-
1
-
-
0028948839
-
A theoretical basis for a biopharmaceutical drug classification: The correlation of in vitro drug product dissolution and in vivo bioavailability
-
G. L. Amidon, H. Lennernäs, V. P. Shah, and J. R. Crison. A theoretical basis for a biopharmaceutical drug classification: The correlation of in vitro drug product dissolution and in vivo bioavailability. Pharm. Res. 12:413-420 (1995).
-
(1995)
Pharm. Res.
, vol.12
, pp. 413-420
-
-
Amidon, G.L.1
Lennernäs, H.2
Shah, V.P.3
Crison, J.R.4
-
2
-
-
0029855969
-
Comparison between permeability coefficients in rat and human jejunum
-
U. Fagerholm, M. Johansson, and H. Lennernäs. Comparison between permeability coefficients in rat and human jejunum. Pharm. Res. 13:1336-1342 (1996).
-
(1996)
Pharm. Res.
, vol.13
, pp. 1336-1342
-
-
Fagerholm, U.1
Johansson, M.2
Lennernäs, H.3
-
3
-
-
0028023628
-
Determination of drug permeability in a flat or distended stirred intestine: Prediction of fraction dose absorbed in humans after oral administration
-
W. L. Chiou. Determination of drug permeability in a flat or distended stirred intestine: Prediction of fraction dose absorbed in humans after oral administration. Int. J. Clin. Pharmacol. Ther. 32:474-482 (1994).
-
(1994)
Int. J. Clin. Pharmacol. Ther.
, vol.32
, pp. 474-482
-
-
Chiou, W.L.1
-
4
-
-
0028877755
-
The validation of the intestinal permeability approach to predict oral fraction of dose absorbed in humans and rats
-
W. L. Chiou. The validation of the intestinal permeability approach to predict oral fraction of dose absorbed in humans and rats. Biopharm. Drug. Disp. 16:71-75 (1995).
-
(1995)
Biopharm. Drug. Disp.
, vol.16
, pp. 71-75
-
-
Chiou, W.L.1
-
5
-
-
0031413597
-
Improved prediction of in vivo peroral absorption from in vitro intestinal permeability using an internal standard to control for intra- and inter-rat variability
-
M. E. Dowty and C. R. Dietsch. Improved prediction of in vivo peroral absorption from in vitro intestinal permeability using an internal standard to control for intra- and inter-rat variability. Pharm. Res. 14:1792-1797 (1997).
-
(1997)
Pharm. Res.
, vol.14
, pp. 1792-1797
-
-
Dowty, M.E.1
Dietsch, C.R.2
-
6
-
-
9844259465
-
Human intestinal permeability of piroxicam, propranolol, phenylalanine, and PEG 400 determined by jejunal perfusion
-
N. Takamatsu, L. S. Welage, N. M. Idkaidek, D. Liu, P. I-Der Lee, Y. Hayashi, J. K. Rhie, H. Lennernäs, J. L. Barnett, V. P. Shah, L. Lesko, and G. L. Amidon. Human intestinal permeability of piroxicam, propranolol, phenylalanine, and PEG 400 determined by jejunal perfusion. Pharm. Res. 14:1127-1132 (1997).
-
(1997)
Pharm. Res.
, vol.14
, pp. 1127-1132
-
-
Takamatsu, N.1
Welage, L.S.2
Idkaidek, N.M.3
Liu, D.4
I-Der Lee, P.5
Hayashi, Y.6
Rhie, J.K.7
Lennernäs, H.8
Barnett, J.L.9
Shah, V.P.10
Lesko, L.11
Amidon, G.L.12
-
7
-
-
0025804183
-
Correlation between oral drug absorption in humans and apparent drug permeability coefficients in human intestinal epithelial (Caco-2) cells
-
P. Artursson and J. Karlsson. Correlation between oral drug absorption in humans and apparent drug permeability coefficients in human intestinal epithelial (Caco-2) cells. Biochem. Biophys. Res. Commun. 175:880-885 (1991).
-
(1991)
Biochem. Biophys. Res. Commun.
, vol.175
, pp. 880-885
-
-
Artursson, P.1
Karlsson, J.2
-
8
-
-
0030588714
-
Caco-2 monolayers in experimental and theoretical predictions of drug transport
-
P. Artursson, K. Palm, and K. Luthman. Caco-2 monolayers in experimental and theoretical predictions of drug transport. Advanced Drug Delivery Reviews 22:67-84 (1996).
-
(1996)
Advanced Drug Delivery Reviews
, vol.22
, pp. 67-84
-
-
Artursson, P.1
Palm, K.2
Luthman, K.3
-
9
-
-
0031413702
-
Intestinal drug absorption and metabolism in cell cultures: Caco-2 and beyond
-
P. Artursson and R. Borchardt. Intestinal drug absorption and metabolism in cell cultures: Caco-2 and beyond. Pharm. Res. 14:1655-1658 (1997).
-
(1997)
Pharm. Res.
