메뉴 건너뛰기




Volumn 33, Issue 12, 2010, Pages 1891-1900

Synthesis and antimicrobial activity of novel 5-amino-4-cyano-1H-pyrazole and quinazolin-4(3H)-one derivatives

Author keywords

5 Amino 4 cyanopyrazole; Antimicrobial activity; Aroylhydrazones; Quinazoline 4 one

Indexed keywords

5 AMINO 4 CYANO 1H PYRAZOLE DERIVATIVE; HYDRAZONE DERIVATIVE; PYRAZOLE DERIVATIVE; PYRIMIDINE DERIVATIVE; QUINAZOLIN 4 (3H) ONE DERIVATIVE; UNCLASSIFIED DRUG;

EID: 78751520443     PISSN: 02536269     EISSN: 19763786     Source Type: Journal    
DOI: 10.1007/s12272-010-1202-5     Document Type: Article
Times cited : (14)

References (42)
  • 1
    • 0344013139 scopus 로고    scopus 로고
    • Synthesis of some functionalized arylaminomethyl-1,2,4-triazoles, 1,3,4-oxa- and thiadiazoles
    • 1:CAS:528:DC%2BD3sXpt1Clsbs%3D 14664332
    • M. T. Abdel-Aal W. A. El-Sayed A. H. Abdel Aleem E. S. H. El-Ashry 2003 Synthesis of some functionalized arylaminomethyl-1,2,4-triazoles, 1,3,4-oxa- and thiadiazoles Pharmazie 58 788 792 1:CAS:528:DC%2BD3sXpt1Clsbs%3D 14664332
    • (2003) Pharmazie , vol.58 , pp. 788-792
    • Abdel-Aal, M.T.1    El-Sayed, W.A.2    Abdel Aleem, A.H.3    El-Ashry, E.S.H.4
  • 2
    • 33846192348 scopus 로고    scopus 로고
    • Synthesis and antiviral evaluation of some sugar arylglycinoylhydrazones and their oxadiazoline derivatives
    • 1:CAS:528:DC%2BD2sXmsFaltg%3D%3D 10.1002/ardp.200600100
    • M. T. Abdel-Aal W. A. El-Sayed E. S. H. El-Ashry 2006 Synthesis and antiviral evaluation of some sugar arylglycinoylhydrazones and their oxadiazoline derivatives Arch. Pharm. (Weinheim) 339 656 663 1:CAS:528:DC%2BD2sXmsFaltg%3D%3D 10.1002/ardp.200600100
    • (2006) Arch. Pharm. (Weinheim) , vol.339 , pp. 656-663
    • Abdel-Aal, M.T.1    El-Sayed, W.A.2    El-Ashry, E.S.H.3
  • 3
    • 46449097021 scopus 로고    scopus 로고
    • Synthesis and antiviral evaluation of novel 5-(N-Aryl-aminomethyl-1,3,4- oxadiazol-2-yl)hydrazines and their sugars, 1,2,4-triazoles, tetrazoles and pyrazolyl derivatives
    • 1:CAS:528:DC%2BD1cXmslWls7Y%3D 10.1002/ardp.200700154
    • M. T. Abdel-Aal W. A. El-Sayed S. M. El-Kosy E. S. H. El-Ashry 2008 Synthesis and antiviral evaluation of novel 5-(N-Aryl-aminomethyl-1,3,4- oxadiazol-2-yl)hydrazines and their sugars, 1,2,4-triazoles, tetrazoles and pyrazolyl derivatives Arch. Pharm. (Weinheim) 341 307 313 1:CAS:528: DC%2BD1cXmslWls7Y%3D 10.1002/ardp.200700154
    • (2008) Arch. Pharm. (Weinheim) , vol.341 , pp. 307-313
    • Abdel-Aal, M.T.1    El-Sayed, W.A.2    El-Kosy, S.M.3    El-Ashry, E.S.H.4
  • 4
    • 0000831354 scopus 로고
    • The N-acylhydrazine grouping as a ligand. I. Coordination compounds of Keto- and Enol-N-acylhydrazines with cobalt(II), nickel (II), and copper (II)
    • 1:CAS:528:DyaE38XmslGlsQ%3D%3D 10.1071/CH9720289
