Synthesis of 2-[3,5-substituted pyrazol-1-yl]-4,6-trisubstituted triazine derivatives as antimalarial agents

Bioorganic and Medicinal Chemistry Letters

Volumn 15, Issue 22, 2005, Pages 4957-4960

  Katiyar, Sanjay Babu ^a   Srivastava, Kumkum ^a   Puri, S K ^a   Chauhan, Prem M S ^a  

^a CENTRAL DRUG RESEARCH INSTITUTE   (India)

Author keywords

Antimalarial; Dihydrofolate reductase; Pyrazolyl triazine

Indexed keywords

ANTIMALARIAL AGENT; CYCLOGUANIL; TRIAZINE DERIVATIVE;

ANTIMALARIAL ACTIVITY; ARTICLE; CONTROLLED STUDY; DRUG POTENCY; DRUG STRUCTURE; DRUG SYNTHESIS; MINIMUM INHIBITORY CONCENTRATION; NONHUMAN; PLASMODIUM FALCIPARUM;

ANIMALS; ANTIMALARIALS; MOLECULAR STRUCTURE; PLASMODIUM FALCIPARUM; PYRAZOLES; STRUCTURE-ACTIVITY RELATIONSHIP; TRIAZINES;

PLASMODIUM FALCIPARUM;

EID: 25844500311     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2005.08.023     Document Type: Article

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