Prolonged intragastric drug delivery mediated by eudragit® E-carrageenan polyelectrolyte matrix tablets

AAPS PharmSciTech

Volumn 12, Issue 1, 2011, Pages 354-361

  Bani Jaber, Ahmad ^a   Al Aani, Leena ^a   Alkhatib, Hatim ^a   Al Khalidi, Bashar ^a  

^a UNIVERSITY OF JORDAN   (Jordan)

Author keywords

carrageenan; Eudragit E; gastric retention; polyelectrolyte complexation

Indexed keywords

BICARBONATE; CARRAGEENAN; EUDRAGIT; METRONIDAZOLE; POLYELECTROLYTE;

ARTICLE; COMPLEX FORMATION; CONTROLLED DRUG RELEASE; DRUG DELIVERY SYSTEM; DRUG SOLUBILITY; EFFERVESCENT TABLET; IN VITRO STUDY; MATRIX TABLET; PRIORITY JOURNAL; VISCOSITY;

ADMINISTRATION, ORAL; ANTI-INFECTIVE AGENTS; CARRAGEENAN; DELAYED-ACTION PREPARATIONS; DIFFUSION; DRUG CARRIERS; DRUG COMPOUNDING; DRUG DELIVERY SYSTEMS; EXCIPIENTS; HUMANS; METRONIDAZOLE; POLYMERS; POLYMETHACRYLIC ACIDS; SOLUBILITY; STOMACH; STOMACH DISEASES; VISCOSITY;

EID: 79954424921     PISSN: None     EISSN: 15309932     Source Type: Journal    
DOI: 10.1208/s12249-011-9595-0     Document Type: Article

References (23)