    • J. F. Alcock R. J. Baker A. A. Diamantis 1972 The N-acylhydrazine grouping as a ligand. I. Coordination compounds of Keto- and Enol-N-acylhydrazines with cobalt(II), nickel (II), and copper (II) Aust. J. Chem. 25 289 302 1:CAS:528:DyaE38XmslGlsQ%3D%3D 10.1071/CH9720289
    • (1972) Aust. J. Chem. , vol.25 , pp. 289-302
    • Alcock, J.F.1    Baker, R.J.2    Diamantis, A.A.3
  • 5
    • 30344476416 scopus 로고    scopus 로고
    • Synthesis of C-6 substituted pyrazolo[1,5-a]pyridines with potent activity against herpesviruses
    • 1:CAS:528:DC%2BD28XhvFOitw%3D%3D 10.1016/j.bmc.2005.09.015 16213142
    • S. H. Allen B. A. Johns K. S. Gudmundsson G. A. Freeman 2006 Synthesis of C-6 substituted pyrazolo[1,5-a]pyridines with potent activity against herpesviruses Bioorg. Med. Chem. 14 944 954 1:CAS:528:DC%2BD28XhvFOitw%3D%3D 10.1016/j.bmc.2005.09.015 16213142
    • (2006) Bioorg. Med. Chem. , vol.14 , pp. 944-954
    • Allen, S.H.1    Johns, B.A.2    Gudmundsson, K.S.3    Freeman, G.A.4
  • 6
    • 4544336251 scopus 로고    scopus 로고
    • In vivo radioprotection of mice by 3-methyl-1-phenyl-2-pyrazolin-5-one (edaravone; Radicut), a clinical drug
    • 1:CAS:528:DC%2BD2cXot1OqtL0%3D 10.1269/jrr.45.319 15304976
    • K. Anzai M. Furuse A. Yoshida A. Matsuyama T. Moritake K. Tsuboi 2004 In vivo radioprotection of mice by 3-methyl-1-phenyl-2-pyrazolin-5-one (edaravone; radicut), a clinical drug J. Radiat. Res. 45 319 323 1:CAS:528: DC%2BD2cXot1OqtL0%3D 10.1269/jrr.45.319 15304976
    • (2004) J. Radiat. Res. , vol.45 , pp. 319-323
    • Anzai, K.1    Furuse, M.2    Yoshida, A.3    Matsuyama, A.4    Moritake, T.5    Tsuboi, K.6
  • 7
    • 33244494206 scopus 로고    scopus 로고
    • Synthesis and leishmanicidal activities of 1-(4-X-phenyl)-N′-[(4-Y- phenyl)methylene]-1H-pyrazole-4-carbohydrazides
    • 1:CAS:528:DC%2BD28XhvVyrsrk%3D 10.1016/j.ejmech.2005.10.007 16300859
    • A. M. R. Bernardino A. O. Gomes K. S. Charret A. C. C. Freitas 2006 Synthesis and leishmanicidal activities of 1-(4-X-phenyl)-N′-[(4-Y-phenyl) methylene]-1H-pyrazole-4-carbohydrazides Eur. J. Med. Chem. 41 80 87 1:CAS:528:DC%2BD28XhvVyrsrk%3D 10.1016/j.ejmech.2005.10.007 16300859
    • (2006) Eur. J. Med. Chem. , vol.41 , pp. 80-87
    • Bernardino, A.M.R.1    Gomes, A.O.2    Charret, K.S.3    Freitas, A.C.C.4
  • 8
    • 0022532716 scopus 로고
    • Chemistry and antiviral activities of acyclonucleosides
    • 1:CAS:528:DyaL28XltlChtrg%3D 10.1002/jhet.5570230201
    • C. K. Chu S. J. Cutler 1986 Chemistry and antiviral activities of acyclonucleosides J. Heterocycl. Chem. 23 289 319 1:CAS:528:DyaL28XltlChtrg%3D 10.1002/jhet.5570230201
    • (1986) J. Heterocycl. Chem. , vol.23 , pp. 289-319
    • Chu, C.K.1    Cutler, S.J.2
  • 9
    • 25144475990 scopus 로고    scopus 로고
    • Synthesis of quinazolinones and quinazolines
    • 1:CAS:528:DC%2BD2MXhtVantbjK 10.1016/j.tet.2005.07.010
