Online fluorescence enhancement assay for the acetylcholine binding protein with parallel mass spectrometric identification

Journal of Medicinal Chemistry

Volumn 53, Issue 12, 2010, Pages 4720-4730

  Kool, Jeroen ^a   De Kloe, Gerdien E ^a   Bruyneel, Ben ^a   De Vlieger, Jon S ^a   Retra, Kim ^a   Wijtmans, Maikel ^a   Van Elk, Rene ^a   Smit, August B ^a   Leurs, Rob ^a   Lingeman, Henk ^a   De Esch, Iwan J P ^a   Irth, Hubertus ^a  

^a VU UNIVERSITY AMSTERDAM   (Netherlands)

Author keywords

[No Author keywords available]

Indexed keywords

ACETYLCHOLINE; EPIBATIDINE; NICOTINE; NICOTINIC RECEPTOR;

ARTICLE; BINDING AFFINITY; DRUG RECEPTOR BINDING; FLUORESCENCE; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; IC 50; MASS SPECTROMETRY; PROTEIN BINDING; PROTEIN DOMAIN; STRUCTURE ACTIVITY RELATION;

ANABASINE; BINDING SITES; CARRIER PROTEINS; CHROMATOGRAPHY, LIQUID; DRUG DISCOVERY; FLOW INJECTION ANALYSIS; FLUOROMETRY; LIGANDS; MASS SPECTROMETRY; PROTEIN BINDING; RADIOLIGAND ASSAY; REPRODUCIBILITY OF RESULTS;

EID: 77953749427     PISSN: 00222623     EISSN: 15204804     Source Type: Journal    
DOI: 10.1021/jm100230k     Document Type: Article

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