A cell-based assay that targets methionine aminopeptidase in a physiologically relevant environment

Bioorganic and Medicinal Chemistry Letters

Volumn 20, Issue 7, 2010, Pages 2129-2132

  Chai, Sergio C ^a   Ye, Qi Zhuang ^a  

^a INDIANA UNIVERSITY SCHOOL OF MEDICINE   (United States)

Author keywords

Antibacterial; Cell based assay; Drug screening; Enzyme inhibitor; Metalloenzyme

Indexed keywords

ENZYME INHIBITOR; METHIONYL AMINOPEPTIDASE;

ARTICLE; BACTERIAL CELL; CELL ASSAY; CONTROLLED STUDY; ENVIRONMENT; ESCHERICHIA COLI; HYDROLYSIS; MONITORING; NONHUMAN; PROTEIN EXPRESSION; VALIDATION STUDY;

AMINOPEPTIDASES; ANTI-BACTERIAL AGENTS; DRUG EVALUATION, PRECLINICAL; ENZYME INHIBITORS; ESCHERICHIA COLI; UP-REGULATION;

BACTERIA (MICROORGANISMS); ESCHERICHIA COLI;

EID: 77949485581     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2010.02.052     Document Type: Article

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