Synthesis and evaluation of a novel series of pseudo-cinnamic derivatives as antituberculosis agents

Bioorganic and Medicinal Chemistry Letters

Volumn 19, Issue 2, 2009, Pages 341-343

  Yoya, Georges Koumba ^a,c   Bedos Belval, Florence ^a,c   Constant, Patricia ^b,d   Duran, Hubert ^a,c   Daffé, Mamadou ^b,d   Baltas, Michel ^a,c  

^a UNIVERSITÉ DE TOULOUSE   (France)

^b UNIVERSITÉ PAUL SABATIER   (France)

^c CNRS   (France)

^d INSTITUT DE PHARMACOLOGIE ET DE BIOLOGIE STRUCTURALE   (France)

Author keywords

Antituberculosis agents; Cinnamic derivatives; Mycobacterium tuberculosis; TB MIC

Indexed keywords

ALKANE DERIVATIVE; AMIDE; CINNAMIC ACID DERIVATIVE; HYDROXYL GROUP; N (2 ACETAMIDOETHYL) 3 [4 (3,7 DIMETHYLOCTA 2,6 DIENYLOXY)PHENYL]ACRYLAMIDE; THIOESTER; TUBERCULOSTATIC AGENT; UNCLASSIFIED DRUG;

ANTIBACTERIAL ACTIVITY; ARTICLE; CHEMICAL REACTION; COLORIMETRY; DRUG ACTIVITY; DRUG STRUCTURE; DRUG SYNTHESIS; MINIMUM INHIBITORY CONCENTRATION; MYCOBACTERIUM TUBERCULOSIS; NONHUMAN; QUANTUM YIELD;

ANTITUBERCULAR AGENTS; CINNAMATES; MICROBIAL SENSITIVITY TESTS; MYCOBACTERIUM TUBERCULOSIS;

MYCOBACTERIUM TUBERCULOSIS;

EID: 57749116991     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2008.11.082     Document Type: Article

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