Seeking ligand bias: Assessing GPCR coupling to β-arrestins for drug discovery

Drug Discovery Today: Technologies

Volumn 7, Issue 1, 2010, Pages

  Bohn, Laura M ^a   McDonald, Patricia H ^a  

^a SCRIPPS RESEARCH INSTITUTE   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ADRENERGIC RECEPTOR; BETA 2 ADRENERGIC RECEPTOR; BETA ADRENERGIC RECEPTOR BLOCKING AGENT; BETA ARRESTIN; BETA GALACTOSIDASE; BETA LACTAMASE; DOPAMINE RECEPTOR; ENHANCED GREEN FLUORESCENT PROTEIN; G PROTEIN COUPLED RECEPTOR; HORMONE; LIGAND; LUCIFERASE; MUTANT PROTEIN; NEUROTRANSMITTER; OPIATE RECEPTOR; PROTEINASE; YELLOW FLUORESCENT PROTEIN;

AGONIST; ARTICLE; ASSAY; BIOASSAY; BIOLUMINESCENCE; BIOLUMINESCENCE RESONANCE ENERGY TRANSFER; COST; DELETION MUTANT; DEVICE; DRUG RESEARCH; DRUG TARGETING; ENZYME ACTIVATION; ENZYME SUBSTRATE; FLUORESCENCE MICROSCOPY; FLUORESCENCE RESONANCE ENERGY TRANSFER; GENETIC TRANSCRIPTION; HIGH CONTENT SCREENING; HIGH THROUGHPUT SCREENING; MEDICAL TECHNOLOGY; MOLECULAR IMAGING; PROTEIN PROTEIN INTERACTION; RECEPTOR BLOCKING; REPORTER GENE; SECOND MESSENGER;

EID: 78649909159     PISSN: 17406749     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.ddtec.2010.06.005     Document Type: Review

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