메뉴 건너뛰기




Volumn 412, Issue 1, 2011, Pages 85-91

Development and characterization of immobilized cannabinoid receptor (CB1/CB2) open tubular column for on-line screening

Author keywords

Basophils; Biochromatography; Cannabinoids; KU 812; Zanthoxylum

Indexed keywords

ACTIVATION ANALYSIS; BINDING ENERGY; CELL CULTURE;

EID: 79952439940     PISSN: 00032697     EISSN: 10960309     Source Type: Journal    
DOI: 10.1016/j.ab.2010.12.034     Document Type: Article
Times cited : (39)

References (31)
  • 1
    • 0029965292 scopus 로고    scopus 로고
    • Structural features of the central cannabinoid CB1 receptor involved in the binding of the specific CB1 antagonist SR 141716A
    • DOI 10.1074/jbc.271.12.6941
    • D. Shire, B. Calandra, M. Delpech, X. Dumont, M. Kaghad, G. Le Fur, D. Caput, and P. Ferrara Structural features of the central cannabinoid CB1 receptor involved in the binding of the specific CB1 antagonist SR 141716A J. Biol. Chem. 271 1996 6941 6946 (Pubitemid 26104790)
    • (1996) Journal of Biological Chemistry , vol.271 , Issue.12 , pp. 6941-6946
    • Shire, D.1    Calandra, B.2    Delpech, M.3    Dumont, X.4    Kaghad, M.5    Le Fur, G.6    Caput, D.7    Ferrara, P.8
  • 4
    • 0029094470 scopus 로고
    • Expression of central and cannabinoid receptors in human immune tissues and leukocyte subpopulations
    • S. Galiegue, S. Mary, J. Marchand, D. Dussossoy, D. Carriere, and P. Carayon Expression of central and cannabinoid receptors in human immune tissues and leukocyte subpopulations Eur. J. Biochem. 232 1995 54 61
    • (1995) Eur. J. Biochem. , vol.232 , pp. 54-61
    • Galiegue, S.1    Mary, S.2    Marchand, J.3    Dussossoy, D.4    Carriere, D.5    Carayon, P.6
  • 6
    • 0034717138 scopus 로고    scopus 로고
    • Genomic and functional changes induced by the activation of the peripheral cannabinoid receptor CB2 in the promyelocytic cells HL-60. Possible involvement of the CB2 receptor in cell differentiation
    • DOI 10.1074/jbc.275.21.15621
    • J.M. Derocq, O. Jbilo, M. Bouaboula, M. Segui, C. Clere, and P. Casellas Genomic and functional changes induced by the activation of the peripheral cannabinoid receptor CB2 in the promyelocytic cells HL-60: possible involvement of the CB2 receptor in cell differentiation J. Biol. Chem. 275 2000 15621 15628 (Pubitemid 30366856)
    • (2000) Journal of Biological Chemistry , vol.275 , Issue.21 , pp. 15621-15628
    • Derocq, J.-M.1    Jbilo, O.2    Bouaboula, M.3    Segui, M.4    Clere, C.5    Casellas, P.6
  • 7
    • 0030611978 scopus 로고    scopus 로고
    • 2 receptors
    • DOI 10.1016/S0163-7258(97)82001-3, PII S0163725896002045
    • R.G. Pertwee The pharmacology of cannabinoid CB1 and CB2 receptors Pharmacol. Ther. 74 1997 129 180 (Pubitemid 27337346)
    • (1997) Pharmacology and Therapeutics , vol.74 , Issue.2 , pp. 129-180
    • Pertwee, R.G.1
  • 8
    • 0033427968 scopus 로고    scopus 로고
    • A light and electron microscopic study of the CB1 cannabinoid receptor in the primate spinal cord
    • DOI 10.1023/A:1007011700677
    • W.Y. Ong, and K. Mackie A light and electron microscopic study of the CB1 cannabinoid receptor in the primate spinal cord J. Neurocytol. 28 1999 39 45 (Pubitemid 30040768)
    • (1999) Journal of Neurocytology , vol.28 , Issue.1 , pp. 39-45
    • Ong, W.Y.1    Mackie, K.2
  • 9
    • 33144480327 scopus 로고    scopus 로고
    • Cannabinoid receptors as therapeutic targets
    • K. Mackie Cannabinoid receptors as therapeutic targets Annu. Rev. Pharmacol. Toxicol. 46 2006 101 122
    • (2006) Annu. Rev. Pharmacol. Toxicol. , vol.46 , pp. 101-122
    • MacKie, K.1
  • 11
    • 33645293110 scopus 로고    scopus 로고
    • Screening assays for cannabinoid-ligand-type modulators of GPR55
    • US patent 2006/0194260 A1
    • T. Drmota, P. Greasley, T. Groblewski, Screening assays for cannabinoid-ligand-type modulators of GPR55, US patent 2006/0194260 A1 (2006).
    • (2006)
    • Drmota, T.1    Greasley, P.2    Groblewski, T.3
