-
1
-
-
0034461768
-
Drug-like properties and the causes of poor solubility and poor permeability
-
DOI 10.1016/S1056-8719(00)00107-6, PII S1056871900001076
-
Lipinski CA. (2000). Drug-like properties and the causes of poor solubility and poor permeability. J Pharmacol Toxicol Methods, 44:235-249 (Pubitemid 32239479)
-
(2000)
Journal of Pharmacological and Toxicological Methods
, vol.44
, Issue.1
, pp. 235-249
-
-
Lipinski, C.A.1
-
2
-
-
0035289779
-
Experimental and computational approaches to estimate solubility and permeability in drug discovery and development settings
-
DOI 10.1016/S0169-409X(00)00129-0, PII S0169409X00001290
-
Lipinski CA, Lombardo F, Dominy BW, Feeney PJ. (2001). Experimental and computational approaches to estimate solubility and permeability in drug discovery and development settings. Adv Drug Deliv Rev, 46:3-26 (Pubitemid 33653411)
-
(2000)
Advanced Drug Delivery Reviews
, vol.46
, Issue.1-3
, pp. 3-26
-
-
Lipinski, C.A.1
Lombardo, F.2
Dominy, B.W.3
Feeney, P.J.4
-
3
-
-
0016737275
-
The influence of polyvinylpyrrolidone on the dissolution properties of hydroflumethiazide
-
Corrigan OI, Timoney RF. (1975). The influence of polyvinylpyrrolidone on the dissolution properties of hydroflumethiazide. J Pharm Pharmacol, 27:759-764
-
(1975)
J Pharm Pharmacol
, vol.27
, pp. 759-764
-
-
Corrigan, O.I.1
Timoney, R.F.2
-
4
-
-
0021329149
-
Amorphous spray-dried hydroflumethiazide-polyvinylpyrrolidone systems: Physicochemical properties
-
Corrigan OI, Holohan EM. (1984). Amorphous spraydried hydroflumethiazide-polyvinylpyrrolidone systems: physiochemical properties. J Pharm Pharmacol, 36:217-221 (Pubitemid 14164792)
-
(1984)
Journal of Pharmacy and Pharmacology
, vol.36
, Issue.4
, pp. 217-221
-
-
Corrigan, O.I.1
Holohan, E.M.2
-
5
-
-
0033460251
-
The effect of dry mixing on the apparent solubility of hydrophobic, sparingly soluble drugs
-
DOI 10.1016/S0928-0987(99)00043-3, PII S0928098799000433
-
Mosharraf M, Nystr C. (1999). The effect of dry mixing on the apparent solubility of hydrophobic, sparingly soluble drugs. Eur J Pharm Sci, 9:145-156 (Pubitemid 30012071)
-
(1999)
European Journal of Pharmaceutical Sciences
, vol.9
, Issue.2
, pp. 145-156
-
-
Mosharraf, M.1
Nystrom, C.2
-
6
-
-
45849152090
-
Effect of amorphous content on dissolution characteristics of rifampicin
-
DOI 10.1080/03639040701842451, PII 793946493
-
Panchagnula R, Bhardwaj V. (2008). Effect of amorphous content on dissolution characteristics of rifampicin. Drug Dev Ind Pharm, 34:642-649 (Pubitemid 351878683)
-
(2008)
Drug Development and Industrial Pharmacy
, vol.34
, Issue.6
, pp. 642-649
-
-
Panchagnula, R.1
Bhardwaj, V.2
-
7
-
-
5144219871
-
Amorphous drug delivery systems: Molecular aspects, design, and performance
-
DOI 10.1615/CritRevTherDrugCarrierSyst.v21.i3.10
-
Kaushal AM, Gupta P, Bansal AK. (2004). Amorphous drug delivery systems: molecular aspects, design, and performance. Crit Rev Ther Drug Carrier Syst, 21:133-193 (Pubitemid 41647581)
-
(2004)
Critical Reviews in Therapeutic Drug Carrier Systems
, vol.21
, Issue.3
, pp. 133-193
-
-
Kaushal, A.M.1
Gupta, P.2
Bansal, A.K.3
-
8
-
-
77956315485
-
-
Academic Press, San Diego
-
Zhang GGZ, Chen Y, Qiu Y. (2009). Crystalline and amorphous solids, in Developing Solid Oral Dosage Forms. Academic Press, San Diego, pp. 25-60
-
(2009)
Crystalline and Amorphous Solids, in Developing Solid Oral Dosage Forms
