Aziridide-based inhibitors of cathepsin L: Synthesis, inhibition activity, and docking studies

ChemMedChem

Volumn 1, Issue 10, 2006, Pages 1126-1141

  Vicik, Radim ^a   Busemann, Matthias ^a,d   Gelhaus, Christoph ^c   Stiefl, Nikolaus ^a   Scheiber, Josef ^a   Schmitz, Werner ^b   Schulz, Franziska ^a   Mladenovic, Milena ^a   Engels, Bernd ^a   Leippe, Matthias ^c   Baumann, Knut ^a   Schirmeister, Tanja ^a  

^a UNIVERSITY OF WÜRZBURG   (Germany)

^b UNIVERSITY OF WÜRZBURG   (Germany)

^c UNIVERSITY OF KIEL   (Germany)

^d 4SC AG   (Germany)

Author keywords

Aziridines; Cathepsins; Cysteine proteases docking; Inhibitors

Indexed keywords

EID: 33750310185     PISSN: 18607179     EISSN: 18607187     Source Type: Journal    
DOI: 10.1002/cmdc.200600106     Document Type: Article

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