Drug. Deliv. Rev. 2001, 50, 61-80.
- (2001) Adv. Drug. Deliv. Rev. , vol.50 , pp. 61-80
- Porter, C.J.H.¹ Charman, W.N.²

24
- 33847394968
- C. J. H. Porter, N. L. Trevaskis, W. N. Charman, Nat. Rev. Drug Discov. 2007, 6, 231-248.
- (2007) Nat. Rev. Drug Discov. , vol.6 , pp. 231-248
- Porter, C.J.H.¹ Trevaskis, N.L.² Charman, W.N.³

25
- 34548049221
- D. J. Hauss, Adv. Drug. Deliv. Rev. 2007, 59, 667-676.
- (2007) Adv. Drug. Deliv. Rev. , vol.59 , pp. 667-676
- Hauss, D.J.¹

26
- 0037020293
- N. C. vanStraten, G. G. Schoonus-Gerritsma, R. G. vanSomeren, J. Draaijer, A. E. Adang, C. M. Timmers, R. G. Hanssen, C. A. vanBoeckel, ChemBioChem 2002, 3, 1023-1026.
- (2002) ChemBioChem , vol.3 , pp. 1023-1026
- vanStraten, N.C.¹ Schoonus-Gerritsma, G.G.² vanSomeren, R.G.³ Draaijer, J.⁴ Adang, A.E.⁵ Timmers, C.M.⁶ Hanssen, R.G.⁷ vanBoeckel, C.A.⁸

27
- 54249130252
- C. J. vanKoppen, G. J. Zaman, C. M. Timmers, J. Kelder, S. Mosselman, R. van de Lagemaat, M. J. Smit, R. G. Hanssen, Naunyn Schmiedebergs Arch. Pharmacol. 2008, 378, 503-514.
- (2008) Naunyn Schmiedebergs Arch. Pharmacol. , vol.378 , pp. 503-514
- van Koppen, C.J.¹ Zaman, G.J.² Timmers, C.M.³ Kelder, J.⁴ Mosselman, S.⁵ van de Lagemaat, R.⁶ Smit, M.J.⁷ Hanssen, R.G.⁸

28
- 61449108160
- R. van de Lagemaat, C. M. Timmers, J. Kelder, C. vanKoppen, S. Mosselman, R. G. J. M. Hanssen, Hum. Reprod. 2009, 24, 640-648.
- (2009) Hum. Reprod. , vol.24 , pp. 640-648
- van de Lagemaat, R.¹ Timmers, C.M.² Kelder, J.³ vanKoppen, C.⁴ Mosselman, S.⁵ Hanssen, R.G.J.M.⁶

29
- 80055022606
- (Ed.: John E. Macor), Academic Press
- N. C. van Straten, C. M. Timmers in Annual Reports in Medicinal Chemistry (Ed.: John E. Macor), Academic Press, 2009, pp.171-188.
- (2009) Annual Reports in Medicinal Chemistry , pp. 171-188
- van Straten, N.C.¹ Timmers, C.M.²

* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.