Synthesis and preliminary biological evaluation of novel N-(3-aryl-1,2,4-triazol-5-yl) cinnamamide derivatives as potential antimycobacterial agents: An operational Topliss Tree approach

Bioorganic and Medicinal Chemistry Letters

Volumn 21, Issue 21, 2011, Pages 6523-6526

  Kakwani, Manoj D ^a   Desai, Nutan H Palsule ^a   Lele, Arundhati C ^a   Ray, Muktikant ^b   Rajan, M G R ^b   Degani, Mariam S ^a  

^a INSTITUTE OF CHEMICAL TECHNOLOGY   (India)

^b TATA MEMORIAL HOSPITAL   (India)

Author keywords

FAS II; Mycobacterium tuberculosis; Topliss tree; Triazoles

Indexed keywords

ANTIMYCOBACTERIAL AGENT; N (3 ARYL 1,2,4 TRIAZOL 5 YL)CINNAMAMIDE DERIVATIVE; N (3 PHENYL 1,2,4 TRIAZOL 5 YL)CINNAMAMIDE DERIVATIVE; UNCLASSIFIED DRUG;

ANTIMICROBIAL ACTIVITY; ARTICLE; CHEMICAL PROCEDURES; CONTROLLED STUDY; DRUG SAFETY; DRUG SCREENING; DRUG SYNTHESIS; MINIMUM INHIBITORY CONCENTRATION; MYCOBACTERIUM TUBERCULOSIS; NONHUMAN; STRUCTURE ACTIVITY RELATION; TOPLISS TREE APPROACH;

MYCOBACTERIUM TUBERCULOSIS;

EID: 80054789009     PISSN: 0960894X     EISSN: 14643405     Source Type: Journal    
DOI: 10.1016/j.bmcl.2011.08.076     Document Type: Article

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