Combinatorial synthesis and biological evaluation of peptide-binding GPCR-targeted library

Bioorganic Chemistry

Volumn 37, Issue 3, 2009, Pages 90-95

  Lee, Ju Yeon ^a   Im, Isak ^a   Webb, Thomas R ^b   McGrath, Douglas ^c   Song, Mi Ryoung ^a   Kim, Yong Chul ^a  

^a Gwangju Institute of Science and Technology (GIST)   (South Korea)

^b ST JUDE CHILDREN S RESEARCH HOSPITAL   (United States)

^c RGo Bioscience LLC   (United States)

Author keywords

Benzodiazepine; Combinatorial synthesis; Melanocortin 4 receptors; Peptidomimetics

Indexed keywords

3 BENZYL 7 (4 FLUOROBENZYLOXY) 4 (4 METHOXYPHENETHYL) 4,5 DIHYDRO 1H BENZO[E][1,4]DIAZEPIN 2(3H) ONE; BENZODIAZEPINE DERIVATIVE; G PROTEIN COUPLED RECEPTOR; GLUTAMIC ACID; LYSINE; MELANOCORTIN 4 RECEPTOR; PHENYLALANINE; SERINE; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; CHO CELL; COMBINATORIAL LIBRARY; CONTROLLED STUDY; DRUG SCREENING; DRUG STRUCTURE; NONHUMAN; PEPTIDOMICS; PRIORITY JOURNAL; PROTEIN BINDING; RECEPTOR BLOCKING;

ANIMALS; AZEPINES; CELL LINE; CHO CELLS; COMBINATORIAL CHEMISTRY TECHNIQUES; CRICETINAE; CRICETULUS; DRUG DISCOVERY; PEPTIDES; RECEPTOR, MELANOCORTIN, TYPE 4;

HUMAN ECHOVIRUS 1;

EID: 67349119570     PISSN: 00452068     EISSN: 10902120     Source Type: Journal    
DOI: 10.1016/j.bioorg.2009.04.001     Document Type: Article

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