-
1
-
-
33749431861
-
Amorphization of indomethacin by co-grinding with neusilin US2: Amorphization kinetics, physical stability and mechanism
-
Bahl D, Bogner RH. 2006. Amorphization of indomethacin by co-grinding with neusilin US2: Amorphization kinetics, physical stability and mechanism. Pharm Res 23(10):2317-2325.
-
(2006)
Pharm Res
, vol.23
, Issue.10
, pp. 2317-2325
-
-
Bahl, D.1
Bogner, R.H.2
-
2
-
-
66249101601
-
Solubility advantage of pharmaceutical cocrystals
-
Good DJ, Rodriguez-Hornedo N. 2009. Solubility advantage of pharmaceutical cocrystals. Cryst Growth Des 9(5):2252-2264.
-
(2009)
Cryst Growth Des
, vol.9
, Issue.5
, pp. 2252-2264
-
-
Good, D.J.1
Rodriguez-Hornedo, N.2
-
3
-
-
0035157406
-
Polymorph screening: Influence of solvents on the rate of solvent-mediated polymorphic transformation
-
Gu C-H, Young V, Jr., Grant DJW. 2001. Polymorph screening: Influence of solvents on the rate of solvent-mediated polymorphic transformation. J Pharm Sci 90(11):1878-1890.
-
(2001)
J Pharm Sci
, vol.90
, Issue.11
, pp. 1878-1890
-
-
Gu, C.-H.1
Young Jr, V.2
Grant, D.J.W.3
-
4
-
-
0030638567
-
Characteristics and significance of the amorphous state in pharmaceutical systems
-
Hancock BC, Zografi G. 1997. Characteristics and significance of the amorphous state in pharmaceutical systems. J Pharm Sci 86(1):1-12.
-
(1997)
J Pharm Sci
, vol.86
, Issue.1
, pp. 1-12
-
-
Hancock, B.C.1
Zografi, G.2
-
5
-
-
76649105411
-
Solubility advantage of amorphous pharmaceuticals: I. A thermodynamic analysis
-
Murdande SB, Pikal MJ, Shanker RM, Bogner RH. 2010. Solubility advantage of amorphous pharmaceuticals: I. A thermodynamic analysis. J Pharm Sci 99(3):1254-1264.
-
(2010)
J Pharm Sci
, vol.99
, Issue.3
, pp. 1254-1264
-
-
Murdande, S.B.1
Pikal, M.J.2
Shanker, R.M.3
Bogner, R.H.4
-
6
-
-
20344391910
-
Trends in solubility of polymorphs
-
Pudipeddi M, Serajuddin ATM. 2005. Trends in solubility of polymorphs. J Pharm Sci 94(5):929-939.
-
(2005)
J Pharm Sci
, vol.94
, Issue.5
, pp. 929-939
-
-
Pudipeddi, M.1
Serajuddin, A.T.M.2
-
7
-
-
34548032742
-
Salt formation to improve drug solubility
-
Serajuddin ATM. 2007. Salt formation to improve drug solubility. Adv Drug Deliv Rev 59(7):603-616.
-
(2007)
Adv Drug Deliv Rev
, vol.59
, Issue.7
, pp. 603-616
-
-
Serajuddin, A.T.M.1
-
9
-
-
1542410398
-
Ritonavir-PEG 8000 amorphous solid dispersions: In vitro and in vivo evaluations
-
Law D, Schmitt EA, Marsh KC, Everitt EA, Wang W, Fort JJ, Krill SL, Qiu Y. 2004. Ritonavir-PEG 8000 amorphous solid dispersions: In vitro and in vivo evaluations. J Pharm Sci 93(3):563-570.
-
(2004)
J Pharm Sci
, vol.93
, Issue.3
, pp. 563-570
-
-
Law, D.1
Schmitt, E.A.2
Marsh, K.C.3
Everitt, E.A.4
Wang, W.5
Fort, J.J.6
Krill, S.L.7
Qiu, Y.8
-
10
-
-
23844499379
-
IV-IVC considerations in the development of immediate-release oral dosage form
-
Li S, He H, Parthiban LJ, Yin H, Serajuddin ATM. 2005. IV-IVC considerations in the development of immediate-release oral dosage form. J Pharm Sci 94(7):1396-1417.
