메뉴 건너뛰기




Volumn 15, Issue 4, 2010, Pages 329-338

Evaluation of drug release kinetics and physico-chemical characteristics of metronidazole floating beads based on calcium silicate and gas-forming agents

Author keywords

alginate beads; calcium silicate; drug loading; kinetic of release; Metronidazole

Indexed keywords

ALGINIC ACID; CALCIUM SILICATE; METRONIDAZOLE; NANOBEAD; POROUS POLYMER; ANTIINFECTIVE AGENT; BICARBONATE; CALCIUM DERIVATIVE; DELAYED RELEASE FORMULATION; DRUG CARRIER; GLUCURONIC ACID; HEXURONIC ACID; SILICATE;

EID: 77954024807     PISSN: 10837450     EISSN: 10979867     Source Type: Journal    
DOI: 10.3109/10837450903196843     Document Type: Article
Times cited : (33)

References (28)
  • 1
    • 41549097189 scopus 로고    scopus 로고
    • Design and evaluation of floating multi-layer coated tablets based on gas formation
    • Sungthongjeen S, Sriamornsak P, Puttipipatkhachorn S. Design and evaluation of floating multi-layer coated tablets based on gas formation. Eur J Pharm Biopharm 2007;9(1):255-263.
    • (2007) Eur J Pharm Biopharm , vol.9 , Issue.1 , pp. 255-263
    • Sungthongjeen, S.1    Sriamornsak, P.2    Puttipipatkhachorn, S.3
  • 2
    • 0033991593 scopus 로고    scopus 로고
    • Floating drug delivery systems: An approach to oral controlled drug delivery via gastric retention
    • Singh BN, Kim KH. Floating drug delivery systems: An approach to oral controlled drug delivery via gastric retention. J Control Release 2000;63(3):235-259.
    • (2000) J Control Release , vol.63 , Issue.3 , pp. 235-259
    • Singh, B.N.1    Kim, K.H.2
  • 4
    • 30744435603 scopus 로고    scopus 로고
    • The use of citric acid to prolong the in vivo gastro-retention of a floating dosage form in the fasted state
    • DOI 10.1016/j.ijpharm.2005.09.036, PII S0378517305007088
    • Stops F, Fell JT, Collett JH, Martini LG, Sharma HL, Smith A-M. The use of citric acid to prolong the in vivo gastro-retention of a floating dosage form in the fasted state. Int J Pharm 2006;308:8-13. (Pubitemid 43097229)
    • (2006) International Journal of Pharmaceutics , vol.308 , Issue.1-2 , pp. 8-13
    • Stops, F.1    Fell, J.T.2    Collett, J.H.3    Martini, L.G.4    Sharma, H.L.5    Smith, A.-M.6
  • 5
    • 30744432383 scopus 로고    scopus 로고
    • Citric acid prolongs the gastro-retention of a floating dosage form and increases bioavailability of riboflavin in the fasted state
    • DOI 10.1016/j.ijpharm.2005.09.039, PII S0378517305007052
    • Stops F, Fell JT, Collett JH, Martini LG, Sharma H, Smith A-M. Citric acid prolongs the gastro-retention of a floating dosage form and increases bioavailability of riboflavin in the fasted state. Int J Pharm 2006;308:14-24. (Pubitemid 43097230)
    • (2006) International Journal of Pharmaceutics , vol.308 , Issue.1-2 , pp. 14-24
    • Stops, F.1    Fell, J.T.2    Collett, J.H.3    Martini, L.G.4    Sharma, H.L.5    Smith, A.-M.6
  • 6
    • 38349161002 scopus 로고    scopus 로고
    • Floating dosage forms to prolong gastro-retention - The characterisation of calcium alginate beads
    • Stops F, Fell JT, Collett JH, Martini LG. Floating dosage forms to prolong gastro-retention - the characterisation of calcium alginate beads. Int J Pharm 2008;350(1-2):301-311.