  • 13
    • 0042934012 scopus 로고    scopus 로고
    • Evidence for cannabinoid receptor-dependent and -independent mechanisms of action in leukocytes
    • DOI 10.1124/jpet.103.051961
    • B.L. Faubert Kaplan, C.E. Rockwell, and N.E. Kaminski Evidence for cannabinoid receptor-dependent and-independent mechanisms of action in leukocytes J. Pharmacol. Exp. Ther. 306 2003 1077 1085 (Pubitemid 37025316)
    • (2003) Journal of Pharmacology and Experimental Therapeutics , vol.306 , Issue.3 , pp. 1077-1085
    • Kaplan, B.L.F.1    Rockwell, C.E.2    Kaminski, N.E.3
  • 14
    • 59849097146 scopus 로고    scopus 로고
    • The preparation and development of cellular membrane affinity chromatography columns
    • R. Moaddel, and I.W. Wainer The preparation and development of cellular membrane affinity chromatography columns Nat. Protoc. 4 2009 197 205
    • (2009) Nat. Protoc. , vol.4 , pp. 197-205
    • Moaddel, R.1    Wainer, I.W.2
  • 16
    • 33748702969 scopus 로고    scopus 로고
    • Comparison of an open tubular column containing immobilized P-glycoprotein with Caco-2 cell monolayers for the purpose of investigating interactions between drug candidates and Pgp
    • R. Moaddel, R. Hamid, S. Patel, I.W. Wainer, and P. Bullock Comparison of an open tubular column containing immobilized P-glycoprotein with Caco-2 cell monolayers for the purpose of investigating interactions between drug candidates and Pgp Anal. Chim. Acta 578 2006 25 30
    • (2006) Anal. Chim. Acta , vol.578 , pp. 25-30
    • Moaddel, R.1    Hamid, R.2    Patel, S.3    Wainer, I.W.4    Bullock, P.5
  • 17
    • 67849084545 scopus 로고    scopus 로고
    • Synthesis, cannabinoid receptor affinity, molecular modeling studies, and in vivo pharmacological evaluation of new substituted 1-aryl-5-(1H-pyrrol-1-yl) -1H-pyrazole-3-carboxamides: 2. Effect of the 3-carboxamide substituent on the affinity and selectivity profile
    • R. Silvestri, A. Ligresti, G. La Regina, F. Piscitelli, V. Gatti, A. Brizzi, S. Pasquini, A. Lavecchia, M. Allar, N. Fantini, M.A. Carai, E. Novellino, G. Colombo, V. Di Marzo, and F. Corelli Synthesis, cannabinoid receptor affinity, molecular modeling studies, and in vivo pharmacological evaluation of new substituted 1-aryl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3- carboxamides: 2. Effect of the 3-carboxamide substituent on the affinity and selectivity profile Bioorg. Med. Chem. 17 2009 5549 5564
    • (2009) Bioorg. Med. Chem. , vol.17 , pp. 5549-5564
    • Silvestri, R.1    Ligresti, A.2    La Regina, G.3    Piscitelli, F.4    Gatti, V.5    Brizzi, A.6    Pasquini, S.7    Lavecchia, A.8    Allar, M.9    Fantini, N.10    Carai, M.A.11    Novellino, E.12    Colombo, G.13    Di Marzo, V.14    Corelli, F.15
  • 20
    • 50249099198 scopus 로고    scopus 로고
    • Investigations on the 4-quinolone-3-carboxylic acid motif: 2. Synthesis and structure-activity relationship of potent and selective cannabinoid-2 receptor agonists endowed with analgesic activity in vivo
    • S. Pasquini, L. Botta, T. Semeraro, C. Mugnaini, A. Ligresti, E. Palazzo, S. Maione, V. Di Marzo, and F. Corelli Investigations on the 4-quinolone-3-carboxylic acid motif: 2. Synthesis and structure-activity relationship of potent and selective cannabinoid-2 receptor agonists endowed with analgesic activity in vivo J. Med. Chem. 51 2008 5075 5084
    • (2008) J. Med. Chem. , vol.51 , pp. 5075-5084
    • Pasquini, S.1    Botta, L.2    Semeraro, T.3    Mugnaini, C.4    Ligresti, A.5    Palazzo, E.6    Maione, S.7    Di Marzo, V.8    Corelli, F.9
  • 21
    • 33746138649 scopus 로고    scopus 로고
    • Cannabinoids induce apoptosis of pancreatic tumor cells via endoplasmic reticulum stress-related genes
    • DOI 10.1158/0008-5472.CAN-06-0169
    • A. Carracedo, M. Gironella, M. Lorente, S. Garcia, M. Guzma, G. Velasco, and J.L. Iovanna Cannabinoids induce apoptosis of pancreatic tumor cells via endoplasmic reticulum stress-related genes Cancer Res. 66 2006 6748 6755 (Pubitemid 44085633)
