Inhibition of ErbB2(Her2) expression with small molecule transcription factor mimics

Bioorganic and Medicinal Chemistry Letters

Volumn 19, Issue 21, 2009, Pages 6233-6236

  Lee, Lori W ^a   Taylor, Christopher E C ^a   Desaulniers, Jean Paul ^a   Zhang, Manchao ^b   Højfeldt, Jonas W ^a   Pan, Quintin ^b   Mapp, Anna K ^a  

^a UNIVERSITY OF MICHIGAN   (United States)

^b THE OHIO STATE UNIVERSITY WEXNER MEDICAL CENTER   (United States)

Author keywords

ErbB2; ESX; Her2; Tanscriptional inhibitor

Indexed keywords

EPIDERMAL GROWTH FACTOR RECEPTOR 2; ISOXAZOLIDINE DERIVATIVE; TRANSCRIPTION FACTOR; TRANSCRIPTION FACTOR ESX; UNCLASSIFIED DRUG;

ANTINEOPLASTIC ACTIVITY; ARTICLE; CANCER CELL; CELL GROWTH; CELL PROLIFERATION; CELL SURFACE; CONTROLLED STUDY; ENZYME INHIBITION; GENE EXPRESSION; GENE OVEREXPRESSION; HUMAN; HUMAN CELL; MOLECULAR MIMICRY; PROTEIN LOCALIZATION; PROTEIN MODIFICATION; TRANSCRIPTION INITIATION;

CELL LINE, TUMOR; GENE EXPRESSION REGULATION, NEOPLASTIC; HUMANS; ISOXAZOLES; RECEPTOR, ERBB-2; TRANSCRIPTION FACTORS; TRANSCRIPTIONAL ACTIVATION;

EUKARYOTA;

EID: 71749098575     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2009.08.090     Document Type: Article

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