Rapid identification of improved protein ligands using peptoid microarrays

Bioorganic and Medicinal Chemistry Letters

Volumn 19, Issue 14, 2009, Pages 3866-3869

  Lim, Hyun Suk ^a,b   Muralidhar Reddy, M ^a,b   Xiao, Xiangshu ^a,b   Wilson, Johnnie ^a,b   Wilson, Rosemary ^a,b   Connell, Steven ^a,b   Kodadek, Thomas ^a,b  

^a UNIVERSITY OF TEXAS SOUTHWESTERN MEDICAL CENTER   (United States)

^b UNIVERSITY OF TEXAS SOUTHWESTERN MEDICAL CENTER   (United States)

Author keywords

Click chemistry; Combinatorial chemistry; Library screening; Microarray; Peptoid

Indexed keywords

LIGAND; PEPTIDE LIBRARY; PEPTOID;

ARTICLE; BINDING AFFINITY; COMBINATORIAL CHEMISTRY; DISSOCIATION CONSTANT; DRUG ISOLATION; MICROARRAY ANALYSIS; PROTEIN BINDING;

LIGANDS; PEPTOIDS; PROTEIN ARRAY ANALYSIS; PROTEINS;

EID: 67649657944     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2009.03.153     Document Type: Article

References (21)

1. Shuker S.B., Hajduk P.J., Meadows R.P., and Fesik S.W. Science 274 (1996) 1531
2. Maly D.J., Choong I.C., and Ellman J.A. Proc. Natl. Acad. Sci. U.S.A. 97 (2000) 2419
3. Erlanson D.A., Wells J.A., and Braisted A.C. Ann. Rev. Biophys. Biomol. Struct. 33 (2004) 199
4. Profit A.A., Lee T.R., and Lawrence D.S. J. Am. Chem. Soc. 121 (1999) 280
5. Cussac D., Vidal M., Leprince C., Liu W.-q., Cornille F., Tiraboschi G., Roques B.P., and Garbay C. FASEB J. 13 (1999) 31
6. Kitov P.I., Shimizu H., Homans S.W., and Bundle D.R. J. Am. Chem. Soc. 125 (2003) 3284
7. Reddy M.M., Bachhawatt-Sikder K., and Kodadek T. Chem. Biol. 11 (2004) 1127
8. Jacobson K.A., Kirk K.L., Padgett W.L., and Daly J.W. Mol. Pharmacol. 29 (1986) 126
9. Jacobson K.A., Marr-Leisy D., Rosenkranz R.P., Verlander M.S., Melmon K.L., and Goodman M. J. Med. Chem. 26 (1983) 492
10. Verlander M.S., Jacobson K.A., Rosenkranz R.P., Melmon K.L., and Goodman M. Biopolymers 22 (1983) 531
11. Combs A.P., Kapoor T.M., Feng S., Chen J.K., Daude-Snow L.F., and Schreiber S.L. J. Am. Chem. Soc. 118 (1996) 287
12. Lawrence D.S. Biochim. Biophys. Acta 1754 (2005) 50
13. Agnew, H. D.; Rohde, R. D.; Millward, S. W.; Nag, A.; Yeo, W. S.; Hein, J. E.; Pitram, S. M.; Tariq, A. A.; Burns, V. M.; Krom, R. J.; Fokin, V. V.; Sharpless, K. B.; Heath, J. R. Angew Chem., Int. Ed., in press, doi:10.1002/anie.200900488.
14. Reddy M.M., and Kodadek T. Proc. Natl. Acad. Sci. U.S.A. 102 (2005) 12672
15. MacBeath G., Koehler A.N., and Schreiber S.L. J. Am. Chem. Soc. 121 (1999) 7967
16. Xiao X., Yu P., Lim H.-S., Sikder D., and Kodadek T. J. Comb. Chem. 9 (2007) 592
17. Xiao X., Yu P., Lim H.S., Sikder D., and Kodadek T. Angew. Chem., Int. Ed. Engl. 46 (2007) 2865
18. Kolb H.C., and Sharpless K.B. Drug Discovery Today 8 (2003) 1128
19. Liang P.H., Wang S.K., and Wong C.H. J. Am. Chem. Soc. 129 (2007) 11177
20. Figliozzi G.M., Goldsmith R., Ng S.C., Banville S.C., and Zuckermann R.N. Methods Enzymol. 267 (1996) 437
21. Alluri P.G., Reddy M.M., Bacchawat-Sikder K., Olivos H.J., and Kodadek T. J. Am. Chem. Soc. 125 (2003) 13995