, vol.14
, pp. 1655-1658
-
-
Artursson, P.1
Borchardt, R.2
-
10
-
-
0029562018
-
The author replies to Lennernäs et al
-
W. L. Chiou. The author replies to Lennernäs et al. J. Pharmacokin. Biopharm. 23:323-331 (1995).
-
(1995)
J. Pharmacokin. Biopharm.
, vol.23
, pp. 323-331
-
-
Chiou, W.L.1
-
11
-
-
0030514291
-
New perspectives on the theory of permeability and resistance in the study of drug transport and absorption
-
W. L. Chiou. New perspectives on the theory of permeability and resistance in the study of drug transport and absorption. J. Pharmacokin. Biopharm. 24:433-442 (1996).
-
(1996)
J. Pharmacokin. Biopharm.
, vol.24
, pp. 433-442
-
-
Chiou, W.L.1
-
12
-
-
0020912679
-
Studies on potential factors affecting incomplete absorption of furosemide: Gastric first-pass effect
-
M. G. Lee and W. L. Chiou. Studies on potential factors affecting incomplete absorption of furosemide: Gastric first-pass effect. J. Pharmacokin. Biopharm. 11:623-640 (1983).
-
(1983)
J. Pharmacokin. Biopharm.
, vol.11
, pp. 623-640
-
-
Lee, M.G.1
Chiou, W.L.2
-
13
-
-
0023605292
-
The phenomenon and cause of dose-dependent oral absorption of chlorothiazide in rats: Extrapolation to human data based on the body surface area concept
-
F. H. Hsu, T. Prueksaritanont, M. G. Lee, and W. L. Chiou. The phenomenon and cause of dose-dependent oral absorption of chlorothiazide in rats: Extrapolation to human data based on the body surface area concept. J. Pharmacokin. Biopharm. 15:369-383 (1987).
-
(1987)
J. Pharmacokin. Biopharm.
, vol.15
, pp. 369-383
-
-
Hsu, F.H.1
Prueksaritanont, T.2
Lee, M.G.3
Chiou, W.L.4
-
14
-
-
0002769936
-
Design and Optimization of dosage regimens; Pharmacokinetic data
-
A. Goodman Gilman, J. G. Hardman, L. E. Limbard, P. B. Molinoff, and R. W. Ruddon (eds.) McGraw Hill, NY
-
L. Z. Benet, S. Øie, and J. B. Schwartz. Design and Optimization of dosage regimens; Pharmacokinetic data. In A. Goodman Gilman, J. G. Hardman, L. E. Limbard, P. B. Molinoff, and R. W. Ruddon (eds.) Goodman and Gilman's The Pharmacological Basis of Therapeutics, 9th edition, pp. 1707-1792, McGraw Hill, NY, 1996.
-
(1996)
Goodman and Gilman's the Pharmacological Basis of Therapeutics, 9th Edition
, pp. 1707-1792
-
-
Benet, L.Z.1
Øie, S.2
Schwartz, J.B.3
-
15
-
-
0029939330
-
In vitro permeability through Caco-2 cells is not quantitatively predictive of in vivo absorption for peptide-like drugs absorbed via the dipeptide transporter system
-
S. Chong, S. A. Dando, K. M. Soucek, and R. A. Morrison. In vitro permeability through Caco-2 cells is not quantitatively predictive of in vivo absorption for peptide-like drugs absorbed via the dipeptide transporter system. Pharm. Res. 13:120-123 (1996).
-
(1996)
Pharm. Res.
, vol.13
, pp. 120-123
-
-
Chong, S.1
Dando, S.A.2
Soucek, K.M.3
Morrison, R.A.4
-
16
-
-
0029991021
-
Measurements of the jejunal unstirred layer in normal subjects and patients with celiac disease
-
A. Strocchi, G. Corazza, J. Furne, C. Fine, A. DiSario, G. Gasbarrini, and M. D. Levitt. Measurements of the jejunal unstirred layer in normal subjects and patients with celiac disease. Am. J. Physiol. 270:G487-G491 (1996).
-
(1996)
Am. J. Physiol.
, vol.270
-
-
Strocchi, A.1
Corazza, G.2
Furne, J.3
Fine, C.4
DiSario, A.5
Gasbarrini, G.6
Levitt, M.D.7
-
17
-
-
0031958251
-
Species differences in size discrimination in the paracellular pathway reflected by oral bioavailability of poly(ethylene glycol) and D-peptides
-
Y. L. He, S. Murby, G. Warhurst, L. Gifford, D. Walker, J. Ayrton, R. Eastmond, and M. Rowland. Species differences in size discrimination in the paracellular pathway reflected by oral bioavailability of poly(ethylene glycol) and D-peptides. J. Pharm. Sci. 87:626-633 (1998).
-
(1998)
J. Pharm. Sci.
, vol.87
, pp. 626-633
-
-
He, Y.L.1
Murby, S.2
Warhurst, G.3
Gifford, L.4
Walker, D.5
Ayrton, J.6
Eastmond, R.7
Rowland, M.8
-
18
-
-
0019831462
-
Chronic dog intestinal loop model for studying drug absorption as exemplified by beta-adrenoceptor blocking agents, atenolol and propranolol
-
D. C. Taylor, R. Grundy, and B. Loveday. Chronic dog intestinal loop model for studying drug absorption as exemplified by beta-adrenoceptor blocking agents, atenolol and propranolol. J. Pharm. Sci. 70:516-21 (1981).
-
(1981)
J. Pharm. Sci.
, vol.70
, pp. 516-521
-
-
Taylor, D.C.1
Grundy, R.2
Loveday, B.3
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