The penultimate arginine of the carboxyl terminus determines slow desensitization in a P2X receptor from the cattle tick Boophilus microplus

Molecular Pharmacology

Volumn 79, Issue 4, 2011, Pages 776-785

  Bavan, Selvan ^a   Farmer, Louise ^a   Singh, Shire K ^a   Straub, Volko A ^a   Guerrero, Felix D ^b   Ennion, Steven J ^a  

^a UNIVERSITY OF LEICESTER   (United Kingdom)

^b U S DEPARTMENT OF AGRICULTURE   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ADENOSINE TRIPHOSPHATE; AMITRAZ; ARGININE; IVERMECTIN; PURINERGIC P2X RECEPTOR; SURAMIN;

ARTICLE; BOOPHILUS MICROPLUS; CARBOXY TERMINAL SEQUENCE; CONTROLLED STUDY; DRUG MECHANISM; DRUG SENSITIVITY; IC 50; KINETICS; MUTATION; NONHUMAN; NUCLEOTIDE SEQUENCE; PHENOTYPE; PRIORITY JOURNAL; RECEPTOR DOWN REGULATION; WILD TYPE;

AMINO ACID SEQUENCE; ANIMALS; ARGININE; CATTLE; FEMALE; MOLECULAR SEQUENCE DATA; MUTATION; PEPTIDE FRAGMENTS; PROTEIN STRUCTURE, TERTIARY; RECEPTORS, PURINERGIC P2X; TICKS; TIME FACTORS; XENOPUS LAEVIS;

EID: 79952999410     PISSN: 0026895X     EISSN: 15210111     Source Type: Journal    
DOI: 10.1124/mol.110.070037     Document Type: Article

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