Ligand-dependent assembly of pregnane X receptor, constitutive androstane receptor and liver X receptor is applicable to identify ligands

Drug Metabolism Letters

Volumn 4, Issue 2, 2010, Pages 88-94

  Kobayashi, Kaoru ^a   Saito, Kosuke ^a   Takagi, Sachiko ^a   Chiba, Kan ^a  

^a CHIBA UNIVERSITY   (Japan)

Author keywords

Constitutive androstane receptor; Ligand; Liver X receptor; Mammalian two hybrid assay; Nuclear receptor; Pregnane X receptor

Indexed keywords

6 (4 CHLOROPHENYL)IMIDAZO[2,1 B][1,3]THIAZOLEB][1,3]THIAZOLE 5 CARBALDEHYDE O (3,4 DICHLOROBENZYL)OXIME; CONSTITUTIVE ANDROSTANE RECEPTOR; LIVER X RECEPTOR; N (2,2,2 TRIFLUOROETHYL) N [4 [2,2,2 TRIFLUORO 1 HYDROXY 1 (TRIFLUOROMETHOXY)ETHYL]PHENYL]BENZENESULFONAMIDE; OXIME DERIVATIVE; PREGNANE X RECEPTOR; RIFAMPICIN; UNCLASSIFIED DRUG; CELL RECEPTOR; LIGAND; ORPHAN NUCLEAR RECEPTOR; RECOMBINANT PROTEIN; STEROID RECEPTOR;

AMINO TERMINAL SEQUENCE; ARTICLE; CARBOXY TERMINAL SEQUENCE; CONTROLLED STUDY; HUMAN; HUMAN CELL; LIGAND BINDING; NUCLEOTIDE SEQUENCE; PRIORITY JOURNAL; PROTEIN ASSEMBLY; PROTEIN CONFORMATION; ANIMAL; BINDING SITE; BIOSYNTHESIS; DOSE RESPONSE; GENETIC TRANSFECTION; METABOLISM; MOUSE; PLASMID; RAT;

MAMMALIA;

ANIMALS; BINDING SITES; DOSE-RESPONSE RELATIONSHIP, DRUG; HUMANS; LIGANDS; MICE; ORPHAN NUCLEAR RECEPTORS; PLASMIDS; RATS; RECEPTORS, CYTOPLASMIC AND NUCLEAR; RECEPTORS, STEROID; RECOMBINANT PROTEINS; TRANSFECTION;

EID: 77953800582     PISSN: 18723128     EISSN: None     Source Type: Journal    
DOI: 10.2174/187231210791292744     Document Type: Article

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