메뉴 건너뛰기




Volumn 22, Issue 3, 2007, Pages 708-716

Novel disulphide esters of carbothioic acid as potent, non-detergent spermicides with low toxicity to Lactobacillus and HeLa cells in vitro

Author keywords

Contraception; Non detergent spermicides; Selective toxicity; Spermicidal activity

Indexed keywords

DISULFIDE; DSE 36 COMPOUND; DSE 37 COMPOUND; DSE-36 COMPOUND; DSE-37 COMPOUND; NONOXINOL; SPERMICIDAL AGENT; UNCLASSIFIED DRUG;

EID: 34247847906     PISSN: 02681161     EISSN: 14602350     Source Type: Journal    
DOI: 10.1093/humrep/del448     Document Type: Article
Times cited : (26)

References (35)
  • 1
    • 0036152866 scopus 로고    scopus 로고
    • Sperm apoptosis in fresh and cryopreserved bull semen detected by flow cytometry and its relationship with fertility
    • Anzar M, He L, Buhr MM, Kroetsch TG and Pauls KP (2002) Sperm apoptosis in fresh and cryopreserved bull semen detected by flow cytometry and its relationship with fertility. Biol Reprod 66,354-360.
    • (2002) Biol Reprod , vol.66 , pp. 354-360
    • Anzar, M.1    He, L.2    Buhr, M.M.3    Kroetsch, T.G.4    Pauls, K.P.5
  • 2
    • 33646259509 scopus 로고    scopus 로고
    • Volatile anaesthetics depolarize neural mitochondria by inhibition of the electron transport chain
    • Bains R, Moe MC, Larsen GA, Berg-Johnsen J and Vinje ML (2006) Volatile anaesthetics depolarize neural mitochondria by inhibition of the electron transport chain. Acta Anaesthesiol Scand 50,572-579.
    • (2006) Acta Anaesthesiol Scand , vol.50 , pp. 572-579
    • Bains, R.1    Moe, M.C.2    Larsen, G.A.3    Berg-Johnsen, J.4    Vinje, M.L.5
  • 5
    • 22044447481 scopus 로고    scopus 로고
    • Vaginal contraceptive activity of a chelated vanadocene
    • D'Cruz OJ and Uckun FM (2005) Vaginal contraceptive activity of a chelated vanadocene. Contraception 72,146-156.
    • (2005) Contraception , vol.72 , pp. 146-156
    • D'Cruz, O.J.1    Uckun, F.M.2
  • 6
    • 0031823092 scopus 로고    scopus 로고
    • Spermicidal activity of chelated complexes of bis(cyclopentadienyl) vanadium (IV)
    • D'Cruz OJ, Ghosh P and Uckun FM (1998a) Spermicidal activity of chelated complexes of bis(cyclopentadienyl) vanadium (IV). Mol Hum Reprod 4,683-693.
    • (1998) Mol Hum Reprod , vol.4 , pp. 683-693
    • D'Cruz, O.J.1    Ghosh, P.2    Uckun, F.M.3
  • 7
    • 0031810656 scopus 로고    scopus 로고
    • Spermicidal activity of metallocene complexes containing vanadium (IV) in humans
    • D'Cruz OJ, Ghosh P and Uckun FM (1998b) Spermicidal activity of metallocene complexes containing vanadium (IV) in humans. Biol Reprod 58,1515-1526.
    • (1998) Biol Reprod , vol.58 , pp. 1515-1526
    • D'Cruz, O.J.1    Ghosh, P.2    Uckun, F.M.3
  • 8
    • 32544454232 scopus 로고    scopus 로고
    • Exploiting common targets in human fertilization and HIV infection: Development of novel contraceptive microbicides
    • Doncel GF (2006) Exploiting common targets in human fertilization and HIV infection: development of novel contraceptive microbicides. Hum Reprod Update 12,103-117.
    • (2006) Hum Reprod Update , vol.12 , pp. 103-117
    • Doncel, G.F.1
  • 9
    • 0035882332 scopus 로고    scopus 로고
    • The molecular basis of nonoxynol-9-induced vaginal inflammation and its possible relevance to human immunodeficiency virus type 1 transmission
    • Fichorova RN, Tucker LD and Anderson DJ (2001) The molecular basis of nonoxynol-9-induced vaginal inflammation and its possible relevance to human immunodeficiency virus type 1 transmission. J Infect Dis 184,418-428.
    • (2001) J Infect Dis , vol.184 , pp. 418-428
    • Fichorova, R.N.1    Tucker, L.D.2    Anderson, D.J.3
  • 10
    • 32144433515 scopus 로고    scopus 로고
    • Microbicidal spermicide or spermicidal microbicide?
    • Gupta G (2005) Microbicidal spermicide or spermicidal microbicide? Eur J Contracept Reprod Health Care 10,212-218.
