Novel synthesis of some phthalazinone derivatives

Chinese Journal of Chemistry

Volumn 29, Issue 7, 2011, Pages 1446-1450

  Mahmoud, Mahmoud R ^a   Abou Elmagd, Wael S I ^a   Derbala, Hamed A ^a   Hekal, Mohamed H ^a  

^a Ain Shams University   (Egypt)

Author keywords

AM1 calculation; condensation; oxadiazole; phthalazinone carbohydrazide; triazolo oxadiazole

Indexed keywords

EID: 79960961022     PISSN: 1001604X     EISSN: 16147065     Source Type: Journal    
DOI: 10.1002/cjoc.201180264     Document Type: Article

References (33)

1. Al-assar, F.,;, Zelenin, K. N.,;, Lesiovskaya, E. E.,;, Benzhan, I. P.,;, Chakchir, B. A.,. Pharm. Chem. J., 2002, 36, 598.
2. Jain, R. P.,;, Vederas, J. C.,. Bioorg. Med. Chem. Lett., 2004, 14, 3655.
3. Carling, R. W.,;, Moore, K. W.,;, Street, L. J.,;, Wild, D.,;, Isted, C.,;, Lesson, P. D.,;, Thomas, S.,;, O'Conner, D.,;, Mckerman, R. M.,;, Quirk, K.,;, Cook, S. M.,;, Atack, J. R.,;, Wafttord, K. A.,;, Thompson, S. A.,;, Dawson, G. R.,;, Ferris, P.,;, Castor, J. L.,. J. Med. Chem., 2004, 47, 1807.
4. Grasso, S.,;, Desarro, G.,;, Micale, N.,;, Zappala, M.,;, Puia, G.,;, Baraldi, M.,;, Demicheli, C.,. J. Med. Chem., 2000, 43, 2851.
5. Kornet, M.,;, Shackleford, G.,. J. Heterocycl. Chem., 1999, 36, 1095.
6. Sivakumar, R.,;, Gnanasam, S. K.,;, Ramachandran, S.,;, Leonard, J. T.,. Eur. J. Med. Chem., 2002, 37, 793.
7. Nomoto, Y.,;, Obase, H.,;, Takai, H.,;, Teranishi, M.,;, Nakamura, J.,;, Kubo, K.,. Chem. Pharm. Bull. (TOKYO), 1990, 38, 2179.
8. Cockcrof, X.,;, Dillon, K. J.,;, Dixon, L.,;, Drzewiecki, J.,;, Everseley, P.,;, Gomes, S.,;, Hoare, J.,;, Kirrigan, F.,;, Nalthews, I.,;, Menear, K. A.,;, Martin, N. M.,;, Newton, R.,;, Paul, J.,;, Smith, G. C.,;, Vile, J.,;, Whittler, A. J.,. Bioorg. Med. Chem. Lett., 2006, 16, 1040.
9. Cockcrof, X.,;, Dillon, K. J.,;, Dixon, L.,;, Drzewiecki, J.,;, Kirrigan, F.,;, Loh, V. M.,;, Martin, N. M.,;, Menear, K. A.,;, Smith, G. C.,. Bioorg. Med. Chem. Lett., 2005, 15, 2235.
10. Kim, J. S.,;, Lee, H.,;, Suh, M.,;, Choo, H. P.,;, Lee, S. K.,;, Park, H. J.,;, Kim, C.,;, Park, S. W.,;, Lee, C.,. Bioorg. Med. Chem., 2004, 12, 3683.
11. Haider, N.,;, Kabicher, J.,;, Kaferbock, J.,;, Plenk, A.,. Molecules, 2007, 12, 1900.
12. Demirayak, S.,;, Karaburun, K.,;, Beis, R.,. Eur. J. Med. Chem., 2004, 39, 1089.
13. Goodman and Gilman's, 11 th ed., Mc Graw-Hill Medical Publishing Division, New York, 2006, p. 860.
14. Watanabe, N.,;, Kabasawa, Y.,;, Takase, Y.,;, Matsukura, M.,;, Miyazaki, K.,;, Ishihara, H.,;, Kodama, K.,;, Adachi, H.,. J. Med. Chem., 1998, 41, 3367.