    • (2008) Int J Pharm , vol.350 , Issue.1-2 , pp. 301-311
    • Stops, F.1    Fell, J.T.2    Collett, J.H.3    Martini, L.G.4
  • 7
    • 24944474831 scopus 로고    scopus 로고
    • Calcium silicate based microspheres of repaglinide for gastroretentive floating drug delivery: Preparation and in vitro characterization
    • Jain SK, Awasthi AM, Jain NK, Agrawal GP. Calcium silicate based microspheres of repaglinide for gastroretentive floating drug delivery: Preparation and in vitro characterization. J Control Release 2005;107(2):300-309.
    • (2005) J Control Release , vol.107 , Issue.2 , pp. 300-309
    • Jain, S.K.1    Awasthi, A.M.2    Jain, N.K.3    Agrawal, G.P.4
  • 8
    • 0033848185 scopus 로고    scopus 로고
    • Use of floating alginate gel beads for stomach-specific drug delivery
    • Murata Y, Sasaki N, Miyamoto E, Kawashima S. Use of floating alginate gel beads for stomach-specific drug delivery. Eur J Pharm Biopharm 2000;50(2):221-226.
    • (2000) Eur J Pharm Biopharm , vol.50 , Issue.2 , pp. 221-226
    • Murata, Y.1    Sasaki, N.2    Miyamoto, E.3    Kawashima, S.4
  • 9
    • 33947590641 scopus 로고    scopus 로고
    • Development and evaluation of a novel floating in situ gelling system of amoxicillin for eradication of Helicobacter pylori
    • Rajinikanth PS, Balasubramaniam J, Mishra B. Development and evaluation of a novel floating in situ gelling system of amoxicillin for eradication of Helicobacter pylori. Int J Pharm 2007;335(1-2):114-122.
    • (2007) Int J Pharm , vol.335 , Issue.1-2 , pp. 114-122
    • Rajinikanth, P.S.1    Balasubramaniam, J.2    Mishra, B.3
  • 10
    • 0034605983 scopus 로고    scopus 로고
    • Amoxycillin release from a floating dosage form based on alginates
    • Whitehead L, Collett JH, Fell JT. Amoxycillin release from a floating dosage form based on alginates. Int J Pharm 2000;210(1-2):45-49.
    • (2000) Int J Pharm , vol.210 , Issue.1-2 , pp. 45-49
    • Whitehead, L.1    Collett, J.H.2    Fell, J.T.3
  • 11
    • 33745262063 scopus 로고    scopus 로고
    • A novel calcium silicate based microspheres of repaglinide: In vivo investigations
    • Jain SK, Agrawal GP, Jain NK. A novel calcium silicate based microspheres of repaglinide: In vivo investigations. J Control Release 2006;113(2):111-116.
    • (2006) J Control Release , vol.113 , Issue.2 , pp. 111-116
    • Jain, S.K.1    Agrawal, G.P.2    Jain, N.K.3
  • 12
    • 33750632215 scopus 로고    scopus 로고
    • The effect of drug concentration and curing time on processing and properties of calcium alginate beads containing metronidazole by response surface methodology
    • Patel YL, Sher P, Pawar AP. The effect of drug concentration and curing time on processing and properties of calcium alginate beads containing metronidazole by response surface methodology. AAPS PharmSciTech 2006;7(4):86.
    • (2006) AAPS PharmSciTech , vol.7 , Issue.4 , pp. 86
    • Patel, Y.L.1    Sher, P.2    Pawar, A.P.3
  • 13
    • 43449107981 scopus 로고    scopus 로고
    • Furosemise-loaded alginate microspheres prepared by ionic cross-linking technique: Morphology and release characteristics