, pp. 25-60
-
-
Ggz, Z.1
Chen, Y.2
Qiu, Y.3
-
9
-
-
0032513499
-
Physico-chemical characterization of solid dispersions of temazepam with polyethylene glycol 6000 and PVP K30
-
DOI 10.1016/S0378-5173(97)00401-8, PII S0378517397004018
-
Van den Mooter G, Augustijns P, Blaton N, Kinget R. (1998). Physico-chemical characterization of solid dispersions of temazepam with polyethylene glycol 6000 and PVP K30. Int J Pharm, 164:67-80 (Pubitemid 28160099)
-
(1998)
International Journal of Pharmaceutics
, vol.164
, Issue.1-2
, pp. 67-80
-
-
Van Den Mooter, G.1
Augustijns, P.2
Blaton, N.3
Kinget, R.4
-
10
-
-
0036806561
-
Comparative physicochemical properties of hydrocortisone-PVP composites prepared using supercritical carbon dioxide by the GAS anti-solvent recrystallization process, by coprecipitation and by spray drying
-
DOI 10.1016/S0378-5173(02)00326-5, PII S0378517302003265
-
Corrigan OI, Crean AM. (2002). Comparative physicochemical properties of hydrocortisone-PVP composites prepared using supercritical carbon dioxide by the GAS anti-solvent recrystallization process, by coprecipitation and by spray drying. Int J Pharm, 245:75-82 (Pubitemid 35299893)
-
(2002)
International Journal of Pharmaceutics
, vol.245
, Issue.1-2
, pp. 75-82
-
-
Corrigan, O.I.1
Crean, A.M.2
-
11
-
-
71649096923
-
Characterisation of the thermal, spectroscopic and drug dissolution properties of mefenamic acid and polyoxyethylene-polyoxypropylene solid dispersions
-
Andrews GP, Zhai H, Tipping S, Jones DS. (2009). Characterisation of the thermal, spectroscopic and drug dissolution properties of mefenamic acid and polyoxyethylene-polyoxypropylene solid dispersions. J Pharm Sci, 98:4545-4556
-
(2009)
J Pharm Sci
, vol.98
, pp. 4545-4556
-
-
Andrews, G.P.1
Zhai, H.2
Tipping, S.3
Jones, D.S.4
-
12
-
-
0033663452
-
Physical stabilisation of amorphous ketoconazole in solid dispersions with polyvinylpyrrolidone K25
-
Van den Mooter G, Wuyts M, Blaton N, Busson R, Grobet P, Augustijns P et al. (2001). Physical stabilisation of amorphous ketoconazole in solid dispersions with polyvinylpyrrolidone K25. Eur J Pharm Sci, 12:261-269
-
(2001)
Eur J Pharm Sci
, vol.12
, pp. 261-269
-
-
Van Den Mooter, G.1
Wuyts, M.2
Blaton, N.3
Busson, R.4
Grobet, P.5
Augustijns, P.6
-
13
-
-
34047252848
-
Preparation of glass solutions of three poorly water soluble drugs by spray drying, melt extrusion and ball milling
-
DOI 10.1016/j.ijpharm.2006.11.030, PII S0378517306009781
-
Patterson JE, James MB, Forster AH, Lancaster RW, Butler JM, Rades T. (2007). Preparation of glass solutions of three poorly water soluble drugs by spray drying, melt extrusion and ball milling. Int J Pharm, 336:22-34 (Pubitemid 46551551)
-
(2007)
International Journal of Pharmaceutics
, vol.336
, Issue.1
, pp. 22-34
-
-
Patterson, J.E.1
James, M.B.2
Forster, A.H.3
Lancaster, R.W.4
Butler, J.M.5
Rades, T.6
-
14
-
-
0029586490
-
Enhancement of dissolution of glyburide by solid dispersion and lyophilization techniques
-
DOI 10.1016/0378-5173(95)04114-1
-
Betageri GV, Makarla KR. (1995). Enhancement of dissolution of glyburide by solid dispersion and lyophilization techniques. Int J Pharm, 126:155-160 (Pubitemid 26015632)
-
(1995)
International Journal of Pharmaceutics
, vol.126
, Issue.1-2
, pp. 155-160
-
-
Betageri, G.V.1
Makarla, K.R.2
-
15
-
-
33646799460
-
