Kinetic analysis of drug-receptor interactions of long-acting β2 sympathomimetics in isolated receptor membranes: Evidence against prolonged effects of salmeterol and formoterol on receptor-coupled adenylyl cyclase

Journal of Pharmacology and Experimental Therapeutics

Volumn 288, Issue 3, 1999, Pages 1084-1092

  Teschemacher, Andrea ^a   Lemoine, Horst ^a  

^a HEINRICH HEINE UNIVERSITY   (Germany)

Author keywords

[No Author keywords available]

Indexed keywords

ADENYLATE CYCLASE; BETA 2 ADRENERGIC RECEPTOR; FORMOTEROL; IODINE 125; IODOPINDOLOL; ISOPRENALINE; SALMETEROL;

ANIMAL CELL; ARTICLE; DISSOCIATION; DRUG DIFFUSION; DRUG HALF LIFE; DRUG RECEPTOR BINDING; LIPOPHILICITY; LUNG ALVEOLUS CELL; NONHUMAN; PRIORITY JOURNAL; RAT; RECEPTOR AFFINITY; TRACHEA MUCOSA;

ADENYLATE CYCLASE; ADRENERGIC BETA-AGONISTS; ADRENERGIC BETA-ANTAGONISTS; ALBUTEROL; ANIMALS; BINDING, COMPETITIVE; BRONCHODILATOR AGENTS; CATTLE; CELL MEMBRANE; ETHANOLAMINES; ISOPROTERENOL; LUNG; MEMBRANES; MUSCLE, SMOOTH; PINDOLOL; RADIOLIGAND ASSAY; RATS; RECEPTORS, DRUG; SYMPATHOMIMETICS; TRACHEA;

EID: 0032982607     PISSN: 00223565     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

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