    • D. J. Connolly D. Cusack T. P. O'sullivan P. J. Guiry 2005 Synthesis of quinazolinones and quinazolines Tetrahedron 61 10153 10202 1:CAS:528: DC%2BD2MXhtVantbjK 10.1016/j.tet.2005.07.010
    • (2005) Tetrahedron , vol.61 , pp. 10153-10202
    • Connolly, D.J.1    Cusack, D.2    O'Sullivan, T.P.3    Guiry, P.J.4
  • 10
    • 33745568982 scopus 로고    scopus 로고
    • Antileishmanial and antibacterial activity of a new pyrazole derivative designated 4-[2-(1-(ethylamino)-2-methyl-propyl) phenyl]-3-(4-methyphenyl)-1- phenylpyrazole
    • 1:CAS:528:DC%2BD28XmtFSksrk%3D 10.1002/ardp.200500266
    • Z. Dardari M. Lemrani A. Sebban A. Bahloul 2006 Antileishmanial and antibacterial activity of a new pyrazole derivative designated 4-[2-(1-(ethylamino)-2-methyl-propyl) phenyl]-3-(4-methyphenyl)-1-phenylpyrazole Arch. Pharm. (Weinheim) 339 291 298 1:CAS:528:DC%2BD28XmtFSksrk%3D 10.1002/ardp.200500266
    • (2006) Arch. Pharm. (Weinheim) , vol.339 , pp. 291-298
    • Dardari, Z.1    Lemrani, M.2    Sebban, A.3    Bahloul, A.4
  • 11
    • 0026019218 scopus 로고
    • Synthesis of certain 2-aminoadamantane derivatives as potential antimicrobial agents
    • 1:CAS:528:DyaK3MXkt12htL4%3D 1909034
    • H. Eisa A. Tantawy M. El-Kerdawy 1991 Synthesis of certain 2-aminoadamantane derivatives as potential antimicrobial agents Pharmazie 46 182 184 1:CAS:528:DyaK3MXkt12htL4%3D 1909034
    • (1991) Pharmazie , vol.46 , pp. 182-184
    • Eisa, H.1    Tantawy, A.2    El-Kerdawy, M.3
  • 12
    • 33751044696 scopus 로고    scopus 로고
    • Acyclonucleosides: Part 1. seco-Nucleosides
    • 10.1016/S0065-2725(08)60074-4
    • E. S. H. El Ashry Y. El Kilany 1996 Acyclonucleosides: part 1. seco-Nucleosides Adv. Heterocycl. Chem. 67 391 438 10.1016/S0065-2725(08)60074-4
    • (1996) Adv. Heterocycl. Chem. , vol.67 , pp. 391-438
    • El Ashry, E.S.H.1    El Kilany, Y.2
  • 13
    • 6744261417 scopus 로고    scopus 로고
    • Acyclonucleosides: Part 2. diseco-Nucleosides
    • 10.1016/S0065-2725(08)60360-8
    • E. S. H. El Ashry Y. El Kilany 1997 Acyclonucleosides: part 2. diseco-Nucleosides Adv. Heterocycl. Chem. 68 1 88 10.1016/S0065-2725(08)60360-8
    • (1997) Adv. Heterocycl. Chem. , vol.68 , pp. 1-88
    • El Ashry, E.S.H.1    El Kilany, Y.2
  • 14
    • 33750826586 scopus 로고    scopus 로고
    • Acyclonucleosides: Part 3. tri-, tetra-, and pentaseco-Nucleosides
    • 10.1016/S0065-2725(08)60082-3
    • E. S. H. El Ashry Y. El Kilany 1997 Acyclonucleosides: part 3. tri-, tetra-, and pentaseco-Nucleosides Adv. Heterocycl. Chem. 69 129 215 10.1016/S0065-2725(08)60082-3
    • (1997) Adv. Heterocycl. Chem. , vol.69 , pp. 129-215
    • El Ashry, E.S.H.1    El Kilany, Y.2
  • 15
    • 77951639714 scopus 로고    scopus 로고
    • Synthesis and antimicrobial activity of new substituted 1,2,4-triazoles and their acyclic C-nucleoside analogues
    • 1:CAS:528:DC%2BC3cXjtFaiurY%3D 20355315
