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Journal of the American Chemical Society

Volumn 132, Issue 39, 2010, Pages 13663-13665

Benzothiazinones: Prodrugs that covalently modify the decaprenylphosphoryl- β-D-ribose 2′-epimerase DprE1 of mycobacterium tuberculosis

(7) Trefzer, Claudia a Rengifo Gonzalez, Monica a Hinner, Marlon J a Schneider, Patricia a Makarov, Vadim a,b Cole, Stewart T a Johnsson, Kai a

a EPFL (Switzerland)

b BACH INSTITUTE OF BIOCHEMISTRY (Russian Federation)

Author keywords

[No Author keywords available]

Indexed keywords

ACTIVE SITE; ANTI-MYCOBACTERIAL; CYSTEINE RESIDUES; D-RIBOSE; MECHANISM OF ACTION; MYCOBACTERIUM TUBERCULOSIS; NITRO GROUP; NITROSO; PRODRUGS;

ANTIMYCOBACTERIAL AGENT; BENZOTHIAZINE DERIVATIVE; CYSTEINE; DECAPRENYLPHOSPHORYL BETA DEXTRO RIBOSE 2' EPIMERASE; EPIMERASE; NITRO DERIVATIVE; NITROSO DERIVATIVE; PRODRUG; UNCLASSIFIED DRUG;

ANTIBACTERIAL ACTIVITY; ARTICLE; CHEMICAL MODIFICATION; COVALENT BOND; DRUG MECHANISM; DRUG POTENCY; DRUG TARGETING; ENZYME ACTIVE SITE; MYCOBACTERIUM BOVIS; MYCOBACTERIUM SMEGMATIS; MYCOBACTERIUM TUBERCULOSIS; NONHUMAN;

ANTI-BACTERIAL AGENTS; CATALYTIC DOMAIN; MOLECULAR CONFORMATION; MYCOBACTERIUM TUBERCULOSIS; PRODRUGS; RACEMASES AND EPIMERASES; STEREOISOMERISM; STRUCTURE-ACTIVITY RELATIONSHIP; THIAZINES;

EID: 77957310736 PISSN: 00027863 EISSN: 15205126 Source Type: Journal
DOI: 10.1021/ja106357w Document Type: Article

Times cited : (193)

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