    • (2005) Eur J Contracept Reprod Health Care , vol.10 , pp. 212-218
    • Gupta, G.1
  • 11
    • 25144436593 scopus 로고    scopus 로고
    • Discovery of substituted isoxazolecarbaldehydes as potent spermicides, acrosin inhibitors and mild anti-fungal agents
    • Gupta G, Jain RK, Maikhuri JP, Shukla PK, Kumar M, Roy AK, Patra A, Singh V and Batra S (2005) Discovery of substituted isoxazolecarbaldehydes as potent spermicides, acrosin inhibitors and mild anti-fungal agents. Hum Reprod 20,2301-2308.
    • (2005) Hum Reprod , vol.20 , pp. 2301-2308
    • Gupta, G.1    Jain, R.K.2    Maikhuri, J.P.3    Shukla, P.K.4    Kumar, M.5    Roy, A.K.6    Patra, A.7    Singh, V.8    Batra, S.9
  • 14
    • 27744498389 scopus 로고    scopus 로고
    • Microbicides for prevention of transmission of sexually transmitted diseases
    • Howett MK and Kuhl JP (2005) Microbicides for prevention of transmission of sexually transmitted diseases. Curr Pharm Des 11,3731-3746.
    • (2005) Curr Pharm des , vol.11 , pp. 3731-3746
    • Howett, M.K.1    Kuhl, J.P.2
  • 15
    • 0021336185 scopus 로고
    • Development of an assay to assess the functional integrity of the human sperm membrane and its relationship to other semen characteristics
    • Jeyendran RS, Vander Ven HH, Perez-Pelaez M, Crabo BG and Zaneveld LJD (1984) Development of an assay to assess the functional integrity of the human sperm membrane and its relationship to other semen characteristics. J Reprod Fertil 70,219-228.
    • (1984) J Reprod Fertil , vol.70 , pp. 219-228
    • Jeyendran, R.S.1    Vander Ven, H.H.2    Perez-Pelaez, M.3    Crabo, B.G.4    Zaneveld, L.J.D.5
  • 18
    • 0035984827 scopus 로고    scopus 로고
    • Comparative in vitro sensitivities of human immune cell lines, vaginal and cervical epithelial cell lines, and primary cells to candidate microbicides nonoxynol 9, C31G, and sodium dodecyl sulfate
    • Krebs FC, Miller SR, Catalone BJ, Fichorova R, Anderson D, Malamud D, Howett MK and Wigdahl B (2002) Comparative in vitro sensitivities of human immune cell lines, vaginal and cervical epithelial cell lines, and primary cells to candidate microbicides nonoxynol 9, C31G, and sodium dodecyl sulfate. Antimicrob Agents Chemother 46,2292-2298.
    • (2002) Antimicrob Agents Chemother , vol.46 , pp. 2292-2298
    • Krebs, F.C.1    Miller, S.R.2    Catalone, B.J.3    Fichorova, R.4    Anderson, D.5    Malamud, D.6    Howett, M.K.7    Wigdahl, B.8
  • 19
    • 0037210258 scopus 로고    scopus 로고
    • Substituted acrylophenones and related mannich bases as possible spermicides and inhibitors of HIV envelope glycoprotein-CD4 interaction
    • Kumaria N, Dwivedi AK, Maikhuri JP, Gupta G, Habib S, Dhar JD and Singh S (2002) Substituted acrylophenones and related mannich bases as possible spermicides and inhibitors of HIV envelope glycoprotein-CD4 interaction. Eur J Med Chem 37,855-864.
    • (2002) Eur J Med Chem , vol.37 , pp. 855-864
    • Kumaria, N.1    Dwivedi, A.K.2    Maikhuri, J.P.3    Gupta, G.4    Habib, S.5    Dhar, J.D.6    Singh, S.7
  • 20
    • 0038058926 scopus 로고    scopus 로고
    • Mechanism of action of some acrylophenones, quinolines and dithiocarbamate as potent, non-detergent spermicidal agents
    • Maikhuri JP, Dwivedi AK, Dhar JD, Setty BS and Gupta G (2003) Mechanism of action of some acrylophenones, quinolines and dithiocarbamate as potent, non-detergent spermicidal agents. Contraception 67,403-408.
    • (2003) Contraception , vol.67 , pp. 403-408
    • Maikhuri, J.P.1    Dwivedi, A.K.2    Dhar, J.D.3    Setty, B.S.4    Gupta, G.5
  • 21
    • 0025369850 scopus 로고
    • The spermicidal compound nonoxynol-9 increases adhesion of Candida species to human epithelial cells in vitro
    • McGroarty JA, Soboh F, Bruce AW and Reid G (1990) The spermicidal compound nonoxynol-9 increases adhesion of Candida species to human epithelial cells in vitro. Infection Immunity 58,2005-2007.
