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Volumn 18, Issue 19, 2010, Pages 7015-7021

Design, synthesis, and binding of homologated truncated 4′-thioadenosine derivatives at the human A3 adenosine receptors

(9) Lee, Hyuk Woo a Kim, Hea Ok a Choi, Won Jun a,b Choi, Sun a Lee, Jin Hee a Park, Seul Gi a Yoo, Lena c Jacobson, Kenneth A c Jeong, Lak Shin a

a Ewha Womans University (South Korea)

b Dongguk University (South Korea)

c NATIONAL INSTITUTE OF DIABETES AND DIGESTIVE AND KIDNEY DISEASES (United States)

Author keywords

A3 adenosine receptor; Binding affinity; Homologation; Truncated 4 thioadenosine

Indexed keywords

ADENOSINE A3 RECEPTOR; ADENOSINE A3 RECEPTOR ANTAGONIST; ADENOSINE DERIVATIVE; ADENOSINE RECEPTOR; CARBENE; NUCLEOSIDE; THIOADENOSINE; UNCLASSIFIED DRUG;

ARTICLE; BINDING AFFINITY; BINDING SITE; CHEMICAL BOND; DRUG DESIGN; HUMAN; SYNTHESIS;

ADENOSINE; ADENOSINE A3 RECEPTOR ANTAGONISTS; BINDING SITES; DRUG DESIGN; HUMANS; MODELS, MOLECULAR; MOLECULAR CONFORMATION; RECEPTOR, ADENOSINE A3; STEREOISOMERISM; STRUCTURE-ACTIVITY RELATIONSHIP; THIONUCLEOSIDES;

EID: 77956651324 PISSN: 09680896 EISSN: None Source Type: Journal
DOI: 10.1016/j.bmc.2010.08.018 Document Type: Article

Times cited : (15)

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