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Bioorganic and Medicinal Chemistry Letters

Volumn 21, Issue 19, 2011, Pages 5707-5710

Effects of linker elongation in a series of N-(2-benzofuranylmethyl)- N′-(methoxyphenylalkyl)piperazine σ 1 receptor ligands

(5) Moussa, Iman A a Banister, Samuel D a Akladios, Fady N a Chua, Sook Wern b Kassiou, Michael a,b

a UNIVERSITY OF SYDNEY (Australia)

b UNIVERSITY OF SYDNEY (Australia)

Author keywords

CNS; Piperazines; Sigma receptors; Structure affinity relationships

Indexed keywords

PENTAZOCINE; PIPERAZINE DERIVATIVE; SIGMA 1 OPIATE RECEPTOR;

ANIMAL TISSUE; ARTICLE; BRAIN HOMOGENATE; DRUG RECEPTOR BINDING; DRUG STRUCTURE; DRUG SYNTHESIS; ISOTOPE LABELING; NONHUMAN; RAT; RECEPTOR AFFINITY;

ANIMALS; BENZOFURANS; DRUG DESIGN; DRUG DISCOVERY; HYDROPHOBIC AND HYDROPHILIC INTERACTIONS; LIGANDS; MODELS, CHEMICAL; MOLECULAR STRUCTURE; PC12 CELLS; PIPERAZINES; PROTEIN BINDING; RADIOLIGAND ASSAY; RATS; RECEPTORS, SEROTONIN; RECEPTORS, SIGMA; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 80052586768 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2011.08.029 Document Type: Article

Times cited : (6)

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