    • W. A. El-Sayed O. M. Ali S. R. El-Dakkony A. A. Abdel-Rahman 2010 Synthesis and antimicrobial activity of new substituted 1,2,4-triazoles and their acyclic C-nucleoside analogues Z. Naturforsch. C 65 15 21 1:CAS:528:DC%2BC3cXjtFaiurY%3D 20355315
    • (2010) Z. Naturforsch. C , vol.65 , pp. 15-21
    • El-Sayed, W.A.1    Ali, O.M.2    El-Dakkony, S.R.3    Abdel-Rahman, A.A.4
  • 16
    • 21744458419 scopus 로고    scopus 로고
    • Synthesis and antibacterial activity of 1H-pyrazolo[3,4-b]pyrazine and -pyridine derivatives
    • 1:CAS:528:DC%2BD2MXlvFKqt7o%3D 10.1016/j.farmac.2005.05.002 15950227
    • H. Foks D. Pancechowska-Ksepko A. Kedzia Z. Zwolska 2005 Synthesis and antibacterial activity of 1H-pyrazolo[3,4-b]pyrazine and -pyridine derivatives Farmaco 60 513 517 1:CAS:528:DC%2BD2MXlvFKqt7o%3D 10.1016/j.farmac.2005.05.002 15950227
    • (2005) Farmaco , vol.60 , pp. 513-517
    • Foks, H.1    Pancechowska-Ksepko, D.2    Kedzia, A.3    Zwolska, Z.4
  • 18
    • 33749265829 scopus 로고    scopus 로고
    • Pyrazolidine-3,5-diones and 5-hydroxy-1H-pyrazol-3(2H)-ones, inhibitors of UDP-N-acetylenolpyruvyl glucosamine reductase
    • 1:CAS:528:DC%2BD28XptlOks70%3D 10.1021/jm060499t 17004716
    • A. M. Gilbert A. Failli J. Shumsky Y. Yang 2006 Pyrazolidine-3,5-diones and 5-hydroxy-1H-pyrazol-3(2H)-ones, inhibitors of UDP-N-acetylenolpyruvyl glucosamine reductase J. Med. Chem 49 6027 6036 1:CAS:528:DC%2BD28XptlOks70%3D 10.1021/jm060499t 17004716
    • (2006) J. Med. Chem , vol.49 , pp. 6027-6036
    • Gilbert, A.M.1    Failli, A.2    Shumsky, J.3    Yang, Y.4
  • 19
    • 0039573050 scopus 로고    scopus 로고
    • Synthesis of some new hydrazide-hydrazones
    • 1:CAS:528:DyaK2sXmsVChsb4%3D 10.1016/S0223-5234(97)88918-0
    • A. Gursoy N. Terzioglu G. Otuk 1997 Synthesis of some new hydrazide-hydrazones Eur. J. Med. Chem. 32 753 757 1:CAS:528:DyaK2sXmsVChsb4%3D 10.1016/S0223-5234(97)88918-0
    • (1997) Eur. J. Med. Chem. , vol.32 , pp. 753-757
    • Gursoy, A.1    Terzioglu, N.2    Otuk, G.3
  • 20
    • 3242773632 scopus 로고    scopus 로고
    • Application of the palladium-catalyzed N-arylation of hydrazones to deactivated heteroaryl halides in the synthesis of pyrazoles
    • 1:CAS:528:DC%2BD2cXlsVyqs7o%3D 10.1016/j.tetlet.2004.05.038
    • N. Haddad A. Salvagno C. Busacca 2004 Application of the palladium-catalyzed N-arylation of hydrazones to deactivated heteroaryl halides in the synthesis of pyrazoles Tetrahedron Lett. 45 5935 5937 1:CAS:528:DC%2BD2cXlsVyqs7o%3D 10.1016/j.tetlet.2004.05.038
    • (2004) Tetrahedron Lett. , vol.45 , pp. 5935-5937
    • Haddad, N.1    Salvagno, A.2    Busacca, C.3
  • 21
    • 0346618165 scopus 로고    scopus 로고
    • Synthesis of D-apio-β-D-furanosyl maleimide, an analogue of showdomycin with transposed hydroxymethyl group
    • 1:CAS:528:DyaK2sXjs1Kitbk%3D 10.1007/BF00807307