Evaluation of Inutec SP1 as a new carrier in the formulation of solid dispersions for poorly soluble drugs
-
DOI 10.1016/j.ijpharm.2006.02.025, PII S0378517306001499
-
Van den Mooter G, Weuts I, De Ridder T, Blaton N. (2006). Evaluation of Inutec SP1 as a new carrier in the formulation of solid dispersions for poorly soluble drugs. Int J Pharm, 316: 1-6 (Pubitemid 43765697)
-
(2006)
International Journal of Pharmaceutics
, vol.316
, Issue.1-2
, pp. 1-6
-
-
Van Den Mooter, G.1
Weuts, I.2
De Ridder, T.3
Blaton, N.4
-
16
-
-
1442309058
-
9-tetrahydrocannabinol
-
DOI 10.1016/j.ejps.2003.11.014, PII S0928098703003348
-
van Drooge DJ, Hinrichs WL, Wegman KA, Visser MR, Eissens AC, Frijlink HW. (2004). Solid dispersions based on inulin for the stabilisation and formulation of delta 9-tetrahydrocannabinol. Eur J Pharm Sci, 21:511-518 (Pubitemid 38283925)
-
(2004)
European Journal of Pharmaceutical Sciences
, vol.21
, Issue.4
, pp. 511-518
-
-
Van Drooge, D.J.1
Hinrichs, W.L.J.2
Wegman, K.A.M.3
Visser, M.R.4
Eissens, A.C.5
Frijlink, H.W.6
-
17
-
-
63649134819
-
Co-solvent evaporation method for enhancement of solubility and dissolution rate of poorly aqueous soluble drug simvastatin: In vitro-in vivo evaluation
-
Pandya P, Gattani S, Jain P, Khirwal L, Surana S. (2008). Co-solvent evaporation method for enhancement of solubility and dissolution rate of poorly aqueous soluble drug simvastatin: in vitro-in vivo evaluation. AAPS Pharmscitech, 9:1247-1252
-
(2008)
AAPS Pharmscitech
, vol.9
, pp. 1247-1252
-
-
Pandya, P.1
Gattani, S.2
Jain, P.3
Khirwal, L.4
Surana, S.5
-
19
-
-
0031749397
-
A pragmatic test of a simple calorimetric method for determining the fragility of some amorphous pharmaceutical materials
-
DOI 10.1023/A:1011931305755
-
Hancock BC, Dalton CR, Pikal MJ, Shamblin SL. (1998). A pragmatic test of a simple calorimetric method for determining the fragility of some amorphous pharmaceutical materials. Pharm Res, 15:762-767 (Pubitemid 28275655)
-
(1998)
Pharmaceutical Research
, vol.15
, Issue.5
, pp. 762-767
-
-
Hancock, B.C.1
Dalton, C.R.2
Pikal, M.J.3
Shamblin, S.L.4
-
20
-
-
33947094816
-
Compositional variation of glasstransition temperatures. 2. Application of the thermodynamic theory to compatible polymer blends
-
Couchman PR. (1978). Compositional variation of glasstransition temperatures. 2. Application of the thermodynamic theory to compatible polymer blends. Macromolecules, 11:1156-1161
-
(1978)
Macromolecules
, vol.11
, pp. 1156-1161
-
-
Couchman, P.R.1
-
21
-
-
4243167095
-
A classical thermodynamic discussion of the effect of composition on glass-transition temperatures
-
Couchman PR, Karasz FE. (1978). A classical thermodynamic discussion of the effect of composition on glass-transition temperatures. Macromolecules, 11:117-119
-
(1978)
Macromolecules
, vol.11
, pp. 117-119
-
-
Couchman, P.R.1
Karasz, F.E.2
-
22
-
-
54749092941
-
Entropy of mixing and the glass transition of amorphous mixtures
-
Pinal R. (2008). Entropy of mixing and the glass transition of amorphous mixtures. Entropy, 10:207-223
-
(2008)
Entropy
, vol.10
, pp. 207-223
-
-
Pinal, R.1
-
23
-
-
0344013128
-
Comparison of the Gordon-Taylor and Couchman-Karasz equations for prediction of the glass transition temperature of glass solutions of drug and polyvinylpyrrolidone prepared by melt extrusion
-