    • Das MK, Senapati PC. Furosemise-loaded alginate microspheres prepared by ionic cross-linking technique: Morphology and release characteristics. Indian J Pharmaceut Sci 2008;70: 77-84.
    • (2008) Indian J Pharmaceut Sci , vol.70 , pp. 77-84
    • Das, M.K.1    Senapati, P.C.2
  • 14
    • 34247173293 scopus 로고    scopus 로고
    • Development of hollow/ porous calcium pectinate beads for floating-pulsatile drug delivery
    • Badve SS, Sher P, Korde A, Pawar AP. Development of hollow/ porous calcium pectinate beads for floating-pulsatile drug delivery. Eur J Pharm Biopharm 2007;65(1):85-93.
    • (2007) Eur J Pharm Biopharm , vol.65 , Issue.1 , pp. 85-93
    • Badve, S.S.1    Sher, P.2    Korde, A.3    Pawar, A.P.4
  • 15
    • 0037370868 scopus 로고    scopus 로고
    • Alginate-diltiazem hydrochloride beads: Optimization of formulation factors, in vitro and in vivo availability
    • El-Kamel AH, Al-Gohary OM, Hosny EA. Alginate-diltiazem hydrochloride beads: Optimization of formulation factors, in vitro and in vivo availability. J Microencapsul 2003;20(2):211-225.
    • (2003) J Microencapsul , vol.20 , Issue.2 , pp. 211-225
    • El-Kamel, A.H.1    Al-Gohary, O.M.2    Hosny, E.A.3
  • 16
    • 0035073301 scopus 로고    scopus 로고
    • Modeling and comparison of dissolution profiles
    • Costa P, Sousa Lobo JM. Modeling and comparison of dissolution profiles. Eur J Pharm Sci 2001;13(2):123-133.
    • (2001) Eur J Pharm Sci , vol.13 , Issue.2 , pp. 123-133
    • Costa, P.1    Sousa Lobo, J.M.2
  • 17
    • 33845960792 scopus 로고    scopus 로고
    • Kinetic analysis of chlorpropamide dissolution from 17 solid dispersions
    • Barzegar-Jalali M, Dastmalchi S. Kinetic analysis of chlorpropamide dissolution from 17 solid dispersions. Drug Dev Ind Pharm 2007;33(1):63-70.
    • (2007) Drug Dev Ind Pharm , vol.33 , Issue.1 , pp. 63-70
    • Barzegar-Jalali, M.1    Dastmalchi, S.2
  • 18
    • 0014592606 scopus 로고
    • Interpretation of percent dissolved-time plots derived from in vitro testing of conventional tablets and capsules
    • Wagner JG. Interpretation of percent dissolved-time plots derived from in vitro testing of conventional tablets and capsules. J Pharm Sci 1969;58(10):1253-1257.
    • (1969) J Pharm Sci , vol.58 , Issue.10 , pp. 1253-1257
    • Wagner, J.G.1
  • 20
    • 0025013269 scopus 로고
    • A model for linearizing drug dissolution data
    • Barzegar-Jalali M. A model for linearizing drug dissolution data. Int J Pharm 1990;63:R6-11.
    • (1990) Int J Pharm , vol.63
    • Barzegar-Jalali, M.1
  • 21
    • 11144234232 scopus 로고    scopus 로고
    • Preparation of chitosan beads by simultaneous cross-linking/ insolubilisation in basic pH. Rheological optimisation and drug loading/release behaviour
    • Barreiro-Iglesias R, Coronilla R, Concheiro A, Varez-Lorenzo C. Preparation of chitosan beads by simultaneous cross-linking/ insolubilisation in basic pH. Rheological optimisation and drug loading/release behaviour. Eur J Pharm Sci 2005;24(1):77-84.
    • (2005) Eur J Pharm Sci , vol.24 , Issue.1 , pp. 77-84
    • Barreiro-Iglesias, R.1    Coronilla, R.2    Concheiro, A.3    Varez-Lorenzo, C.4
  • 22
    • 0037018959 scopus 로고    scopus 로고
    • Preparation of alginate beads for floating drug delivery system: Effects of CO(2) gasforming agents
