Combinatorial target-guided ligand assembly: Identification of potent subtype-selective c-Src inhibitors

Proceedings of the National Academy of Sciences of the United States of America

Volumn 97, Issue 6, 2000, Pages 2419-2424

  Maly, Dustin J ^a   Choong, Ingrid C ^a   Ellman, Jonathan A ^a  

^a UNIVERSITY OF CALIFORNIA   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

LIGAND; PROTEIN KINASE INHIBITOR; PROTEIN KINASE P60;

ARTICLE; ENZYME INHIBITION; ENZYME PHOSPHORYLATION; ENZYME SUBSTRATE; LIGAND BINDING; MOLECULAR DYNAMICS; PRIORITY JOURNAL;

ADENOSINE TRIPHOSPHATE; COMBINATORIAL CHEMISTRY TECHNIQUES; DRUG DESIGN; INHIBITORY CONCENTRATION 50; LIGANDS; MAGNETIC RESONANCE SPECTROSCOPY; MODELS, CHEMICAL; PEPTIDE LIBRARY; PHOSPHORYLATION; PROTEIN BINDING; PROTEIN-TYROSINE KINASES;

EID: 0034646370     PISSN: 00278424     EISSN: None     Source Type: Journal    
DOI: 10.1073/pnas.97.6.2419     Document Type: Article

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