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Volumn 46, Issue 23, 2010, Pages 4021-4042

Total synthesis of (+)-A83586C, (+)-kettapeptin and (+)-azinothricin: Powerful new inhibitors of β-catenin/TCF4-and E2F-mediated gene transcription

(3) Hale, Karl J a Manaviazar, Soraya a George, Jonathan b

a QUEEN'S UNIVERSITY BELFAST (United Kingdom)

b UNIVERSITY OF OXFORD (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

A 83586C; ANTIBIOTIC AGENT; ANTIINFECTIVE AGENT; ANTINEOPLASTIC AGENT; ANTINEOPLASTIC ANTIBIOTIC; AZINOTHRICIN; BETA CATENIN; CITROPEPTIN; GE 3; KETTAPEPTIN; MITOMYCIN C; OSTEOPONTIN; PIPALAMYCIN; POLYOXYPEPTIN A; TACROLIMUS; TRANSCRIPTION FACTOR E2F; UNCLASSIFIED DRUG; VERUCOPEPTIN; BASIC HELIX LOOP HELIX LEUCINE ZIPPER TRANSCRIPTION FACTOR; DEPSIPEPTIDE; PEPTIDE; TCF4 PROTEIN, HUMAN; TRANSCRIPTION FACTOR;

ANTINEOPLASTIC ACTIVITY; ASYMMETRIC SYNTHESIS; CANCER CELL; COLON CANCER; DRUG MECHANISM; DRUG STRUCTURE; DRUG SYNTHESIS; GENETIC TRANSCRIPTION; HUMAN; METASTASIS; MINIMUM INHIBITORY CONCENTRATION; NONHUMAN; REVIEW; SINGLE DRUG DOSE; STREPTOMYCES; ANTAGONISTS AND INHIBITORS; COLONIC NEOPLASMS; DRUG EFFECTS; GENETICS; METABOLISM; SYNTHESIS; TUMOR CELL LINE;

BASIC HELIX-LOOP-HELIX LEUCINE ZIPPER TRANSCRIPTION FACTORS; BETA CATENIN; CELL LINE, TUMOR; COLONIC NEOPLASMS; DEPSIPEPTIDES; E2F TRANSCRIPTION FACTORS; HUMANS; PEPTIDES; TRANSCRIPTION FACTORS; TRANSCRIPTION, GENETIC;

EID: 77953202408 PISSN: 13597345 EISSN: None Source Type: Journal
DOI: 10.1039/c000603c Document Type: Review

Times cited : (29)

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