Design, synthesis and antimycobacterial activity of cinnamide derivatives: A molecular hybridization approach

Bioorganic and Medicinal Chemistry Letters

Volumn 21, Issue 7, 2011, Pages 1997-1999

  Kakwani, Manoj D ^a   Suryavanshi, Prashant ^c   Ray, Muktikant ^b   Rajan, M G R ^b   Majee, Sharmila ^c   Samad, Abdul ^c   Devarajan, Padma ^a   Degani, Mariam S ^a  

^a INSTITUTE OF CHEMICAL TECHNOLOGY   (India)

^b TATA MEMORIAL HOSPITAL   (India)

^c BOMBAY VETERINARY COLLEGE   (India)

Author keywords

Antimycobacterial activity; Cinnamic acid; Diamine; Hybridization; Mycobacterium tuberculosis (Mtb); Synergy

Indexed keywords

ANTIINFECTIVE AGENT; CERULENIN; CINNAMAMIDE DERIVATIVE; ETHAMBUTOL; ISONIAZID; RIFAMPICIN; UNCLASSIFIED DRUG;

ANTIMICROBIAL ACTIVITY; ARTICLE; CONTROLLED STUDY; DRUG DESIGN; DRUG POTENCY; DRUG POTENTIATION; DRUG SAFETY; DRUG STRUCTURE; DRUG SYNTHESIS; MINIMUM INHIBITORY CONCENTRATION; MOLECULAR HYBRIDIZATION; NONHUMAN; PROCESS OPTIMIZATION; STRUCTURE ACTIVITY RELATION; VERO CELL;

ANIMALS; ANTITUBERCULAR AGENTS; CERCOPITHECUS AETHIOPS; CINNAMATES; DRUG DESIGN; MICROBIAL SENSITIVITY TESTS; MYCOBACTERIUM; NUCLEIC ACID HYBRIDIZATION; VERO CELLS;

MYCOBACTERIUM TUBERCULOSIS;

EID: 79952490524     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2011.02.022     Document Type: Article

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