    • (1990) Infection Immunity , vol.58 , pp. 2005-2007
    • McGroarty, J.A.1    Soboh, F.2    Bruce, A.W.3    Reid, G.4
  • 22
    • 0032577937 scopus 로고    scopus 로고
    • A regulatory role of sulfhydryl groups in modulation of sperm membrane conformation by heavy metals: Sulfhydryl groups as markers for infertility assessment
    • Nivsarkar M, Cherian B and Patel S (1998) A regulatory role of sulfhydryl groups in modulation of sperm membrane conformation by heavy metals: sulfhydryl groups as markers for infertility assessment. Biochem Biophys Res Commun 247,716-718.
    • (1998) Biochem Biophys Res Commun , vol.247 , pp. 716-718
    • Nivsarkar, M.1    Cherian, B.2    Patel, S.3
  • 23
    • 0035660614 scopus 로고    scopus 로고
    • Involvement of endometrial membrane sulphydryl groups in blastocyst implantation: Sulphydryl groups as a potential target for contraceptive research
    • Nivsarkar M, Sethi A, Bapu C, Patel M and Padh H (2001) Involvement of endometrial membrane sulphydryl groups in blastocyst implantation: sulphydryl groups as a potential target for contraceptive research. Contraception 64,255-259.
    • (2001) Contraception , vol.64 , pp. 255-259
    • Nivsarkar, M.1    Sethi, A.2    Bapu, C.3    Patel, M.4    Padh, H.5
  • 24
    • 0041828422 scopus 로고    scopus 로고
    • Effect of spermicides on Lactobacillus acidophilus in vitro-nonoxynol-9 vs. Sapindus saponins
    • Ojha P, Maikhuri JP and Gupta G (2003) Effect of spermicides on Lactobacillus acidophilus in vitro-nonoxynol-9 vs. Sapindus saponins. Contraception 68,135-138.
    • (2003) Contraception , vol.68 , pp. 135-138
    • Ojha, P.1    Maikhuri, J.P.2    Gupta, G.3
  • 25
    • 0001737437 scopus 로고
    • Practical method for testing the spermicidal action of chemical contraceptives
    • Sander FV and Cramer SD (1941) Practical method for testing the spermicidal action of chemical contraceptives. Hum Fertil 6,134-137.
    • (1941) Hum Fertil , vol.6 , pp. 134-137
    • Sander, F.V.1    Cramer, S.D.2
  • 27
    • 0027715835 scopus 로고
    • Methyl xanthine and altered biomembrane dynamics: Demonstration of protein mobility and enzyme inhibition by caffeine in sperm model system
    • Sinha S, Kumar P and Laloraya M (1993) Methyl xanthine and altered biomembrane dynamics: demonstration of protein mobility and enzyme inhibition by caffeine in sperm model system. Biochem Mol Biol Int 31,1141-1148.
    • (1993) Biochem Mol Biol Int , vol.31 , pp. 1141-1148
    • Sinha, S.1    Kumar, P.2    Laloraya, M.3
  • 30
    • 0034705969 scopus 로고    scopus 로고
    • Widely used spermicide may increase, not decrease, risk of HIV transmission
    • Stephenson J (2000) Widely used spermicide may increase, not decrease, risk of HIV transmission. JAMA 284,949.
    • (2000) JAMA , vol.284 , pp. 949
    • Stephenson, J.1
  • 31
  • 33
    • 0011143724 scopus 로고    scopus 로고
    • CONRAD WHO, Geneva
    • WHO/CONRAD (2001) Technical consultation on nonoxynol-9, WHO, Geneva (http://www.who.International/reproductive-health/publications/rhr-03-8/ Nonoxynol-9.pdf).
    • (2001) Technical Consultation on Nonoxynol-9
  • 34
    • 0029883862 scopus 로고    scopus 로고
    • Studies of human and rat blood under oxidative stress: Changes in plasma thiol level, antioxidant enzyme activity, protein carbonyl content, and fluidity of erythrocyte membrane
    • Yelinova V, Glazachev Y, Khramtsov V, Kudryashova L, Rykova V and Salganik R (1996) Studies of human and rat blood under oxidative stress: changes in plasma thiol level, antioxidant enzyme activity, protein carbonyl content, and fluidity of erythrocyte membrane. Biochem Biophys Res Commun 221,300-303.
    • (1996) Biochem Biophys Res Commun , vol.221 , pp. 300-303
    • Yelinova, V.1    Glazachev, Y.2    Khramtsov, V.3    Kudryashova, L.4    Rykova, V.5    Salganik, R.6


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.