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European Journal of Medicinal Chemistry

Volumn 44, Issue 10, 2009, Pages 4211-4217

Design, synthesis and anticancer evaluation of novel tetrahydroquinoline derivatives containing sulfonamide moiety

(3) Ghorab, Mostafa M a Ragab, Fatma A b Hamed, Mostafa M c

a NATIONAL CENTER FOR RADIATION RESEARCH AND TECHNOLOGY (Egypt)

b CAIRO UNIVERSITY (Egypt)

c German University in Cairo (Egypt)

Author keywords

Anticancer; Carbonic anhydrase; Quinoline; Sulfonamide

Indexed keywords

ANTINEOPLASTIC AGENT; CARBONATE DEHYDRATASE INHIBITOR; DOXORUBICIN; N' (3 CYANO 4 METHYL 5,6,7,8 TETRAHYDROQUINOLIN 2 YL) N [4 [N (5 METHYLISOXAZOL 3 YL)SULFAMOYL]PHENYL]FORMIMIDAMIDE; N' (3 CYANO 4,7,7 TRIMETHYL 5 OXO 5,6,7,8 TETRAHYDROQUINOLIN 2 YL) N [4 [N (5 METHYLISOXAZOL 3 YL)SULFAMOYL]PHENYL]FORMIMIDAMIDE; PYRIMIDO[4,5 B]QUINOLINE; QUINOLINE DERIVATIVE; SULFONAMIDE; TETRAHYDROQUINOLINE DERIVATIVE; UNCLASSIFIED DRUG;

ANTINEOPLASTIC ACTIVITY; ARTICLE; CANCER CELL CULTURE; CELL STRAIN MCF 7; CRYSTAL STRUCTURE; DRUG CYTOTOXICITY; DRUG SYNTHESIS; ENZYME ACTIVE SITE; IN VITRO STUDY; MOLECULAR DOCKING; PROTON NUCLEAR MAGNETIC RESONANCE;

ANTINEOPLASTIC AGENTS; BREAST NEOPLASMS; CARBONIC ANHYDRASE II; CARBONIC ANHYDRASE INHIBITORS; CATALYTIC DOMAIN; CELL LINE, TUMOR; CELL SURVIVAL; DRUG SCREENING ASSAYS, ANTITUMOR; FEMALE; HUMANS; MODELS, MOLECULAR; PROTEIN BINDING; QUINOLINES; STRUCTURE-ACTIVITY RELATIONSHIP; SULFONAMIDES;

EID: 67651165007 PISSN: 02235234 EISSN: 17683254 Source Type: Journal
DOI: 10.1016/j.ejmech.2009.05.017 Document Type: Article

Times cited : (141)

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