    • F. Hammerschmidt B. Peric E. Ohler 1997 Synthesis of D-apio-β-D- furanosyl maleimide, an analogue of showdomycin with transposed hydroxymethyl group Monatsh. Chem. 128 183 190 1:CAS:528:DyaK2sXjs1Kitbk%3D 10.1007/BF00807307
    • (1997) Monatsh. Chem. , vol.128 , pp. 183-190
    • Hammerschmidt, F.1    Peric, B.2    Ohler, E.3
  • 22
    • 0023194835 scopus 로고
    • Phosphonylmethyl analogs of nucleotides and their derivatives: Chemistry and biology
    • 1:CAS:528:DyaL1cXhsFSrsLc%3D 10.1080/07328318708056188
    • A. Holy 1987 Phosphonylmethyl analogs of nucleotides and their derivatives: chemistry and biology Nucleosides Nucleotides 6 147 155 1:CAS:528:DyaL1cXhsFSrsLc%3D 10.1080/07328318708056188
    • (1987) Nucleosides Nucleotides , vol.6 , pp. 147-155
    • Holy, A.1
  • 23
    • 0025050434 scopus 로고
    • Microwave synthesis of 4-hydroxyquinazolinone
    • 1:CAS:528:DyaK3cXlsFagt7c%3D 2393953
    • M. Hori A. R. Iemur H. Hara A. Ozaki 1990 Microwave synthesis of 4-hydroxyquinazolinone Chem. Pharm. Bull. 38 1286 1291 1:CAS:528: DyaK3cXlsFagt7c%3D 2393953
    • (1990) Chem. Pharm. Bull. , vol.38 , pp. 1286-1291
    • Hori, M.1    Iemur, A.R.2    Hara, H.3    Ozaki, A.4
  • 24
    • 25844500311 scopus 로고    scopus 로고
    • Synthesis of 2-[3,5-substituted pyrazol-1-yl]-4,6-trisubstituted triazine derivatives as antimalarial agents
    • 1:CAS:528:DC%2BD2MXhtVynu7%2FJ 10.1016/j.bmcl.2005.08.023 16168643
    • S. B. Katiyar K. Srivastava S. K. Purib P. M. S. Chauhana 2005 Synthesis of 2-[3,5-substituted pyrazol-1-yl]-4,6-trisubstituted triazine derivatives as antimalarial agents Bioorg. Med. Chem. Lett. 15 4957 4960 1:CAS:528: DC%2BD2MXhtVynu7%2FJ 10.1016/j.bmcl.2005.08.023 16168643
    • (2005) Bioorg. Med. Chem. Lett. , vol.15 , pp. 4957-4960
    • Katiyar, S.B.1    Srivastava, K.2    Purib, S.K.3    Chauhana, P.M.S.4
  • 25
    • 1542486191 scopus 로고
    • Analytical applications of hydrazones
    • 1:CAS:528:DyaE2MXhsl2rtLg%3D 10.1016/0039-9140(75)80161-5 18961633
    • M. Katyal Y. Dutta 1975 Analytical applications of hydrazones Talanta 22 151 166 1:CAS:528:DyaE2MXhsl2rtLg%3D 10.1016/0039-9140(75)80161-5 18961633
    • (1975) Talanta , vol.22 , pp. 151-166
    • Katyal, M.1    Dutta, Y.2
  • 26
    • 0020961558 scopus 로고
    • Antiherpetic activity and mechanism of action of 9-(4-hydroxybutyl) guanine
    • 1:CAS:528:DyaL3sXlsFWkt7s%3D 10.1016/0166-3542(83)90028-1 6312878
    • A. Larsson S. Alenius N. G. Johnsson B. Oberg 1983 Antiherpetic activity and mechanism of action of 9-(4-hydroxybutyl) guanine Antiviral. Res. 3 77 86 1:CAS:528:DyaL3sXlsFWkt7s%3D 10.1016/0166-3542(83)90028-1 6312878
    • (1983) Antiviral. Res. , vol.3 , pp. 77-86
    • Larsson, A.1    Alenius, S.2    Johnsson, N.G.3    Oberg, B.4
  • 27
    • 0031470110 scopus 로고    scopus 로고
    • On the conformation of tiazofurin analogues
    • 1:CAS:528:DyaK2sXnt1Ogtbw%3D 10.1021/jm970129s 9406604
