Design and synthesis of 3-(azol-1-yl)phenylpropanes as microbicidal spermicides for prophylactic contraception

Bioorganic and Medicinal Chemistry Letters

Volumn 21, Issue 1, 2011, Pages 176-181

  Kumar, Lalit ^a   Sarswat, Amit ^a   Lal, Nand ^a   Jain, Ashish ^a   Kumar, Sumit ^b   Kiran Kumar, S T V S ^a   Maikhuri, Jagdamba P ^a   Pandey, Atindra K ^a   Shukla, Praveen K ^a   Gupta, Gopal ^a   Sharma, Vishnu L ^a  

^a CENTRAL DRUG RESEARCH INSTITUTE   (India)

^b National Institute of Pharmaceutical Education and Research (NIPER)   (India)

Author keywords

Anticandida; Antitrichomonas; Fluoxetine; Nonoxynol 9; Spermicides

Indexed keywords

FLUCONAZOLE; METRONIDAZOLE; MICROBICIDE; NONOXINOL 9; SPERMICIDAL AGENT;

ANTIFUNGAL ACTIVITY; ANTIPROTOZOAL ACTIVITY; ARTICLE; CANDIDA; CONTRACEPTION; CYTOTOXICITY; DRUG DESIGN; DRUG POTENCY; DRUG SAFETY; DRUG SYNTHESIS; HUMAN; HUMAN CELL; IMMOBILIZED CELL; LACTOBACILLUS; MALE; MINIMUM INHIBITORY CONCENTRATION; NONHUMAN; SPERMATOZOON; TRICHOMONAS VAGINALIS; VAGINA FLORA;

ANTI-INFECTIVE AGENTS; ANTIFUNGAL AGENTS; CONTRACEPTIVE AGENTS, FEMALE; DRUG DESIGN; FEMALE; HELA CELLS; HUMANS; LACTOBACILLUS; PROPANE; SPERMATOCIDAL AGENTS; STRUCTURE-ACTIVITY RELATIONSHIP; TRICHOMONAS VAGINALIS;

LACTOBACILLUS; TRICHOMONAS VAGINALIS;

EID: 78650511625     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2010.11.042     Document Type: Article

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