SCOPUS 정보 검색 플랫폼

Bioorganic and Medicinal Chemistry Letters

Volumn 20, Issue 13, 2010, Pages 3863-3867

Activity of substituted thiophene sulfonamides against malarial and mammalian cyclin dependent protein kinases

(4) Caridha, Diana a Kathcart, April K a Jirage, Dayadevi a Waters, Norman C a

a WALTER REED ARMY INSTITUTE OF RESEARCH (United States)

Author keywords

Cancer; CDK inhibitor; CDK7; Cell cycle; Kinase; Malaria; Pfmrk; Plasmodium

Indexed keywords

ALSTERPAULLONE; ANTIMALARIAL AGENT; BENZENE DERIVATIVE; BENZENE SULFONAMIDE DERIVATIVE; BROMOHYDROSULFONYLACETAMIDE DERIVATIVE; CYCLIN DEPENDENT KINASE; CYCLIN DEPENDENT KINASE 1; CYCLIN DEPENDENT KINASE 2; CYCLIN DEPENDENT KINASE 6; CYCLIN DEPENDENT KINASE 7; CYCLIN DEPENDENT KINASE INHIBITOR; INDIRUBIN; MEFLOQUINE; PFMRK PROTEIN; SULFONAMIDE; THIOPHENE DERIVATIVE; THIOPHENE SULFONAMIDE DERIVATIVE; UNCLASSIFIED DRUG;

ANIMAL CELL; ANTIMALARIAL ACTIVITY; ANTIMALARIAL DRUG RESISTANCE; ARTICLE; CONTROLLED STUDY; DRUG POTENCY; HUMAN; HUMAN CELL; HUMAN CELL CULTURE; IC 50; IN VITRO STUDY; NONHUMAN; PLASMODIUM FALCIPARUM; RAT; SEQUENCE HOMOLOGY;

ANIMALS; ANTIMALARIALS; ANTINEOPLASTIC AGENTS; CELL LINE, TUMOR; CELL PROLIFERATION; CYCLIN-DEPENDENT KINASES; ENZYME INHIBITORS; HUMANS; MACROPHAGES; MICROBIAL SENSITIVITY TESTS; PLASMODIUM FALCIPARUM; RATS; STRUCTURE-ACTIVITY RELATIONSHIP; SULFONAMIDES; THIOPHENES;

EUKARYOTA; MAMMALIA; PLASMODIUM (APICOMPLEXA); PLASMODIUM FALCIPARUM;

EID: 77954312308 PISSN: 0960894X EISSN: None Source Type: Journal
DOI: 10.1016/j.bmcl.2010.05.039 Document Type: Article

Times cited : (35)

References (33)

1
- 0031466305
- D.O. Morgan Annu. Rev. Cell Dev. Biol. 13 1997 261
- (1997) Annu. Rev. Cell Dev. Biol. , vol.13 , pp. 261
- Morgan, D.O.¹

2
- 0035805201
- B.A. Edgar, and T.L. Orr-Weaver Cell 105 2001 297
- (2001) Cell , vol.105 , pp. 297
- Edgar, B.A.¹ Orr-Weaver, T.L.²

3
- 67649295460
- Z. Ullah, C.Y. Lee, and M.L. Depamphilis Cell Div. 4 2009 10
- (2009) Cell Div. , vol.4 , pp. 10
- Ullah, Z.¹ Lee, C.Y.² Depamphilis, M.L.³

4
- 49749107218
- P.E. Puig, M.N. Guilly, A. Bouchot, N. Droin, D. Cathelin, F. Bouyer, L. Favier, F. Ghiringhelli, G. Kroemer, E. Solary, F. Martin, and B. Chauffert Cell Biol. Int. 32 2008 1031
- (2008) Cell Biol. Int. , vol.32 , pp. 1031
- Puig, P.E.¹ Guilly, M.N.² Bouchot, A.³ Droin, N.⁴ Cathelin, D.⁵ Bouyer, F.⁶ Favier, L.⁷ Ghiringhelli, F.⁸ Kroemer, G.⁹ Solary, E.¹⁰ Martin, F.¹¹ Chauffert, B.¹²