-
(2005)
J Pharm Sci
, vol.94
, Issue.7
, pp. 1396-1417
-
-
Li, S.1
He, H.2
Parthiban, L.J.3
Yin, H.4
Serajuddin, A.T.M.5
-
11
-
-
0034607382
-
Salt form selection and characterization of LY333531 mesylate monohydrate
-
Engel GL, Farid NA, Faul MM, Richardson LA, Winneroski LL. 2000. Salt form selection and characterization of LY333531 mesylate monohydrate. Int J Pharm 198(2):239-247.
-
(2000)
Int J Pharm
, vol.198
, Issue.2
, pp. 239-247
-
-
Engel, G.L.1
Farid, N.A.2
Faul, M.M.3
Richardson, L.A.4
Winneroski, L.L.5
-
12
-
-
5444250003
-
Oral absorption and pharmacokinetics of rebamipide and rebamipide lysinate in rats
-
Shin BS, Kim CH, Jun YS, Yoon CH, Rho JI, Lee KC, Han HS, Yoo SD. 2004. Oral absorption and pharmacokinetics of rebamipide and rebamipide lysinate in rats. Drug Dev Ind Pharm 30(8):869-876.
-
(2004)
Drug Dev Ind Pharm
, vol.30
, Issue.8
, pp. 869-876
-
-
Shin, B.S.1
Kim, C.H.2
Jun, Y.S.3
Yoon, C.H.4
Rho, J.I.5
Lee, K.C.6
Han, H.S.7
Yoo, S.D.8
-
13
-
-
0037406422
-
Dissolution behavior of a poorly water soluble compound in the presence of Tween 80
-
Chen LR, Wesley JA, Bhattachar S, Ruiz B, Bahash K, Babu SR. 2003. Dissolution behavior of a poorly water soluble compound in the presence of Tween 80. Pharm Res 20(5):797-801.
-
(2003)
Pharm Res
, vol.20
, Issue.5
, pp. 797-801
-
-
Chen, L.R.1
Wesley, J.A.2
Bhattachar, S.3
Ruiz, B.4
Bahash, K.5
Babu, S.R.6
-
14
-
-
0033403992
-
Tablet dissolution affected by a moisture mediated solid-state interaction between drug and disintegrant
-
Rohrs BR, Thamann TJ, Gao P, Stelzer DJ, Bergren MS, Chao RS. 1999. Tablet dissolution affected by a moisture mediated solid-state interaction between drug and disintegrant. Pharm Res 16(12):1850-1856.
-
(1999)
Pharm Res
, vol.16
, Issue.12
, pp. 1850-1856
-
-
Rohrs, B.R.1
Thamann, T.J.2
Gao, P.3
Stelzer, D.J.4
Bergren, M.S.5
Chao, R.S.6
-
16
-
-
0029559913
-
Dissolution kinetics and solubilities of p-aminosalicylic acid and its salts
-
Forbes RT, York P, Davidson JR. 1995. Dissolution kinetics and solubilities of p-aminosalicylic acid and its salts. Int J Pharm 126(1, 2):199-208.
-
(1995)
Int J Pharm
, vol.126
, Issue.1-2
, pp. 199-208
-
-
Forbes, R.T.1
York, P.2
Davidson, J.R.3
-
17
-
-
0001266165
-
The kinetics of solvent-mediated phase transformations. Proc Royal Soc London, Ser A: Math
-
Cardew PT, Davey RJ. 1985. The kinetics of solvent-mediated phase transformations. Proc Royal Soc London, Ser A: Math. Phys Eng Sci 398(1815):415-428.
-
(1985)
Phys Eng Sci
, vol.398
, Issue.1815
, pp. 415-428
-
-
Cardew, P.T.1
Davey, R.J.2
-
18
-
-
33846212349
-
In situ measurement of solvent-mediated phase transformations during dissolution testing
-
Aaltonen J, Heinanen P, Peltonen L, Korteiarvi H, Tanninen VP, Christiansen L, Hirvonen J, Yliruusi J, Rantanen J. 2006. In situ measurement of solvent-mediated phase transformations during dissolution testing. J Pharm Sci 95(12):2730-2737.