    • (2006) Cancer Research , vol.66 , Issue.13 , pp. 6748-6755
    • Carracedo, A.1    Gironella, M.2    Lorente, M.3    Garcia, S.4    Guzman, M.5    Velasco, G.6    Iovanna, J.L.7
  • 24
    • 56449110129 scopus 로고    scopus 로고
    • Characterization of a multiple ligand-gated ion channel cellular membrane affinity chromatography (CMAC) column and identification of endogenously expressed receptors in astrocytoma cell lines
    • T. Kitabatake, R. Moaddel, R. Cole, M. Gandhari, C. Frazier, J. Hartenstein, A. Rosenberg, M. Bernier, and I.W. Wainer Characterization of a multiple ligand-gated ion channel cellular membrane affinity chromatography (CMAC) column and identification of endogenously expressed receptors in astrocytoma cell lines Anal. Chem. 80 2008 8673 8680
    • (2008) Anal. Chem. , vol.80 , pp. 8673-8680
    • Kitabatake, T.1    Moaddel, R.2    Cole, R.3    Gandhari, M.4    Frazier, C.5    Hartenstein, J.6    Rosenberg, A.7    Bernier, M.8    Wainer, I.W.9
  • 25
    • 8844232736 scopus 로고    scopus 로고
    • On-line screening of conformationally constrained nicotines and anabasines for agonist activity at the α3β4- and α4β2- nicotinic acetylcholine receptors using immobilized receptor-based liquid chromatographic stationary phases
    • DOI 10.1016/j.jchromb.2004.09.042, PII S1570023204007780
    • R. Moaddel, K. Jozwiak, R. Yamaguchi, C. Cobello, K. Whittington, T. Sarkar, S. Basak, and I.W. Wainer On-line screening of conformationally constrained nicotines and anabasines for agonist activity at the α3β4 and α4β2-nicotinic acetylcholine receptors using immobilized receptor based liquid chromatographic stationary phases J. Chromatogr. B 813 2004 235 240 (Pubitemid 39535451)
    • (2004) Journal of Chromatography B: Analytical Technologies in the Biomedical and Life Sciences , vol.813 , Issue.1-2 , pp. 235-240
    • Moaddel, R.1    Jozwiak, K.2    Yamaguchi, R.3    Cobello, C.4    Whittington, K.5    Sarkar, T.K.6    Basak, S.7    Wainer, I.W.8
  • 27
    • 67349244423 scopus 로고    scopus 로고
    • Comparison of alkylamide yield in ethanolic extracts prepared from fresh versus dry Echinacea purpurea utilizing HPLC-ESI-MS
    • K. Spelman, M.H. Wetschler, and N.B. Cech Comparison of alkylamide yield in ethanolic extracts prepared from fresh versus dry Echinacea purpurea utilizing HPLC-ESI-MS J. Pharm. Biomed. Anal. 49 2009 1141 1149
    • (2009) J. Pharm. Biomed. Anal. , vol.49 , pp. 1141-1149
    • Spelman, K.1    Wetschler, M.H.2    Cech, N.B.3
  • 28
    • 8844271735 scopus 로고    scopus 로고
    • Echinacea alkylamides modulate TNF-α gene expression via cannabinoid receptor CB2 and multiple signal transduction pathways
    • DOI 10.1016/j.febslet.2004.10.064, PII S0014579304013183
    • J. Gertsch, R. Schoop, U. Kuenzle, and A. Suter Echinacea alkylamides modulate TNF-α gene expression via cannabinoid receptor CB2 and multiple signal transduction pathways FEBS Lett. 577 2004 563 569 (Pubitemid 39535349)
    • (2004) FEBS Letters , vol.577 , Issue.3 , pp. 563-569
    • Gertsch, J.1    Schoop, R.2    Kuenzle, U.3    Suter, A.4
  • 29
    • 33744916587 scopus 로고    scopus 로고
    • Alkylamides from Echinacea are a new class of cannabinomimetics: Cannabinoid type 2 receptor-dependent and -independent immunomodulatory effects
    • DOI 10.1074/jbc.M601074200
    • S. Raduner, A. Majewska, J.-Z. Chen, X.-Q. Xie, J. Hamon, B. Faller, K.-H. Altmann, and J. Gertsch Alkylamides from Echinacea are a new class of cannabinomimetics: cannabinoid type 2 receptor-dependent and -independent immunomodulatory effects J. Biol. Chem. 281 2006 14192 14206 (Pubitemid 43848347)
    • (2006) Journal of Biological Chemistry , vol.281 , Issue.20 , pp. 14192-14206
    • Raduner, S.1    Majewska, A.2    Chen, J.-Z.3    Xie, X.-Q.4    Hamon, J.5    Faller, B.6    Altmann, K.-H.7    Gertsch, J.8


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.