5
- 37549036250
- M. Malumbres, P. Pevarello, M. Barbacid, and J.R. Bischoff Trends Pharmacol. Sci. 29 2008 16
- (2008) Trends Pharmacol. Sci. , vol.29 , pp. 16
- Malumbres, M.¹ Pevarello, P.² Barbacid, M.³ Bischoff, J.R.⁴

6
- 40049110045
- J.G. Breman, and C.N. Holloway Am. J. Trop. Med. Hyg. 77 2007 36
- (2007) Am. J. Trop. Med. Hyg. , vol.77 , pp. 36
- Breman, J.G.¹ Holloway, C.N.²

7
- 29144446249
- C. Doerig, O. Billker, D. Pratt, and J. Endicott Biochim. Biophys. Acta 1754 2005 132
- (2005) Biochim. Biophys. Acta , vol.1754 , pp. 132
- Doerig, C.¹ Billker, O.² Pratt, D.³ Endicott, J.⁴

8
- 33847720940
- F. Canduri, P.C. Perez, R.A. Caceres, and W.F. de Azevedo Jr. Curr. Drug Targets 8 2007 389
- (2007) Curr. Drug Targets , vol.8 , pp. 389
- Canduri, F.¹ Perez, P.C.² Caceres, R.A.³ De Azevedo, Jr.W.F.⁴

9
- 0028224015
- P.B. Ross-Macdonald, R. Graeser, B. Kappes, R. Franklin, and D.H. Williamson Eur. J. Biochem. 220 1994 693
- (1994) Eur. J. Biochem. , vol.220 , pp. 693
- Ross-Macdonald, P.B.¹ Graeser, R.² Kappes, B.³ Franklin, R.⁴ Williamson, D.H.⁵

10
- 0030581694
- R. Graeser, B. Wernli, R.M. Franklin, and B. Kappes Mol. Biochem. Parasitol. 82 1996 37
- (1996) Mol. Biochem. Parasitol. , vol.82 , pp. 37
- Graeser, R.¹ Wernli, B.² Franklin, R.M.³ Kappes, B.⁴

11
- 0029862051
- J.L. Li, K.J. Robson, J.L. Chen, G.A. Targett, and D.A. Baker Eur. J. Biochem. 241 1996 805
- (1996) Eur. J. Biochem. , vol.241 , pp. 805
- Li, J.L.¹ Robson, K.J.² Chen, J.L.³ Targett, G.A.⁴ Baker, D.A.⁵

12
- 0034654447
- N.C. Waters, C.L. Woodard, and S.T. Prigge Mol. Biochem. Parasitol. 107 2000 45
- (2000) Mol. Biochem. Parasitol. , vol.107 , pp. 45
- Waters, N.C.¹ Woodard, C.L.² Prigge, S.T.³

13
- 33745872589
- Y. Chen, D. Jirage, D. Caridha, A.K. Kathcart, E.A. Cortes, R.A. Dennull, J.A. Geyer, S.T. Prigge, and N.C. Waters Mol. Biochem. Parasitol. 149 2006 48
- (2006) Mol. Biochem. Parasitol. , vol.149 , pp. 48
- Chen, Y.¹ Jirage, D.² Caridha, D.³ Kathcart, A.K.⁴ Cortes, E.A.⁵ Dennull, R.A.⁶ Geyer, J.A.⁷ Prigge, S.T.⁸ Waters, N.C.⁹

14
- 77952547764
- D. Jirage, Y. Chen, M. O'Neil, D. Caridha, F. Eyase, W. Witola, B. Choukri, and N.C. Waters Mol. Biochem. Parasitol. 172 2010 9
- (2010) Mol. Biochem. Parasitol. , vol.172 , pp. 9
- Jirage, D.¹ Chen, Y.² O'Neil, M.³ Caridha, D.⁴ Eyase, F.⁵ Witola, W.⁶ Choukri, B.⁷ Waters, N.C.⁸