-
(2006)
J Pharm Sci
, vol.95
, Issue.12
, pp. 2730-2737
-
-
Aaltonen, J.1
Heinanen, P.2
Peltonen, L.3
Korteiarvi, H.4
Tanninen, V.P.5
Christiansen, L.6
Hirvonen, J.7
Yliruusi, J.8
Rantanen, J.9
-
19
-
-
1642457353
-
Use of glancing angle X-Ray powder diffractometry to depth-profile phase transformations during dissolution of indomethacin and theophylline tablets
-
Debnath S, Predecki P, Suryanarayanan R. 2004. Use of glancing angle X-Ray powder diffractometry to depth-profile phase transformations during dissolution of indomethacin and theophylline tablets. Pharm Res 21(1):149-159.
-
(2004)
Pharm Res
, vol.21
, Issue.1
, pp. 149-159
-
-
Debnath, S.1
Predecki, P.2
Suryanarayanan, R.3
-
20
-
-
0037057317
-
Solution-mediated phase transformation of anhydrous to dihydrate carbamazepine and the effect of lattice disorder
-
Murphy D, Rodriguez-Cintron F, Langevin B, Kelly RC, Rodriguez-Hornedo N. 2002. Solution-mediated phase transformation of anhydrous to dihydrate carbamazepine and the effect of lattice disorder. Int J Pharm 246(1-2):121-134.
-
(2002)
Int J Pharm
, vol.246
, Issue.1-2
, pp. 121-134
-
-
Murphy, D.1
Rodriguez-Cintron, F.2
Langevin, B.3
Kelly, R.C.4
Rodriguez-Hornedo, N.5
-
21
-
-
0026699429
-
Phase transition and heterogeneous/epitaxial nucleation of hydrated and anhydrous theophylline crystals
-
Rodriguez-Hornedo N, Lechuga-Ballesteros D, Wu HJ. 1992. Phase transition and heterogeneous/epitaxial nucleation of hydrated and anhydrous theophylline crystals. Int J Pharm 85(1-3):149-162.
-
(1992)
Int J Pharm
, vol.85
, Issue.1-3
, pp. 149-162
-
-
Rodriguez-Hornedo, N.1
Lechuga-Ballesteros, D.2
Wu, H.J.3
-
22
-
-
0842332474
-
Surfactant-facilitated crystallization of dihydrate carbamazepine during dissolution of anhydrous polymorph
-
Rodriguez-Hornedo N, Murphy D. 2004. Surfactant-facilitated crystallization of dihydrate carbamazepine during dissolution of anhydrous polymorph. J Pharm Sci 93(2):449-460.
-
(2004)
J Pharm Sci
, vol.93
, Issue.2
, pp. 449-460
-
-
Rodriguez-Hornedo, N.1
Murphy, D.2
-
23
-
-
0344603644
-
Significance of controlling crystallization mechanisms and kinetics in pharmaceutical systems
-
Rodriguez-Hornedo N, Murphy D. 1999. Significance of controlling crystallization mechanisms and kinetics in pharmaceutical systems. J Pharm Sci 88(7):651-660.
-
(1999)
J Pharm Sci
, vol.88
, Issue.7
, pp. 651-660
-
-
Rodriguez-Hornedo, N.1
Murphy, D.2
-
24
-
-
37349115571
-
Trends in active pharmaceutical ingredient salt selection based on analysis of the orange book database
-
Paulekuhn GS, Dressman JB, Saal C. 2007. Trends in active pharmaceutical ingredient salt selection based on analysis of the orange book database. J Med Chem 50(26):6665-6672.
-
(2007)
J Med Chem
, vol.50
, Issue.26
, pp. 6665-6672
-
-
Paulekuhn, G.S.1
Dressman, J.B.2
Saal, C.3
-
25
-
-
0003460950
-
-
Janicki CA, Ko CY, Eds.. New York: Academic Press.
-
Janicki CA, Ko CY, Eds. 1980. Analytical profiles of drug substances. New York: Academic Press.
