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Volumn 18, Issue 14, 2008, Pages 3844-3847

Synthesis and structure-activity relationship of 1H-indole-3-carboxylic acid pyridine-3-ylamides: A novel series of 5-HT2C receptor antagonists

Author keywords

5 HT2C receptor antagonists; Anxiety; Depression; GPCR

Indexed keywords

1H INDOLE 3 CARBOXYLIC ACID [6 (2 CHLOROPYRIDIN 3 YLOXY)PYRIDIN 3 YL]AMIDE; 5 METHYL 1 [[2 [(2 METHYL 3 PYRIDYL)OXY] 5 PYRIDYL]CARBAMOYL] 6 TRIFLUOROMETHYLINDOLINE; DOPAMINE 2 RECEPTOR; DOPAMINE 3 RECEPTOR; DOPAMINE 4 RECEPTOR; MESULERGINE; SEROTONIN 1A RECEPTOR; SEROTONIN 2A RECEPTOR; SEROTONIN 2C ANTAGONIST; SEROTONIN 6 RECEPTOR;

EID: 47149116818     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2008.06.064     Document Type: Article
Times cited : (23)

References (27)
  • 6
    • 47149094668 scopus 로고    scopus 로고
    • Bromidge, S. M.; Lovell, P. J.; Moss, S. F.; Serafinowska, H. T.; WO Patent 2002014273, 2002.
    • Bromidge, S. M.; Lovell, P. J.; Moss, S. F.; Serafinowska, H. T.; WO Patent 2002014273, 2002.
  • 7
    • 25844508919 scopus 로고    scopus 로고
    • Chem. Abstr. 136 (2002) 183704
    • (2002) Chem. Abstr. , vol.136 , pp. 183704
  • 10
    • 33748668483 scopus 로고    scopus 로고
    • King F.D. (Ed), The Royal Society of Chemistry, Cambridge, UK
    • Bromidge S.M. In: King F.D. (Ed). Medicinal Chemistry. 2nd ed. (2002), The Royal Society of Chemistry, Cambridge, UK 382-396
    • (2002) Medicinal Chemistry. 2nd ed. , pp. 382-396
    • Bromidge, S.M.1
  • 23
    • 47149106246 scopus 로고    scopus 로고
    • 50 (nM) values.
    • 50 (nM) values.
  • 24
    • 47149097119 scopus 로고    scopus 로고
    • 3 receptor in JP 03161470.
    • 3 receptor in JP 03161470.
  • 27
    • 47149113335 scopus 로고    scopus 로고
    • 35S]GTPγS was classified as an antagonist.
    • 35S]GTPγS was classified as an antagonist.


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.