    • Choi BY, Park HJ, Hwang SJ, Park JB. Preparation of alginate beads for floating drug delivery system: Effects of CO(2) gasforming agents. Int J Pharm 2002;239(1-2):81-91.
    • (2002) Int J Pharm , vol.239 , Issue.1-2 , pp. 81-91
    • Choi, B.Y.1    Park, H.J.2    Hwang, S.J.3    Park, J.B.4
  • 23
    • 33751253485 scopus 로고    scopus 로고
    • Evaluation of porous carrierbased floating orlistat microspheres for gastric delivery
    • Jain SK, Agrawal GP, Jain NK. Evaluation of porous carrierbased floating orlistat microspheres for gastric delivery. AAPS PharmSciTech 2006;7(4):90.
    • (2006) AAPS PharmSciTech , vol.7 , Issue.4 , pp. 90
    • Jain, S.K.1    Agrawal, G.P.2    Jain, N.K.3
  • 24
    • 40949123807 scopus 로고    scopus 로고
    • Effect of core and surface cross-linking on the entrapment of metronidazole in pectin beads
    • Pawar AP, Gadhe AR, Venkatachalam P, Sher P, Mahadik KR. Effect of core and surface cross-linking on the entrapment of metronidazole in pectin beads. Acta Pharm 2008;58(1):78-85.
    • (2008) Acta Pharm , vol.58 , Issue.1 , pp. 78-85
    • Pawar, A.P.1    Gadhe, A.R.2    Venkatachalam, P.3    Sher, P.4    Mahadik, K.R.5
  • 25
    • 0037422349 scopus 로고    scopus 로고
    • Effect of HPMC and carbopol on the release and floating properties of gastric floating drug delivery system using factorial design
    • Li S, Lin S, Daggy BP, Mirchandani HL, Chien YW. Effect of HPMC and carbopol on the release and floating properties of gastric floating drug delivery system using factorial design. Int J Pharm 2003;253(1-2):13-22.
    • (2003) Int J Pharm , vol.253 , Issue.1-2 , pp. 13-22
    • Li, S.1    Lin, S.2    Daggy, B.P.3    Mirchandani, H.L.4    Chien, Y.W.5
  • 26
    • 24744457523 scopus 로고    scopus 로고
    • Alginate-coated alginate-polyethyleneimine beads for prolonged release of furosemide in simulated intestinal fluid
    • Setty CM, Sahoo SS, Sa B. Alginate-coated alginate-polyethyleneimine beads for prolonged release of furosemide in simulated intestinal fluid. Drug Dev Ind Pharm 2005;(4-5):435-446.
    • (2005) Drug Dev Ind Pharm , vol.4-5 , pp. 435-446
    • Setty, C.M.1    Sahoo, S.S.2    Sa, B.3
  • 27
    • 14144252473 scopus 로고    scopus 로고
    • Emulsion gel beads of calcium pectinate capable of floating on the gastric fluid: Effect of some additives, hardening agent or coating on release behavior of metronidazole
    • Sriamornsak P, Thirawong N, Puttipipatkhachorn S. Emulsion gel beads of calcium pectinate capable of floating on the gastric fluid: Effect of some additives, hardening agent or coating on release behavior of metronidazole. Eur J Pharm Sci 2005;24(4):363-373.
    • (2005) Eur J Pharm Sci , vol.24 , Issue.4 , pp. 363-373
    • Sriamornsak, P.1    Thirawong, N.2    Puttipipatkhachorn, S.3
  • 28
    • 33645321628 scopus 로고    scopus 로고
    • Low density multiparticulate system for pulsatile release of meloxicam
    • Sharma S, Pawar A. Low density multiparticulate system for pulsatile release of meloxicam. Int J Pharm 2006;313(1-2):150-158.
    • (2006) Int J Pharm , vol.313 , Issue.1-2 , pp. 150-158
    • Sharma, S.1    Pawar, A.2


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.