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Volumn 18, Issue 14, 2010, Pages 4928-4938

Constrained peptidomimetics as antiplasmodial falcipain-2 inhibitors

(9) Bova, Floriana a Ettari, Roberta a Micale, Nicola a Carnovale, Caterina a Schirmeister, Tanja b Gelhaus, Christoph c Leippe, Matthias c Grasso, Silvana a Zappalà, Maria a

a UNIVERSITY OF MESSINA (Italy)

b UNIVERSITY OF WÜRZBURG (Germany)

c UNIVERSITY OF KIEL (Germany)

Author keywords

Cysteine proteases; Falcipain 2 inhibitors; Peptidomimetics; Rhodesain inhibitors

Indexed keywords

ANTITRYPANOSOMAL AGENT; CATHEPSIN B; CATHEPSIN L; CHLOROQUINE; CYSTEINE PROTEINASE INHIBITOR; FALCIPAIN 2; METHYL 4 [2 [3 [(ADAMANTAN 1 YLCARBAMOYLOXY)METHYL] 2 OXO 5 PHENYL 2,3 DIHYDRO 1H BENZO[E][1,4]DIAZEPIN 1 YL]ACETAMIDO]BUT 2 ENOATE; PEPTIDOMIMETIC AGENT; PROTOZOAL PROTEIN; RECOMBINANT ENZYME; RHODESAIN; UNCLASSIFIED DRUG;

ANTIPROTOZOAL ACTIVITY; ARTICLE; CELL CULTURE; CONTROLLED STUDY; DRUG MECHANISM; DRUG SCREENING; DRUG SELECTIVITY; DRUG SYNTHESIS; ENZYME INHIBITION; ERYTHROCYTE; HUMAN; HUMAN CELL; IC 50; NONHUMAN; PARASITE CULTIVATION; PARASITE VIABILITY; PLASMODIUM FALCIPARUM; STRUCTURE ACTIVITY RELATION; TRYPANOSOMA RHODESIENSE;

PLASMODIUM FALCIPARUM; TRYPANOSOMA BRUCEI RHODESIENSE;

EID: 77955337502 PISSN: 09680896 EISSN: None Source Type: Journal
DOI: 10.1016/j.bmc.2010.06.010 Document Type: Article

Times cited : (38)

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