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Volumn 6, Issue 4, 2011, Pages 593-599

Developing Pyrrole-Derived Antimycobacterial Agents: A Rational Lead Optimization Approach

(8) Biava, Mariangela a Porretta, Giulio Cesare b Poce, Giovanna a Battilocchio, Claudio a Alfonso, Salvatore a deLogu, Alessandro b Manetti, Fabrizio c Botta, Maurizio c

a SAPIENZA UNIVERSITY OF ROME (Italy)

b UNIVERSITY OF CAGLIARI (Italy)

c UNIVERSITY OF SIENA (Italy)

Author keywords

Antimycobacterial agents; Cytotoxicity; Pharmacophores; Pyrrole derivatives; Tuberculosis

Indexed keywords

ANTIMYCOBACTERIAL AGENT; ISONIAZID; PYRROLE DERIVATIVE; RIFAMPICIN; TUBERCULOSTATIC AGENT;

ANTIBACTERIAL ACTIVITY; CONTROLLED STUDY; CYTOTOXICITY; DRUG SYNTHESIS; MINIMUM INHIBITORY CONCENTRATION; MYCOBACTERIUM TUBERCULOSIS; NONHUMAN; PRIORITY JOURNAL; REACTION OPTIMIZATION; REVIEW; STRUCTURE ACTIVITY RELATION;

ANIMALS; ANTITUBERCULAR AGENTS; DRUG DESIGN; HUMANS; MYCOBACTERIUM TUBERCULOSIS; PYRROLES; STRUCTURE-ACTIVITY RELATIONSHIP; TUBERCULOSIS;

EID: 79953052237 PISSN: 18607179 EISSN: 18607187 Source Type: Journal
DOI: 10.1002/cmdc.201000526 Document Type: Review

Times cited : (44)

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