    • G. M. Makara G. M. Keseru 1997 On the conformation of tiazofurin analogues J. Med. Chem. 40 4154 4159 1:CAS:528:DyaK2sXnt1Ogtbw%3D 10.1021/jm970129s 9406604
    • (1997) J. Med. Chem. , vol.40 , pp. 4154-4159
    • Makara, G.M.1    Keseru, G.M.2
  • 28
    • 0027074210 scopus 로고
    • 4H-thieno[3,4-c]pyrazole derivatives with antiinflammatory, analgesic, antipyretic and platelet antiaggregating activities
    • 1:CAS:528:DyaK3sXhvVaqurs%3D 1294166
    • G. Menozzi L. Mosti P. Schenone M. D'Amico A. Filippelli F. Rossi 1992 4H-thieno[3,4-c]pyrazole derivatives with antiinflammatory, analgesic, antipyretic and platelet antiaggregating activities Farmaco 47 1495 511 1:CAS:528:DyaK3sXhvVaqurs%3D 1294166
    • (1992) Farmaco , vol.47 , pp. 1495-511
    • Menozzi, G.1    Mosti, L.2    Schenone, P.3    D'Amico, M.4    Filippelli, A.5    Rossi, F.6
  • 29
    • 0036171878 scopus 로고    scopus 로고
    • Synthesis and biological activity of some 4-substituted 1-[1-(2,3-dihydroxy-1-propoxy)methyl-1,2,3-triazol-(4 & 5)-ylmethyl]-1H- pyrazolo[3,4-d]pyrimidines
    • 1:CAS:528:DC%2BD38XhtF2isr0%3D 10.1016/S0014-827X(01)01152-1 11902642
    • O. Moukha-Chafiq M. L. Taha H. B. Lazrek J. J. Vasseur 2002 Synthesis and biological activity of some 4-substituted 1-[1-(2,3-dihydroxy-1-propoxy)methyl- 1,2,3-triazol-(4 & 5)-ylmethyl]-1H-pyrazolo[3,4-d]pyrimidines Farmaco 57 27 32 1:CAS:528:DC%2BD38XhtF2isr0%3D 10.1016/S0014-827X(01)01152-1 11902642
    • (2002) Farmaco , vol.57 , pp. 27-32
    • Moukha-Chafiq, O.1    Taha, M.L.2    Lazrek, H.B.3    Vasseur, J.J.4
  • 30
    • 0014278027 scopus 로고
    • Biologically active pyrazoles
    • 1:CAS:528:DyaF1cXhtFejt7s%3D 10.1002/jps.2600570401
    • R. E. Orth 1968 Biologically active pyrazoles J. Pharmaceutical Sci. 57 537 556 1:CAS:528:DyaF1cXhtFejt7s%3D 10.1002/jps.2600570401
    • (1968) J. Pharmaceutical Sci. , vol.57 , pp. 537-556
    • Orth, R.E.1
  • 31
    • 0018380346 scopus 로고
    • Synthesis of substituted 2-methyl-3-(3,4-dimethoxy/dihydroxyphenylethyl) 4-quinazolones as possible antiparkinson drugs
    • 10.1002/jhet.5570160307
    • S. S. Parmer S. P. Singh 1979 Synthesis of substituted 2-methyl-3-(3,4-dimethoxy/dihydroxyphenylethyl)4-quinazolones as possible antiparkinson drugs J. Heterocycl. Chem. 16 449 452 10.1002/jhet.5570160307
    • (1979) J. Heterocycl. Chem. , vol.16 , pp. 449-452
    • Parmer, S.S.1    Singh, S.P.2
  • 32
    • 0037205947 scopus 로고    scopus 로고
    • 1,3-Diphenylpyrazoles: Synthesis and antiparasitic activities of azomethine derivatives
    • 1:CAS:528:DC%2BD38XlvVGhu7k%3D 10.1016/S0223-5234(02)01388-0 12161064
    • P. Rathelot N. Azas H. El-Kashef F. Delmas 2002 1,3-Diphenylpyrazoles: synthesis and antiparasitic activities of azomethine derivatives Eur. J. Med. Chem. 37 671 679 1:CAS:528:DC%2BD38XlvVGhu7k%3D 10.1016/S0223-5234(02)01388-0 12161064