15. Johnsen, M.,;, Rehese, K.,;, Pertz, H.,;, Stasch, J.,;, Bischoff, E.,. Arch. Pharm. (Weinheim), 2003, 336, 591.
16. Madhavan, G. R.,;, Chakrabarti, R.,;, Kumar, S. K.,;, Misra, P.,;, Mamidi, R. N.,;, Balarzu, V.,;, ksiram, K.,;, Babu, R. K.,;, Suresh, J.,;, Lohray, B. B.,;, Lohray, V. B.,;, Iqbal, J.,;, Raiagopalan, R.,. Eur. J. Med. Chem., 2001, 36, 627.
17. Lenz, E. M.,;, Wilson, I. D.,;, Wright, B.,;, Partidge, E. A.,;, Rodgers, C. T.,;, Haycock, P. R.,;, Lindon, J. C.,;, Nicholson, J. K.,. J. Pharm. Biomed. Anal., 2002, 28, 31.
18. Cardia, M. C.,;, Distinto, E.,;, Maccioni, E.,;, Delogu, A.,. J. Heterocycl. Chem., 2003, 40, 1011.
19. Shetgiri, N. P.,;, Nayak, B. N.,. Ind. J. Chem., 2005, 448, 1267.
20. Dogruer, D. S.,;, Kupeli, E.,;, Yesilada, E.,;, Sahin, M. F.,. Arch. Pharm. (Weinheim), 2004, 337, 303.
21. Napoletano, M.,;, Norcini, G.,;, Pellacini, F.,;, Marchini, F.,;, Moraazzoni, G.,;, Ferlenga, P.,;, Peradella, L.,. Bioorg. Med. Chem. Lett., 2000, 10, 2235.
22. Van der Mey, M.,;, Hatzelmann, A.,;, Vanklink, G. B.,;, Van der Lann, I. J.,;, Sterk, G. J.,;, THibaut, U.,;, Timmerman, H.,. J. Med. Chem., 2001, 44, 2511.
23. Van der Mey, M.,;, Hildgard, B.,;, Dennis, G.,;, Hatzelmann, A.,;, Timmerman, H.,. J. Med. Chem., 2002, 45, 2526.
24. Shubin, K. M.,;, Kuznetsov, V. A.,;, Galishev, V. A.,. Tetrahedron Lett., 2004, 45, 1407.
25. Brad, H.,;, Qiang, G.,;, Partha, P. C.,;, Games, R. F.,;, Liping, P.,;, Robert, M. R.,;, Anthony, B. R.,;, Andreas, R.,;, Kelvin, S.,;, Maya, T.,;, Ryan, P. W.,;, Shimin, X.,;, Dawei, Z.,;, Faye, H.,;, Matthew, R. L.,;, Rashed, S.,;, Vivian, L.,;, David, G.,;, Matthew, H. P.,;, Bradley, H.,;, Lisa, S.,;, Scot, M.,;, Lu, M. W.,;, Andrew, S. T.,. J. Med. Chem., 2008, 51, 6271.
26. Kim, J. S.,;, Lee, H. J.,;, Suh, M. E.,. Bioorg. Med. Chem., 2004, 12, 3683.
27. Chakraborti, A. K.,;, Gopalakrishnan, B.,;, Sobbia, E.,;, Malde, A.,. Bioorg. Med. Chem. Lett., 2003, 13, 2473.
28. Duncton, M. A.,;, Piatnitski, E. L.,;, Katoch-Rouse, R.,. Bioorg. Med. Chem. Lett., 2006, 16, 1579.
29. Hwang, J. Y.,;, Choi, H. S.,;, Gong, Y. D.,. Tetrahedron Lett., 2005, 46, 3107.
30. Mahmoud, M. R.,;, El-Shahawi, M. M.,;, El-Bordany, E. A.,;, Abu El-Azm, F. S. M.,. Synth. Commun., 2010, 40, 666.
31. Mahmoud, M. R.,;, El-Shahawi, M. M.,;, El-Bordany, E. A.,;, Abu El-Azm, F. S. M.,. Eur. J. Chem., 2010, 1(2), 134.
32. Dewar, M. J.,;, Zobisch, E.,;, Healy, E. F.,;, Stewart, J. P.,. J. Am. Chem. Soc., 1985, 107, 3902.
33. Mahmoud, M. R.,;, El-Bordany, E. A.,;, Hassan, N. F.,;, Abu El-Azm, F. S. M.,. Phosphorus, Sulfur, Silicon, 2007, 182, 2507.