Forster A, Hempenstall J, Rades T. (2003). Comparison of the Gordon-Taylor and Couchman-Karasz equations for prediction of the glass transition temperature of glass solutions of drug and polyvinylpyrrolidone prepared by melt extrusion. Pharmazie, 58:838-839 (Pubitemid 37462471)
-
(2003)
Pharmazie
, vol.58
, Issue.11
, pp. 838-839
-
-
Forster, A.1
Hempenstall, J.2
Rades, T.3
-
24
-
-
15244352688
-
Physicochemical evaluation of PVP-thiazide diuretic interactions in co-spray-dried composites - Analysis of glass transition composition relationships
-
DOI 10.1016/j.ejps.2005.01.007
-
Tajber L, Corrigan OI, Healy AM. (2005). Physicochemical evaluation of PVP-thiazide diuretic interactions in co-spray-dried composites-analysis of glass transition composition relationships. Eur J Pharm Sci, 24:553-563 (Pubitemid 40387269)
-
(2005)
European Journal of Pharmaceutical Sciences
, vol.24
, Issue.5
, pp. 553-563
-
-
Tajber, L.1
Corrigan, O.I.2
Healy, A.M.3
-
25
-
-
0035964472
-
Influence of various drugs on the glass transition temperature of poly(vinylpyrrolidone): A thermodynamic and spectroscopic investigation
-
DOI 10.1016/S0378-5173(01)00767-0, PII S0378517301007670
-
Nair R, Nyamweya N, Gien S, Martiez-Miranda LJ, Hoag SW. (2001). Influence of various drugs on the glass transition temperature of poly(vinylpyrrolidone): a thermodynamic and spectroscopic investigation. Int J Pharm, 225:83-96 (Pubitemid 32728202)
-
(2001)
International Journal of Pharmaceutics
, vol.225
, Issue.1-2
, pp. 83-96
-
-
Nair, R.1
Nyamweya, N.2
Gonen, S.3
Martinez-Miranda, L.J.4
Hoag, S.W.5
-
27
-
-
64649105426
-
FTIR studies on differential intermolecular association in crystalline and amorphous states of structurally related non-steroidal antiinflammatory drugs
-
Kaushal AM, Chakraborti AK, Bansal AK. (2008). FTIR studies on differential intermolecular association in crystalline and amorphous states of structurally related non-steroidal antiinflammatory drugs. Mol Pharm, 5:937-945
-
(2008)
Mol Pharm
, vol.5
, pp. 937-945
-
-
Kaushal, A.M.1
Chakraborti, A.K.2
Bansal, A.K.3
-
28
-
-
84895919989
-
Adsorption at solid surfaces: Pharmaceutical applications
-
J., Swarbrick, ed Informa Healthcare, New York
-
Wen H. (2006). Adsorption at solid surfaces: pharmaceutical applications, in Encyclopedia of Pharmaceutical Technology, J., Swarbrick, ed. Informa Healthcare, New York, pp. 34-45
-
(2006)
Encyclopedia of Pharmaceutical Technology
, pp. 34-45
-
-
Wen, H.1
-
29
-
-
33747361036
-
The influence of PVP incorporation on moisture-induced surface crystallization of amorphous spray-dried lactose particles
-
DOI 10.1016/j.ijpharm.2006.05.016, PII S0378517306003838
-
Mahlin D, Berggren J, Gelius U, Engstri S, Alderborn G. (2006). The influence of PVP incorporation on moisture-induced surface crystallization of amorphous spray-dried lactose particles. Int J Pharm, 321:78-85 (Pubitemid 44247422)
-
(2006)
International Journal of Pharmaceutics
, vol.321
, Issue.1-2
, pp. 78-85
-
-
Mahlin, D.1
Berggren, J.2
Gelius, U.3
Engstrom, S.4
Alderborn, G.5
-
30
-
-
1142303337
-
What is the true solubility advantage for amorphous pharmaceuticals?
-
DOI 10.1023/A:1007516718048
-
Hancock BC, Parks M. (2000). What is the true solubility advantage for amorphous pharmaceuticals? Pharm Res, 17:397-404 (Pubitemid 30395293)
-
(2000)
Pharmaceutical Research
, vol.17
, Issue.4
, pp. 397-404
-
-
Hancock, B.C.1
Parks, M.2
|