    • (2002) Eur. J. Med. Chem. , vol.37 , pp. 671-679
    • Rathelot, P.1    Azas, N.2    El-Kashef, H.3    Delmas, F.4
  • 33
    • 84936300247 scopus 로고
    • Acyclic nucleosides other than acyclovir as potential antiviral agents
    • 1:CAS:528:DyaL2MXlvFKgtL0%3D 10.1080/07328318508056172
    • R. J. Remy J. A. Secrist 1985 Acyclic nucleosides other than acyclovir as potential antiviral agents Nucleosides Nucleotides 4 411 427 1:CAS:528:DyaL2MXlvFKgtL0%3D 10.1080/07328318508056172
    • (1985) Nucleosides Nucleotides , vol.4 , pp. 411-427
    • Remy, R.J.1    Secrist, J.A.2
  • 34
    • 15444361739 scopus 로고    scopus 로고
    • Tyrosine kinase inhibitors. structureactivity relationships for methylamino-substituted derivatives of 4-[(3-bromophenyl)amino]-6-(methylamino)- pyrido[3,4-d]pyrimidine (PD 158780), a potent and specific inhibitor of the tyrosine kinase activity of receptors for the EGF family of growth factors
    • 1:CAS:528:DyaK1cXosFejsw%3D%3D 10.1021/jm970641d 9513602
    • G. W. Rewcastle D. K. Murray W. Elliot 1998 Tyrosine kinase inhibitors. structureactivity relationships for methylamino-substituted derivatives of 4-[(3-bromophenyl)amino]-6-(methylamino)-pyrido[3,4-d]pyrimidine (PD 158780), a potent and specific inhibitor of the tyrosine kinase activity of receptors for the EGF family of growth factors J. Med. Chem. 41 742 751 1:CAS:528: DyaK1cXosFejsw%3D%3D 10.1021/jm970641d 9513602
    • (1998) J. Med. Chem. , vol.41 , pp. 742-751
    • Rewcastle, G.W.1    Murray, D.K.2    Elliot, W.3
  • 35
    • 0036178191 scopus 로고    scopus 로고
    • Synthesis and antimicrobial activity of some new hydrazones of 4-fluorobenzoic acid hydrazide and 3-acetyl-2,5-disubstituted-1,3,4- oxadiazolines
    • 1:CAS:528:DC%2BD38XhsFCru7s%3D 10.1016/S0014-827X(01)01192-2 11902660
    • S. Rollas N. Gulerman H. Erdeniz 2002 Synthesis and antimicrobial activity of some new hydrazones of 4-fluorobenzoic acid hydrazide and 3-acetyl-2,5-disubstituted-1,3,4-oxadiazolines Farmaco 57 171 174 1:CAS:528:DC%2BD38XhsFCru7s%3D 10.1016/S0014-827X(01)01192-2 11902660
    • (2002) Farmaco , vol.57 , pp. 171-174
    • Rollas, S.1    Gulerman, N.2    Erdeniz, H.3
  • 36
    • 0345552086 scopus 로고
    • Synthesis of some 4h-3,1 benzoxazin-4-ones and 4-quinazolones and their reaction with hydrazines
    • 1:CAS:528:DyaE38XltFCgt7w%3D
    • A. Sammour M. I. B. Selim M. A. Abdo 1971 Synthesis of some 4h-3,1 benzoxazin-4-ones and 4-quinazolones and their reaction with hydrazines U.A.R. J. Chem. 14 197 205 1:CAS:528:DyaE38XltFCgt7w%3D
    • (1971) U.A.R. J. Chem. , vol.14 , pp. 197-205
    • Sammour, A.1    Selim, M.I.B.2    Abdo, M.A.3
  • 37
    • 0019193419 scopus 로고
    • Synthese von diamino- und trichloromethylaminoderivate der pyrazolkarbons/iure
    • 10.1002/zfch.19800200305
