GSK4112, a small molecule chemical probe for the cell biology of the nuclear heme receptor rev-erbα

ACS Chemical Biology

Volumn 5, Issue 10, 2010, Pages 925-932

  Grant, Daniel ^a   Yin, Lei ^b,c   Collins, Jon L ^a   Parks, Derek J ^a   Orband Miller, Lisa A ^a   Wisely, G Bruce ^a   Joshi, Shree ^b   Lazar, Mitchell A ^b   Willson, Timothy M ^a   Zuercher, William J ^a  

^a GLAXOSMITHKLINE   (United States)

^b UNIVERSITY OF PENNSYLVANIA   (United States)

^c UNIVERSITY OF MICHIGAN MEDICAL SCHOOL   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

AGENTS INTERACTING WITH TRANSMITTER, HORMONE OR DRUG RECEPTORS; CELL NUCLEUS RECEPTOR; GLUCOSE; GSK4112; HEME; NUCLEAR RECEPTOR COREPRESSOR; PROTEIN REV ERBALPHA; RECEPTOR INTERACTING PROTEIN 140; UNCLASSIFIED DRUG;

ARTICLE; CIRCADIAN RHYTHM; CYTOLOGY; GENE EXPRESSION; GENE REPRESSION; GLUCONEOGENESIS; LIVER CELL; METABOLISM; MOLECULAR PROBE; PRIORITY JOURNAL; PROTEIN PROTEIN INTERACTION; TRANSCRIPTION REGULATION;

AMINO ACID SEQUENCE; ANIMALS; BINDING, COMPETITIVE; CELL LINE; CELLS, CULTURED; CIRCADIAN RHYTHM; HEME; HEPATOCYTES; HUMANS; MALE; MICE; MICE, INBRED C57BL; MOLECULAR SEQUENCE DATA; NUCLEAR RECEPTOR CO-REPRESSOR 1; NUCLEAR RECEPTOR SUBFAMILY 1, GROUP D, MEMBER 1; PEPTIDES; PROTEIN INTERACTION MAPPING; SMALL MOLECULE LIBRARIES;

EID: 77958081830     PISSN: 15548929     EISSN: 15548937     Source Type: Journal    
DOI: 10.1021/cb100141y     Document Type: Article

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