-
(1980)
Analytical profiles of drug substances
-
-
-
26
-
-
23844475290
-
Effect of chloride ion on dissolution of different salt forms of haloperidol, a model basic drug
-
Li S, Doyle P, Metz S, Royce AE, Serajuddin ATM. 2005. Effect of chloride ion on dissolution of different salt forms of haloperidol, a model basic drug. J Pharm Sci 94(10):2224-2231.
-
(2005)
J Pharm Sci
, vol.94
, Issue.10
, pp. 2224-2231
-
-
Li, S.1
Doyle, P.2
Metz, S.3
Royce, A.E.4
Serajuddin, A.T.M.5
-
27
-
-
18044381309
-
Investigation of solubility and dissolution of a free base and two different salt forms as a function of pH
-
Li S, Wong S, Sethia S, Almoazen H, Joshi YM, Serajuddin ATM. 2005. Investigation of solubility and dissolution of a free base and two different salt forms as a function of pH. Pharm Res 22(4):628-635.
-
(2005)
Pharm Res
, vol.22
, Issue.4
, pp. 628-635
-
-
Li, S.1
Wong, S.2
Sethia, S.3
Almoazen, H.4
Joshi, Y.M.5
Serajuddin, A.T.M.6
-
28
-
-
77957730547
-
-
USA: (USA), U.S. Patent 2,008,013,8261, June 12, 2008.
-
Bogner RH, Bergman TL, Greco K, Michaels DJ, Chawarski SJ. 2008. Flow-through apparatus for microscopic investigation of dissolution of pharmaceutical solids. USA: (USA), U.S. Patent 2, 008, 013, 8261, June 12, 2008.
-
(2008)
Flow-through apparatus for microscopic investigation of dissolution of pharmaceutical solids
-
-
Bogner, R.H.1
Bergman, T.L.2
Greco, K.3
Michaels, D.J.4
Chawarski, S.J.5
-
29
-
-
77957741630
-
Design and characterization of a laminar flow-through dissolution apparatus: Comparison of hydrodynamic conditions to those of common dissolution techniques
-
Greco K, Bergman TL, Bogner R. Design and characterization of a laminar flow-through dissolution apparatus: Comparison of hydrodynamic conditions to those of common dissolution techniques. Pharmaceutical Development and Technology. 16(1):75-87.
-
Pharmaceutical Development and Technology
, vol.16
, Issue.1
, pp. 75-87
-
-
Greco, K.1
Bergman, T.L.2
Bogner, R.3
-
30
-
-
0016835216
-
Evaluation of a convective diffusion drug dissolution rate model
-
Shah AC, Nelson KG. 1975. Evaluation of a convective diffusion drug dissolution rate model. J Pharm Sci 64(9):1518-1520.
-
(1975)
J Pharm Sci
, vol.64
, Issue.9
, pp. 1518-1520
-
-
Shah, A.C.1
Nelson, K.G.2
-
31
-
-
23844516181
-
A Novel in vitro and numerical analysis of shear-induced drug release from extended-release tablets in the fed stomach
-
Abrahamsson B, Pal A, Sjoeberg M, Carlsson M, Laurell E, Brasseur JG. 2005. A Novel in vitro and numerical analysis of shear-induced drug release from extended-release tablets in the fed stomach. Pharm Res 22(8):1215-1226.
-
(2005)
Pharm Res
, vol.22
, Issue.8
, pp. 1215-1226
-
-
Abrahamsson, B.1
Pal, A.2
Sjoeberg, M.3
Carlsson, M.4
Laurell, E.5
Brasseur, J.G.6
-
32
-
-
16644369504
-
Gastric flow and mixing studied using computer simulation
-
Pal A, Indireshkumar K, Schwizer W, Abrahamsson B, Fried M, Brasseur JG. 2004. Gastric flow and mixing studied using computer simulation. Proc Biol Sci 271(1557):2587-2594.
-
(2004)
Proc Biol Sci
, vol.271
, Issue.1557
, pp. 2587-2594
-
-
Pal, A.1
Indireshkumar, K.2
Schwizer, W.3
Abrahamsson, B.4
Fried, M.5
Brasseur, J.G.6
-
34
-
-
0031171011
-
Numerical simulations of laminar flow over a 3D backward-facing step
-
Williams PT, Baker AJ. 1997. Numerical simulations of laminar flow over a 3D backward-facing step. Int J Numer Methods Fluids 24(11):1159-1183.