15
- 60649093106
- F.C. Koyama, D. Chakrabarti, and C.R. Garcia Mol. Biochem. Parasitol. 165 2009 1
- (2009) Mol. Biochem. Parasitol. , vol.165 , pp. 1
- Koyama, F.C.¹ Chakrabarti, D.² Garcia, C.R.³

16
- 0033631382
- C. Doerig, D. Chakrabarti, B. Kappes, and K. Mathews Prog. Cell Cycle Res. 2000 163
- (2000) Prog. Cell Cycle Res. , pp. 163
- Doerig, C.¹ Chakrabarti, D.² Kappes, B.³ Mathews, K.⁴

17
- 61849123390
- S. Holton, A. Merckx, D. Burgess, C. Deorig, M.E. Noble, and J. Endicott Structure 11 2003 1139
- (2003) Structure , vol.11 , pp. 1139
- Holton, S.¹ Merckx, A.² Burgess, D.³ Deorig, C.⁴ Noble, M.E.⁵ Endicott, J.⁶

18
- 12744281184
- S.M. Keenan, J.A. Geyer, W.J. Welsh, S.T. Prigge, and N.C. Waters Comb. Chem. High Throughput Screening 8 2005 27
- (2005) Comb. Chem. High Throughput Screening , vol.8 , pp. 27
- Keenan, S.M.¹ Geyer, J.A.² Welsh, W.J.³ Prigge, S.T.⁴ Waters, N.C.⁵

19
- 6044260115
- A.K. Bhattacharjee, J.A. Geyer, C.L. Woodard, A.K. Kathcart, D.A. Nichols, S.T. Prigge, Z. Li, B.T. Mott, and N.C. Waters J. Med. Chem. 47 2004 5418
- (2004) J. Med. Chem. , vol.47 , pp. 5418
- Bhattacharjee, A.K.¹ Geyer, J.A.² Woodard, C.L.³ Kathcart, A.K.⁴ Nichols, D.A.⁵ Prigge, S.T.⁶ Li, Z.⁷ Mott, B.T.⁸ Waters, N.C.⁹

20
- 24944573556
- Y. Peng, S.M. Keenan, and W.J. Welsh J. Mol. Graphics Modell. 24 2005 72
- (2005) J. Mol. Graphics Modell. , vol.24 , pp. 72
- Peng, Y.¹ Keenan, S.M.² Welsh, W.J.³

21
- 34547569777
- C.L. Woodard, S.M. Keenan, L. Gerena, W.J. Welsh, J.A. Geyer, and N.C. Waters Bioorg. Med. Chem. Lett. 17 2007 4961
- (2007) Bioorg. Med. Chem. Lett. , vol.17 , pp. 4961
- Woodard, C.L.¹ Keenan, S.M.² Gerena, L.³ Welsh, W.J.⁴ Geyer, J.A.⁵ Waters, N.C.⁶

22
- 0042420753
- C.L. Woodard, Z. Li, A.K. Kathcart, J. Terrell, L. Gerena, M. Lopez-Sanchez, D.E. Kyle, A.K. Bhattacharjee, D.A. Nichols, W. Ellis, S.T. Prigge, J.A. Geyer, and N.C. Waters J. Med. Chem. 46 2003 3877
- (2003) J. Med. Chem. , vol.46 , pp. 3877
- Woodard, C.L.¹ Li, Z.² Kathcart, A.K.³ Terrell, J.⁴ Gerena, L.⁵ Lopez-Sanchez, M.⁶ Kyle, D.E.⁷ Bhattacharjee, A.K.⁸ Nichols, D.A.⁹ Ellis, W.¹⁰ Prigge, S.T.¹¹ Geyer, J.A.¹² Waters, N.C.¹³

23
- 61849181566
- J.A. Geyer, S.M. Keenan, C.L. Woodard, P.A. Thompson, L. Gerena, D.A. Nichols, C.E. Gutteridge, and N.C. Waters Bioorg. Med. Chem. Lett. 19 2009 1982
- (2009) Bioorg. Med. Chem. Lett. , vol.19 , pp. 1982
- Geyer, J.A.¹ Keenan, S.M.² Woodard, C.L.³ Thompson, P.A.⁴ Gerena, L.⁵ Nichols, D.A.⁶ Gutteridge, C.E.⁷ Waters, N.C.⁸

