N1-benzenesulfonylgramine and N 1-benzenesulfonylskatole: Novel 5-HT6 receptor ligand templates

Bioorganic and Medicinal Chemistry Letters

Volumn 13, Issue 19, 2003, Pages 3355-3359

  Pullagurla, Manik R ^a   Dukat, Małgorzata ^a   Setola, Vincent ^b   Roth, Bryan ^b   Glennon, Richard A ^a  

^a VIRGINIA COMMONWEALTH UNIVERSITY   (United States)

^b CASE WESTERN RESERVE UNIVERSITY SCHOOL OF MEDICINE   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

1 BENZENESULFONYLGRAMINE; AMINOBENZENESULFONYLSKATOLE; SEROTONIN ANTAGONIST; UNCLASSIFIED DRUG;

ARTICLE; CELL STRAIN; CONTROLLED STUDY; DRUG ACTIVITY; DRUG DETERMINATION; DRUG INHIBITION; DRUG RECEPTOR BINDING; HUMAN; HUMAN CELL; IC 50; STRUCTURE ACTIVITY RELATION;

EID: 0042781556     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(03)00612-7     Document Type: Article

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