    • M. K. Spassova R. D. Zakharieva E. V. Golovinsky 1980 Synthese von diamino- und trichloromethylaminoderivate der pyrazolkarbons/iure Z. Chem. 20 95 96 10.1002/zfch.19800200305
    • (1980) Z. Chem. , vol.20 , pp. 95-96
    • Spassova, M.K.1    Zakharieva, R.D.2    Golovinsky, E.V.3
  • 38
    • 3042552189 scopus 로고    scopus 로고
    • Synthesis and antibacterial activity of a novel series of potent DNA gyrase inhibitors. Pyrazole Derivatives
    • 1:CAS:528:DC%2BD2cXksF2hs70%3D 10.1021/jm030394f 15214796
    • A. Tanitame Y. Oyamada K. Ofugi M. Fujimoto N. Iwai Y. Hiyama K. M. Suzuki J. Yamagishi 2004 Synthesis and antibacterial activity of a novel series of potent DNA gyrase inhibitors. Pyrazole Derivatives J. Med. Chem. 47 3693 3696 1:CAS:528:DC%2BD2cXksF2hs70%3D 10.1021/jm030394f 15214796
    • (2004) J. Med. Chem. , vol.47 , pp. 3693-3696
    • Tanitame, A.1    Oyamada, Y.2    Ofugi, K.3    Fujimoto, M.4    Iwai, N.5    Hiyama, Y.6    Suzuki, K.M.7    Yamagishi, J.8
  • 39
    • 0019522758 scopus 로고
    • Nicotinic acid hydrazide carcinogenesis in mice
    • 1:CAS:528:DyaL3MXhvVKls7o%3D 10.1159/000225532 7465158
    • B. Toth 1981 Nicotinic acid hydrazide carcinogenesis in mice Oncology 38 106 109 1:CAS:528:DyaL3MXhvVKls7o%3D 10.1159/000225532 7465158
    • (1981) Oncology , vol.38 , pp. 106-109
    • Toth, B.1
  • 40
    • 0020506475 scopus 로고
    • Synthesis of 3,4-dihydro-4-oxoquinazoline derivatives as potential anticonvulsants
    • 10.1021/jm00364a012
    • N. A. Vaidja C. H. Panos A. Kite W. B. Iturrian C. D. Blanton 1983 Synthesis of 3,4-dihydro-4-oxoquinazoline derivatives as potential anticonvulsants J. Med. Chem. 26 1422 1425 10.1021/jm00364a012
    • (1983) J. Med. Chem. , vol.26 , pp. 1422-1425
    • Vaidja, N.A.1    Panos, C.H.2    Kite, A.3    Iturrian, W.B.4    Blanton, C.D.5
  • 41
    • 0037046859 scopus 로고    scopus 로고
    • Hydrazones of 1,2-benzisothiazole hydrazides: Synthesis, antimicrobial activity and QSAR investigations
    • 1:CAS:528:DC%2BD38Xltlams7o%3D 10.1016/S0223-5234(02)01378-8 12126774
    • P. Vicini F. Zani P. Cozzini I. Doytchinova 2002 Hydrazones of 1,2-benzisothiazole hydrazides: synthesis, antimicrobial activity and QSAR investigations Eur. J. Med. Chem. 37 553 564 1:CAS:528:DC%2BD38Xltlams7o%3D 10.1016/S0223-5234(02)01378-8 12126774
    • (2002) Eur. J. Med. Chem. , vol.37 , pp. 553-564
    • Vicini, P.1    Zani, F.2    Cozzini, P.3    Doytchinova, I.4
  • 42
    • 0037405042 scopus 로고    scopus 로고
    • Recent developments in the field of quinazoline chemistry
    • 1:CAS:528:DC%2BD3sXivVemurk%3D 10.2174/1385272033486738
    • A. Witt A. Bergman 2003 Recent developments in the field of quinazoline chemistry Curr. Org. Chem. 7 659 677 1:CAS:528:DC%2BD3sXivVemurk%3D 10.2174/1385272033486738
    • (2003) Curr. Org. Chem. , vol.7 , pp. 659-677
    • Witt, A.1    Bergman, A.2


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.