-
(1997)
Int J Numer Methods Fluids
, vol.24
, Issue.11
, pp. 1159-1183
-
-
Williams, P.T.1
Baker, A.J.2
-
35
-
-
0004012624
-
-
Prentice Hall: Upper Saddle River, New Jersey
-
Levich VG. 1962. Physicochemical hydrodynamics. Prentice Hall: Upper Saddle River, New Jersey, pp 60-78.
-
(1962)
Physicochemical hydrodynamics
, pp. 60-78
-
-
Levich, V.G.1
-
36
-
-
0035795769
-
Weak interactions involving organic fluorine: Analysis of structural motifs in flunarizine and haloperidol
-
Prasanna MD, Row TNG. 2001. Weak interactions involving organic fluorine: Analysis of structural motifs in flunarizine and haloperidol. J Mol Struct 562(1-3):55-61.
-
(2001)
J Mol Struct
, vol.562
, Issue.1-3
, pp. 55-61
-
-
Prasanna, M.D.1
Row, T.N.G.2
-
37
-
-
0022533161
-
Dissolution of acidic and basic compounds from the rotating disk: Influence of convective diffusion and reaction
-
McNamara DP, Amidon GL. 1986. Dissolution of acidic and basic compounds from the rotating disk: Influence of convective diffusion and reaction. J Pharm Sci 75(9):858-868.
-
(1986)
J Pharm Sci
, vol.75
, Issue.9
, pp. 858-868
-
-
McNamara, D.P.1
Amidon, G.L.2
-
38
-
-
0019365865
-
Dissolution kinetics of carboxylic acids. I: Effect of pH under unbuffered conditions
-
Mooney KG, Mintun MA, Himmelstein KJ, Stella VJ. 1981. Dissolution kinetics of carboxylic acids. I: Effect of pH under unbuffered conditions. J Pharm Sci 70(1):13-22.
-
(1981)
J Pharm Sci
, vol.70
, Issue.1
, pp. 13-22
-
-
Mooney, K.G.1
Mintun, M.A.2
Himmelstein, K.J.3
Stella, V.J.4
-
39
-
-
0019350675
-
Dissolution kinetics of carboxylic acids. II: Effects of buffers
-
Mooney KG, Mintun MA, Himmelstein KJ, Stella VJ. 1981. Dissolution kinetics of carboxylic acids. II: Effects of buffers. J Pharm Sci 70(1):22-32.
-
(1981)
J Pharm Sci
, vol.70
, Issue.1
, pp. 22-32
-
-
Mooney, K.G.1
Mintun, M.A.2
Himmelstein, K.J.3
Stella, V.J.4
-
40
-
-
68149179817
-
Powder dissolution method for estimating rotating disk intrinsic dissolution rates of low solubility drugs
-
Tsinman K, Avdeef A, Tsinman O, Voloboy D. 2009. Powder dissolution method for estimating rotating disk intrinsic dissolution rates of low solubility drugs. Pharm Res 26(9):2093-2100.
-
(2009)
Pharm Res
, vol.26
, Issue.9
, pp. 2093-2100
-
-
Tsinman, K.1
Avdeef, A.2
Tsinman, O.3
Voloboy, D.4
-
41
-
-
48549084486
-
Measurement of surface pH of pharmaceutical solids: A critical evaluation of indicator dye-sorption method and its comparison with slurry pH method
-
Pudipeddi M, Zannou EA, Vasanthavada M, Dontabhaktuni A, Royce AE, Joshi YM, Serajuddin ATM. 2008. Measurement of surface pH of pharmaceutical solids: A critical evaluation of indicator dye-sorption method and its comparison with slurry pH method. J Pharm Sci 97(5):1831-1842.
-
(2008)
J Pharm Sci
, vol.97
, Issue.5
, pp. 1831-1842
-
-
Pudipeddi, M.1
Zannou, E.A.2
Vasanthavada, M.3
Dontabhaktuni, A.4
Royce, A.E.5
Joshi, Y.M.6
Serajuddin, A.T.M.7
|