Tryptamine derivatives as novel non-nucleosidic inhibitors against hepatitis B virus

Bioorganic and Medicinal Chemistry

Volumn 19, Issue 10, 2011, Pages 3120-3127

  Qu, Shi Jin ^a   Wang, Gui Feng ^a   Duan, Wen Hu ^a   Yao, Shan Yan ^a   Zuo, Jian Ping ^a   Tan, Chang Heng ^a   Zhu, Da Yuan ^a  

^a SHANGHAI INSTITUTE OF MATERIA MEDICA   (China)

Author keywords

Anti HBV activity; Non nucleosidic inhibitors; Tryptamine derivatives

Indexed keywords

5 CHLORO N,N DIMETHYLTRYPTAMINE N12 OXIDE; COTRIMOXAZOLE; LAMIVUDINE; N,N BIS(2,4,5 TRIMETHOXYBENZYL)TRYPTAMINE; N,N BIS(3 NITROBENZYL)TRYPTAMINE; N,N BIS(FURAN 2 YL METHYL)TRYPTAMINE; N,N BIS(FURAN 2 YL METHYL)TRYPTAMINE N12 OXIDE; N,N BIS(PYRIDIN 2 YL METHYL)TRYPTAMINE; N,N BIS(PYRIDIN 2 YL METHYL)TRYPTAMINE N12 OXIDE; N,N BIS(THIOPHEN 2 YL METHYL)TRYPTAMINE; N,N BIS(THIOPHEN 2 YL METHYL)TRYPTAMINE N12 OXIDE; N,N DIBENZYLTRYPTAMINE; N,N DIBENZYLTRYPTAMINE N12 OXIDE; N,N DICYCLOHEXYLMETHYLTRYPTAMINE; N,N DICYCLOHEXYLMETHYLTRYPTAMINE N12 OXIDE; N,N DICYCLOPROPYLMETHYLTRYPTAMINE; N,N DICYCLOPROPYLMETHYLTRYPTAMINE N12 OXIDE; N,N DIETHYLTRYPTAMINE; N,N DIETHYLTRYPTAMINE N12 OXIDE; N,N DIISOBUTYLTRYPTAMINE; N,N DIISOBUTYLTRYPTAMINE N12 OXIDE; N,N DIISOPENTYLTRYPTAMINE; N,N DIISOPENTYLTRYPTAMINE N12 OXIDE; N,N DIMETHYLTRYPTAMINE; N,N DIMETHYLTRYPTAMINE N12 OXIDE; N,N DIPROPYLTRYPTAMINE; N,N DIPROPYLTRYPTAMINE N12 OXIDE; N12 ISOPENTYLTRYPTAMINE; TRYPTAMINE DERIVATIVE; UNCLASSIFIED DRUG; UNINDEXED DRUG;

ALKYLATION; ANTIVIRAL ACTIVITY; ARTICLE; CARBON NUCLEAR MAGNETIC RESONANCE; CONTROLLED STUDY; CYTOTOXICITY; DRUG POTENCY; DRUG STRUCTURE; DRUG SYNTHESIS; HEPATITIS B VIRUS; HUMAN; HUMAN CELL; IC 50; OXIDATION; PROTON NUCLEAR MAGNETIC RESONANCE; STRUCTURE ACTIVITY RELATION;

ANTIVIRAL AGENTS; CELL SURVIVAL; DNA, VIRAL; HEP G2 CELLS; HEPATITIS B; HEPATITIS B VIRUS; HUMANS; STRUCTURE-ACTIVITY RELATIONSHIP; TRYPTAMINES;

HEPATITIS B VIRUS;

EID: 79956197917     PISSN: 09680896     EISSN: 14643391     Source Type: Journal    
DOI: 10.1016/j.bmc.2011.04.004     Document Type: Article

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