24
- 0035814077
- Z. Xiao, N.C. Waters, C.L. Woodard, Z. Li, and P.K. Li Bioorg. Med. Chem. Lett. 11 2001 2875
- (2001) Bioorg. Med. Chem. Lett. , vol.11 , pp. 2875
- Xiao, Z.¹ Waters, N.C.² Woodard, C.L.³ Li, Z.⁴ Li, P.K.⁵

25
- 2942597981
- P.M. Fischer Curr. Med. Chem. 11 2004 1563
- (2004) Curr. Med. Chem. , vol.11 , pp. 1563
- Fischer, P.M.¹

26
- 1642323740
- M.E. Noble, J.A. Endicott, and L.N. Johnson Science 303 2004 1800
- (2004) Science , vol.303 , pp. 1800
- Noble, M.E.¹ Endicott, J.A.² Johnson, L.N.³

27
- 7944231428
- G. Lolli, E.D. Lowe, N.R. Brown, and L.N. Johnson Structure (Camb.) 12 2004 2067
- (2004) Structure (Camb.) , vol.12 , pp. 2067
- Lolli, G.¹ Lowe, E.D.² Brown, N.R.³ Johnson, L.N.⁴

28
- 0037168033
- T. Owa, A. Yokoi, K. Yamazaki, K. Yoshimatsu, T. Yamori, and T. Nagasu J. Med. Chem. 45 2002 4913
- (2002) J. Med. Chem. , vol.45 , pp. 4913
- Owa, T.¹ Yokoi, A.² Yamazaki, K.³ Yoshimatsu, K.⁴ Yamori, T.⁵ Nagasu, T.⁶

29
- 50849103033
- H.M. Faidallah, M.S. Al-Saadi, S.A.F. Rostom, and H.T.Y. Fahmy Med. Chem. Res. 16 2007 300
- (2007) Med. Chem. Res. , vol.16 , pp. 300
- Faidallah, H.M.¹ Al-Saadi, M.S.² Rostom, S.A.F.³ Fahmy, H.T.Y.⁴

30
- 0030756156
- K. Yoshimatsu, A. Yamaguchi, H. Yoshino, N. Koyanagi, and K. Kitoh Cancer Res. 57 1997 3208
- (1997) Cancer Res. , vol.57 , pp. 3208
- Yoshimatsu, K.¹ Yamaguchi, A.² Yoshino, H.³ Koyanagi, N.⁴ Kitoh, K.⁵

31
- 0033598320
- T. Owa, H. Yoshino, T. Okauchi, K. Yoshimatsu, Y. Ozawa, N.H. Sugi, T. Nagasu, N. Koyanagi, and K. Kitoh J. Med. Chem. 42 1999 3789
- (1999) J. Med. Chem. , vol.42 , pp. 3789
- Owa, T.¹ Yoshino, H.² Okauchi, T.³ Yoshimatsu, K.⁴ Ozawa, Y.⁵ Sugi, N.H.⁶ Nagasu, T.⁷ Koyanagi, N.⁸ Kitoh, K.⁹

32
- 0033614949
- C. Schultz, A. Link, M. Leost, D.W. Zaharevitz, R. Gussio, E.A. Sausville, L. Meijer, and C. Kunick J. Med. Chem. 42 1999 2909
- (1999) J. Med. Chem. , vol.42 , pp. 2909
- Schultz, C.¹ Link, A.² Leost, M.³ Zaharevitz, D.W.⁴ Gussio, R.⁵ Sausville, E.A.⁶ Meijer, L.⁷ Kunick, C.⁸

33
- 0035147448
- D. Marko, S. Schatzle, A. Friedel, A. Genzlinger, H. Zankl, L. Meijer, and G. Eisenbrand Br. J. Cancer 84 2001 283
- (2001) Br. J. Cancer , vol.84 , pp. 283
- Marko, D.¹ Schatzle, S.² Friedel, A.³ Genzlinger, A.⁴ Zankl, H.⁵ Meijer, L.⁶ Eisenbrand, G.⁷

* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.