Inhibition of coumarin 7-hydroxylase activity in human liver microsomes

Archives of Biochemistry and Biophysics

Volumn 341, Issue 1, 1997, Pages 47-61

  Draper, Alison J ^a   Madan, Ajay ^a   Parkinson, Andrew ^a  

^a UNIVERSITY OF KANSAS SCHOOL OF MEDICINE   (United States)

Author keywords

CYP2A6, chemical inhibition of coumarin 7 hydroxylation; cytochrome P450, chemical inhibition; inhibition of human coumarin 7 hydroxylase

Indexed keywords

CAFFEINE; CHLORZOXAZONE; CIMETIDINE; COUMARIN; DEXTROMETHORPHAN; DIAZEPAM; DIOXANE DERIVATIVE; ELLIPTICINE; FLUCONAZOLE; HEXOBARBITAL; KETOCONAZOLE; MEPHENYTOIN; MICONAZOLE; NICOTINE; OXYGENASE; PAPAVERINE; PHENACETIN; QUINIDINE; SPIRONOLACTONE; TETRAHYDROFURAN; THIAMAZOLE; TOLBUTAMIDE; TRANYLCYPROMINE; TROLEANDOMYCIN;

ARTICLE; BIOTRANSFORMATION; COMPETITIVE INHIBITION; DRUG METABOLISM; DRUG OVERDOSE; ENZYME ACTIVITY; ENZYME INHIBITION; ENZYME SPECIFICITY; HUMAN; HUMAN TISSUE; HYDROXYLATION; IMMUNOREACTIVITY; LIVER MICROSOME; PRIORITY JOURNAL; XENOBIOTIC METABOLISM;

EID: 0031149716     PISSN: 00039861     EISSN: None     Source Type: Journal    
DOI: 10.1006/abbi.1997.9964     Document Type: Article

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