An estimation of β 2-adrenoceptor reserve on human bronchial smooth muscle for some sympathomimetic bronchodilators

British Journal of Pharmacology

Volumn 158, Issue 1, 2009, Pages 287-299

  Giembycz, Mark A ^a  

^a UNIVERSITY OF CALGARY   (Canada)

Author keywords

2 adrenoceptor reserve; Agonist affinity estimation; Airways smooth muscle; Asthma; Bronchodilatation; Comparative method; DCITC; Fractional receptor inactivation; Operational curve fitting

Indexed keywords

BETA 2 ADRENERGIC RECEPTOR; FORMOTEROL; METHACHOLINE; PROCATEROL; SALBUTAMOL; TERBUTALINE;

ADOLESCENT; ADRENERGIC ACTIVITY; ADULT; ANIMAL CELL; ARTICLE; BRONCHUS MUSCLE; DRUG RECEPTOR BINDING; EOSINOPHIL; FEMALE; GUINEA PIG; HUMAN; HUMAN TISSUE; INTRINSIC SYMPATHOMIMETIC ACTIVITY; MALE; NONHUMAN; PRIORITY JOURNAL; RECEPTOR AFFINITY; RESPIRATORY BURST;

ADOLESCENT; ADULT; ALBUTEROL; ANIMALS; BRONCHI; BRONCHODILATOR AGENTS; FEMALE; GUINEA PIGS; HUMANS; MALE; MIDDLE AGED; MODELS, BIOLOGICAL; MUSCLE, SMOOTH; PROTEIN BINDING; RECEPTORS, ADRENERGIC, BETA-2; SYMPATHOMIMETICS; TERBUTALINE; YOUNG ADULT;

EID: 69249202370     PISSN: 00071188     EISSN: 14765381     Source Type: Journal    
DOI: 10.1111/j.1476-5381.2009.00277.x     Document Type: Article

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