Thiomers: Inhibition of cytochrome P450 activity

European Journal of Pharmaceutics and Biopharmaceutics

Volumn 78, Issue 3, 2011, Pages 361-365

  Iqbal, Javed ^a   Sakloetsakun, Duangkamon ^b   Bernkop Schnürch, Andreas ^a  

^a UNIVERSITY OF INNSBRUCK   (Austria)

^b KHON KAEN UNIVERSITY   (Thailand)

Author keywords

CYP2A6; CYP3A4; Cytochrome P450; Fluorescent probe assays; Inhibition; Thiomers

Indexed keywords

CHITOSAN; COUMARIN DERIVATIVE; CYSTEINE; CYTOCHROME P450 2A6; CYTOCHROME P450 3A4; CYTOCHROME P450 INHIBITOR; MACROGOL; MACROGOL STEARATE; POLIDOCANOL; POLYACRYLIC ACID; POLYETHYLENE; POLYMER; THIOGLYCOLIC ACID; UMBELLIFERONE; VERAPAMIL;

ARTICLE; CATALYSIS; CONTROLLED STUDY; DRUG BIOAVAILABILITY; DRUG SCREENING; ENZYME ACTIVITY; ENZYME ASSAY; ENZYME INHIBITION; FLUORESCENCE; HUMAN; HUMAN CELL; IC 50; LOOSE FECES; METABOLISM;

ARYL HYDROCARBON HYDROXYLASES; CHITOSAN; COUMARINS; CYSTEINE; CYTOCHROME P-450 CYP3A; CYTOCHROME P-450 ENZYME SYSTEM; DRUG CARRIERS; DRUG COMPOUNDING; DRUG DELIVERY SYSTEMS; ENZYME ASSAYS; ENZYME INHIBITORS; EXCIPIENTS; INDICATORS AND REAGENTS; POLYMERS; SULFHYDRYL COMPOUNDS; VERAPAMIL;

EID: 79960571701     PISSN: 09396411     EISSN: 18733441     Source Type: Journal    
DOI: 10.1016/j.ejpb.2011.02.017     Document Type: Article

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