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Bioorganic and Medicinal Chemistry Letters

Volumn 20, Issue 17, 2010, Pages 5221-5224

Synthesis and SAR of (piperazin-1-yl-phenyl)-arylsulfonamides: A novel series of atypical antipsychotic agents

(5) Park, Chul Min a Kim, So Young a Park, Woo Kyu a Choi, Jung Hwan a Seong, Churl Min a

a Korea Research Institute of Chemical Technology (South Korea)

Author keywords

5 HT2C receptor; 5 HT6 receptor; Antagonist; Arylsulfonamide; Serotonin

Indexed keywords

ATYPICAL ANTIPSYCHOTIC AGENT; DOPAMINE 2 RECEPTOR; DOPAMINE 3 RECEPTOR; DOPAMINE 4 RECEPTOR; NAPHTHALENE 2 SULFONIC ACID ISOPROPYL[3 (4 METHYL PIPERAZIN 1 YL)PHENYL]AMIDE; SEROTONIN; SEROTONIN 6 RECEPTOR; SULFONAMIDE; UNCLASSIFIED DRUG;

ARTICLE; DRUG SYNTHESIS; STRUCTURE ACTIVITY RELATION;

ANTIPSYCHOTIC AGENTS; PIPERAZINES; RECEPTORS, SEROTONIN; STRUCTURE-ACTIVITY RELATIONSHIP; SULFONAMIDES;

EID: 77955659877 PISSN: 0960894X EISSN: None Source Type: Journal
DOI: 10.1016/j.bmcl.2010.06.150 Document Type: Article

Times cited : (5)

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