1. MV Risbud AA Hardikar SV Bhat RR Bhonde 2000 pH-sensitive freeze-dried chitosan-polyvinyl pyrrolidone hydrogels as controlled release system for antibiotic delivery J Control Release 68 23 30 10884576 10.1016/S0168-3659(00) 00208-X 1:CAS:528:DC%2BD3cXksV2ltb4%3D (Pubitemid 30407059)
2. S Burton N Washington RJ Steele R Musson L Feely 1995 Intragastric distribution of ion-exchange resins: a drug delivery system for the topical treatment of the gastric mucosa J Pharm Pharmacol 47 901 906 8708983 1:CAS:528:DyaK28XnslGlsw%3D%3D (Pubitemid 26020148)
3. Y Wu R Fassihi 2005 Stability of metronidazole, tetracycline hcl and famotidine alone and in combination Int J Pharm 290 1 13 15664125 10.1016/j.ijpharm.2004.10.015 1:CAS:528:DC%2BD2MXkvVSlug%3D%3D (Pubitemid 40139039)
4. G Santus C Lazzarini G Bottoni EP Sandefer RC Page WJ Doll UY Ryo GA Digenis 1997 An in vitro-in vivo investigation of oral bioadhesive controlled release furosemide formulations Eur J Pharm Biopharm 44 39 52 10.1016/S0939-6411(97)00100-8 1:CAS:528:DyaK2sXmtFShtrs%3D (Pubitemid 28298774)
5. AA Deshpande CT Rhodes NH Shah AW Malick 1996 Controlled-release drug delivery systems for prolonged gastric residence: an overview Drug Dev Ind Pharm 22 531 539 10.3109/03639049609108355 1:CAS:528:DyaK28XjtlWqt7c%3D (Pubitemid 26197851)
6. AA Deshpande NH Shah CT Rhodes AW Malick 1997 Development of a novel controlled-release system for gastric retention Pharm Res 14 815 819 9210203 10.1023/A:1012171010492 1:CAS:528:DyaK2sXkt1yitLY%3D (Pubitemid 27281680)
7. A Menon WA Ritschel A Sakr 1994 Development and evaluation of a monolithic floating dosage form for furosemide J Pharm Sci 83 239 245 8169797 10.1002/jps.2600830225 1:CAS:528:DyaK2cXmt1WqsA%3D%3D (Pubitemid 24224185)
8. L Whitehead JT Fell JH Collett HL Sharma AM Smith 1998 Floating dosage forms: an in vivo study demonstrating prolonged gastric retention J Control Release 55 3 12 9795000 10.1016/S0168-3659(97)00266-6 1:CAS:528: DyaK1cXmslWjsr0%3D (Pubitemid 28477559)
9. MN Gambhire KW Ambade SD Kurmi VJ Kadam KR Jadhav 2007 Development and in vitro evaluation of an oral floating matrix tablet formulation of diltiazem hydrochloride AAPS PharmSciTech 8 E73 17915823 10.1208/pt0803073
10. S Li S Lin YW Chien BP Daggy HL Mirchandani 2001 Statistical optimization of gastric floating system for oral controlled delivery of calcium AAPS PharmSciTech 2 E1 14727887 10.1208/pt020101 1:STN:280:DC%2BD2c%2FivVOqtg%3D%3D
11. G Xu MJ Groves 2001 Effect of FITC-dextran molecular weight on its release from floating cetyl alcohol and HPMC tablets J Pharm Pharmacol 53 49 56 11206192 10.1211/0022357011775181 1:CAS:528:DC%2BD3MXht1Shsro%3D (Pubitemid 32123699)
12. BN Singh KH Kim 2000 Floating drug delivery systems: an approach to oral controlled drug delivery via gastric retention J Control Release 63 235 259 10601721 10.1016/S0168-3659(99)00204-7 1:CAS:528:DyaK1MXnvFSmu7w%3D
13. L Shan-Yang Y Hui-Ling 2000 Microscopic Fourier transform infrared/differential scanning calorimetry system used to study the different thermal behaviors of polymethacrylate copolymers of Eudragits RS, RL, E 30D, or E J Appl Polym Sci 78 8298 35
14. L Shan-Yang Y Hui-Ling L Mei-Jane 1999 Formation of six-membered cyclic anhydrides by thermally induced intramolecular ester condensation in Eudragit E Film Polymer 40 3589 3593 10.1016/S0032-3861(98)00488-1 (Pubitemid 30122579)
15. K Picker 1999 The use of carrageenan in mixture with microcrystalline cellulose and its functionality for making tablets Eur J Pharm Biopharm 48 27 36 10477325 10.1016/S0939-6411(99)00009-0 1:CAS:528:DyaK1MXlslagsrs%3D (Pubitemid 29308922)
16. HJ Prado MC Matulewicz P Bonelli AL Cukierman 2008 Basic butylated methacrylate copolymer/kappa-carrageenan interpolyelectrolyte complex: preparation, characterization and drug release behaviour Eur J Pharm Biopharm 70 171 178 18583115 10.1016/j.ejpb.2008.04.017 1:CAS:528:DC%2BD1cXhtVOitrjP
17. M Jaimini AC Rana YS Tanwar 2007 Formulation and evaluation of famotidine floating tablets Curr Drug Deliv 4 51 55 17269917 10.2174/156720107779314730 1:CAS:528:DC%2BD2sXitlamtbo%3D (Pubitemid 46066414)
18. LG Bakre KT Jaiyeoba 2009 Effects of drying methods on the physicochemical and compressional characteristics of okra powder and the release properties of its metronidazole tablet formulation Arch Pharm Res 32 259 67 19280157 10.1007/s12272-009-1231-0 1:CAS:528:DC%2BD1MXislanu78%3D
19. Sankalia MG, Mashru RC, Sankalia JM, Sutariya VB. Stability improvement of alpha-amylase entrapped in kappa-carrageenan beads: physicochemical characterization and optimization using composite index. Int J Pharm. 2006;312:1-14.
20. R Moustafine I Zaharov V Kemenova 2006 Physicochemical Characterization and Drug Release Properties of Eudragit E PO/Eudragit L 100-55 Inter Polyelectrolyte Complexes Eur J Pharm Biopharm 63 26 36 16380241 10.1016/j.ejpb.2005.10.005 1:CAS:528:DC%2BD28XjtFGhur0%3D
21. M Bonferoni S Rossi F Ferrari G Bettinetti C Caramella 2000 Characterization of a diltiazem-λ-carrageenan complex Int J Pharm 200 207 216 10867250 10.1016/S0378-5173(00)00389-6 1:CAS:528:DC%2BD3cXktFemsrs%3D (Pubitemid 30364907)
22. R Korsmeyer R Gurny E Doelker P Buri N Peppas 1983 Mechanism of solute release from porous hydrophilic polymers Int J Pharm 15 25 35 10.1016/0378-5173(83)90064-9 1:CAS:528:DyaL3sXksVens7Y%3D (Pubitemid 13092121)
23. N Peppas 1985 Analysis of Fickian and non-Fickian drug release from polymers Pharm Acta Helv 60 110 111 4011621 1:CAS:528:DyaL2MXktFWgtb8%3D