Novel 4-(morpholin-4-yl)-N′-(arylidene)benzohydrazides: Synthesis, antimycobacterial activity and QSAR investigations

European Journal of Medicinal Chemistry

Volumn 44, Issue 10, 2009, Pages 3954-3960

  Raparti, Vyankatesh ^a   Chitre, Trupti ^a   Bothara, Kailas ^a   Kumar, Vanaja ^b   Dangre, Sudarshan ^a   Khachane, Chetan ^a   Gore, Suraj ^a   Deshmane, Bhavana ^a  

^a AISSMS COLLEGE OF PHARMACY   (India)

^b NATIONAL INSTITUTE FOR RESEARCH IN TUBERCULOSIS   (India)

Author keywords

2D QSAR; 3D QSAR; Antimycobacterial; Morpholine; Schiff base

Indexed keywords

4 (MORPHOLIN 4 YL) N' (3 PHENYLALLYLIDENE)BENZOHYDRAZIDE; 4 (MORPHOLIN 4 YL) N' (4 CHLOROBENZYLIDENE)BENZOHYDRAZIDE; 4 (MORPHOLIN 4 YL) N' (4 FLUOROBENZYLIDENE)BENZOHYDRAZIDE; 4 (MORPHOLIN 4 YL) N' (4 METHOXYBENZYLIDENE)BENZOHYDRAZIDE; 4 (MORPHOLIN 4 YL) N' (4 METHYLBENZYLIDENE)BENZOHYDRAZIDE; 4 (MORPHOLIN 4 YL) N' (FURAN 2 YLIDENE)BENZOHYDRAZIDE; 4 CHLOROBENZONITRILE; ANTIMYCOBACTERIAL AGENT; BENZONITRILE; BENZYLIDENE DERIVATIVE; HYDRAZIDE DERIVATIVE; ISONIAZID; LUCIFERASE; MORPHOLINE; UNCLASSIFIED DRUG;

ANTIBACTERIAL ACTIVITY; ARTICLE; BACTERIAL STRAIN; CONTROLLED STUDY; DRUG SCREENING; DRUG SYNTHESIS; IC 50; MYCOBACTERIOPHAGE; MYCOBACTERIUM TUBERCULOSIS; NONHUMAN; QUANTITATIVE STRUCTURE ACTIVITY RELATION;

ANTITUBERCULAR AGENTS; MICROBIAL SENSITIVITY TESTS; MORPHOLINES; MYCOBACTERIUM TUBERCULOSIS; QUANTITATIVE STRUCTURE-ACTIVITY RELATIONSHIP; SCHIFF BASES; TUBERCULOSIS;

EID: 67749101754     PISSN: 02235234     EISSN: 17683254     Source Type: Journal    
DOI: 10.1016/j.ejmech.2009.04.023     Document Type: Article

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